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Volumn , Issue , 2016, Pages 1046-1052

Potent and Selective Monoamine Oxidase-B Inhibitory Activity: Fluoro- vs. Trifluoromethyl-4-hydroxylated Chalcone Derivatives

(8) Mathew, Bijo a Mathew, Githa Elizabeth b Uçar, Gülberk c Baysal, Ipek c Suresh, Jerad d Mathew, Sincy b Haridas, Abitha b Jayaprakash, Venkatesan e

a Department of Pharmaceutical Chemistry (India)

b Grace College of Pharmacy (India)

c HACETTEPE UNIVERSITY (Turkey)

d MADRAS MEDICAL COLLEGE (India)

e BIRLA INSTITUTE OF TECHNOLOGY (India)

Author keywords

Chalcone; MAO A; MAO B; Molecular docking

Indexed keywords

(2) 1 (4 HYDROXYPHENYL) 3 [2 (TRIFLUOROMETHYL)PHENYL]PROP 2 EN 1 ONE; (2) 1 (4 HYDROXYPHENYL) 3 [4 (TRIFLUOROMETHYL)PHENYL]PROP 2 EN 1 ONE; (2) 3 (2 FLUOROPHENYL) 1 (4 HYDROXYPHENYL)PROP 2 EN 1 ONE; (2) 3 (3 FLUOROPHENYL) 1 (4 HYDROXYPHENYL)PROP 2 EN 1 ONE; (2) 3 (4 FLUOROPHENYL) 1 (4 HYDROXYPHENYL)PROP 2 EN 1 ONE; CHALCONE DERIVATIVE; LAZABEMIDE; MOCLOBEMIDE; MONOAMINE OXIDASE B INHIBITOR; SELEGILINE; UNCLASSIFIED DRUG;

ARTICLE; CLAISEN CONDENSATION; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; HYDROGEN BOND; MOLECULAR DOCKING; SELECTIVITY INDEX; STRUCTURE ACTIVITY RELATION;

EID: 84983032366 PISSN: 16121872 EISSN: 16121880 Source Type: Journal
DOI: 10.1002/cbdv.201500367 Document Type: Article

Times cited : (45)

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