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Angewandte Chemie - International Edition

Volumn 52, Issue 52, 2013, Pages 14055-14059

4-Acyl pyrroles: Mimicking acetylated lysines in histone code reading

(9) Lucas, Xavier a Wohlwend, Daniel a Hügle, Martin a Schmidtkunz, Karin a Gerhardt, Stefan a Schüle, Roland b Jung, Manfred a Einsle, Oliver a Günther, Stefan a

a UNIVERSITY OF FREIBURG (Germany)

b UNIVERSITY OF FREIBURG (Germany)

Author keywords

4 acyl pyrroles; bromodomain inhibition; drug discovery; epigenetics; virtual screening

Indexed keywords

4-ACYL PYRROLES; ANTI-CANCER AGENTS; ANTI-INFLAMMATORIES; ANTI-PROLIFERATIVE ACTIVITIES; DRUG DISCOVERY; EPIGENETICS; PYRROLE DERIVATIVES; VIRTUAL SCREENING;

AMINO ACIDS; ANTIVIRAL AGENTS; CELL CULTURE; DRUG PRODUCTS; PROTEINS;

POTASSIUM COMPOUNDS;

HISTONE; LYSINE; PYRROLE DERIVATIVE;

4-ACYL PYRROLES; ACETYLATION; ARTICLE; BROMODOMAIN INHIBITION; DRUG DEVELOPMENT; EPIGENETICS; GENETICS; HISTONE CODE; HUMAN; METABOLISM; VIRTUAL SCREENING;

4-ACYL PYRROLES; BROMODOMAIN INHIBITION; DRUG DISCOVERY; EPIGENETICS; VIRTUAL SCREENING;

ACETYLATION; HISTONE CODE; HISTONES; HUMANS; LYSINE; PYRROLES;

EID: 84890680254 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201307652 Document Type: Article

Times cited : (94)

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