SCOPUS 정보 검색 플랫폼

Volumn 7, Issue 3, 2016, Pages 2322-2330

A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain

(12) Cox, Oakley B a,b,c Krojer, Tobias a Collins, Patrick c Monteiro, Octovia a,b Talon, Romain a Bradley, Anthony a Fedorov, Oleg a,b Amin, Jahangir d Marsden, Brian D a,e Spencer, John d Von Delft, Frank a,c,f Brennan, Paul E a,b

a UNIVERSITY OF OXFORD (United Kingdom)

b UNIVERSITY OF OXFORD (United Kingdom)

c DIAMOND LIGHT SOURCE LTD (United Kingdom)

d UNIVERSITY OF SUSSEX (United Kingdom)

e UNIVERSITY OF OXFORD (United Kingdom)

f UNIVERSITY OF JOHANNESBURG (South Africa)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACIDS; BINDING SITES; BINS; CRYSTALLOGRAPHY; DIAGNOSIS; LIGANDS;

ASPARAGINE RESIDUE; CHEMICAL BIOLOGY; COMPETITION ASSAYS; DISEASE PROGRESSION; FOLLOW UP; PARALLEL CHEMISTRY; PRIMARY FRAGMENTS; STRUCTURAL DATA;

X RAY CRYSTALLOGRAPHY;

EID: 84959450667 PISSN: 20416520 EISSN: 20416539 Source Type: Journal
DOI: 10.1039/c5sc03115j Document Type: Article

Times cited : (119)

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