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Bioorganic and Medicinal Chemistry Letters

Volumn 26, Issue 12, 2016, Pages 2806-2809

Synthesis and biological evaluation of novel 1,2,4-triazine derivatives bearing carbazole moiety as potent α-glucosidase inhibitors

(6) Wang, Guangcheng a Wang, Jing a He, Dianxiong a Li, Xin a Li, Juan a Peng, Zhiyun a

a JISHOU UNIVERSITY (China)

Author keywords

1,2,4 Triazine; Carbazole; Enzyme kinetic study; Molecular docking; Glucosidase inhibitor

Indexed keywords

1,2,4 TRIAZINE DERIVATIVE; ALPHA GLUCOSIDASE INHIBITOR; CARBAZOLE DERIVATIVE; 1,2,4-TRIAZINE; ALPHA GLUCOSIDASE; CARBAZOLE; GLYCOSIDASE INHIBITOR; TRIAZINE DERIVATIVE;

ANTIFUNGAL ACTIVITY; ANTINEOPLASTIC ACTIVITY; ANTIOXIDANT ACTIVITY; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG SCREENING; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; IC50; MOLECULAR DOCKING; NONHUMAN; PROTEIN NUCLEIC ACID INTERACTION; SACCHAROMYCES CEREVISIAE; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; ENZYMOLOGY; HUMAN; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ALPHA-GLUCOSIDASES; CARBAZOLES; DOSE-RESPONSE RELATIONSHIP, DRUG; GLYCOSIDE HYDROLASE INHIBITORS; HUMANS; MOLECULAR DOCKING SIMULATION; MOLECULAR STRUCTURE; SACCHAROMYCES CEREVISIAE; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZINES;

EID: 84971349504 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2016.04.071 Document Type: Article

Times cited : (65)

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