The prediction of the palatability of orally disintegrating tablets by an electronic gustatory system

International Journal of Pharmaceutics

Volumn 493, Issue 1-2, 2015, Pages 305-312

  Nakamura, Hideshi ^a,b   Uchida, Shinya ^a   Sugiura, Takeshi ^b   Namiki, Noriyuki ^a  

^a UNIVERSITY OF SHIZUOKA   (Japan)

^b National Cerebral and Cardiovascular Center 30602   (Japan)

Author keywords

Amlodipine; Electronic gustatory system; Famotidine; Orally disintegrating tablet; Taste masking; Visual analogue scale

Indexed keywords

AMLODIPINE; ETHYL CELLULOSE; FAMOTIDINE; MAGNESIUM STEARATE; MANNITOL; MENTHOL; PEPPERMINT; SILICIC ACID; SWEETENING AGENT; TABLET;

ADULT; ARTICLE; CONTROLLED STUDY; CROSSOVER PROCEDURE; DRUG GRANULE; FEMALE; GUSTATORY SYSTEM; HUMAN; HUMAN EXPERIMENT; MALE; NORMAL HUMAN; ORGANOLEPTIC PROPERTY; PALATABILITY; PREDICTION; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RANDOMIZED CONTROLLED TRIAL; SINGLE BLIND PROCEDURE; TABLET DISINTEGRATION; TABLET FORMULATION; VISUAL ANALOG SCALE; YOUNG ADULT; ELECTRICAL EQUIPMENT; ORAL DRUG ADMINISTRATION; TABLET; TASTE;

ADMINISTRATION, ORAL; ADULT; AMLODIPINE; ELECTRICAL EQUIPMENT AND SUPPLIES; FAMOTIDINE; FEMALE; HUMANS; MALE; TABLETS; TASTE; TASTE PERCEPTION; YOUNG ADULT;

EID: 84938824971     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2015.07.056     Document Type: Article

References (32)

1. Alpha, M.O.S., 2004. Astree electrochemical sensor technology. Technical note T-SA.S-S04.
2. A.M. Carlsson Assessment of chronic pain. I. Aspects of the reliability and validity of the visual analogue scale Pain 16 1983 87 101
3. R.K. Chang, X. Guo, B.A. Burnside, and R.A. Couch Fast-dissolving tablets Pharm. Technol. 6 2000 52 58
4. C. Eckert, C. Lutz, J. Breitkreutz, and K. Woertz Quality control of oral herbal products by an electronic tongue - case study on sage lozenges Sens. Actuators B Chem. 156 2011 204 212
5. FDA Orally Disintegrating Tablets 2008 Guidance for Industry Rockvill, MD 2008
6. Y. Gao, F.D. Cui, Y. Guan, L. Yang, Y.S. Wang, and L.N. Zhang Preparation of roxithromycin-polymeric microspheres by the emulsion solvent diffusion method for taste masking Int. J. Pharm. 318 2006 62 69
7. H. Hames, J.A. Seabrook, D. Matsui, M.J. Rieder, and G.I. Joubert A palatability study of a flavored dexamethasone preparation versus prednisolone liquid in children Can. J. Clin. Pharmacol. 15 2008 e95 e98
8. Y. Hashimoto, C. Matsunaga, E. Tokuyama, E. Tsuji, T. Uchida, and H. Okada The quantitative prediction of bitterness-suppressing effect of sweetness on the bitterness of famotidine by sweetness-responsive sensor Chem. Pharm. Bull. 55 2007 739 746
9. Y. Inoue, H. Shimazaki, I. Murata, M. Kimura, and I. Kanamoto Study of the physicochemical properties of tulobuterol dry syrups using taste and smell sensors Chem. Pharm. Bull. 60 2012 442 448
10. M. Ito, K. Ikehama, K. Yoshuida, T. Haraguchi, M. Yoshida, K. Wada, and T. Uchida Bitterness prediction of H1-antihistamines and prediction of masking effects of artificial sweeteners using an electronic tongue Int. J. Pharm. 441 2013 121 127
11. K.L. Julie, P.R. Joseph, H. Ondrej, H.W. Jeffrey, and D.P. Vanik Evaluation of a taste sensor instrument (electronic tongue) for use in formulation development Int. J. Pharm. 367 2009 65 72
12. A. Lieberman, L. Lachman, and J.B. Schwartz 2nd ed. Pharmaceutical Dosage Forms: Tablets 1 1989 Marcel Dekker New York Chapter 2
13. M. Maniruzzaman, and D. Douroumis An in-vitro-in-vivo taste assessment of bitter drug: comparative electronic tongues study J. Pharm. Pharmacol. 67 2014 43 55
14. R. Matsui, S. Uchida, and N. Namiki Combination effect of physical and gustatory taste masking for propiverine hydrochloride orally disintegrating tablets on palatability Chem. Pharm. Bull. 38 2015 17 22
15. Y. Nakano, A. Maeda, S. Uchida, and N. Namiki Preparation and evaluation of unpleasant taste-masked pioglitazone orally disintegrating tablets Int. J. Pharm. 446 2013 160 165
16. Y. Okuda, Y. Irisawa, K. Okimoto, T. Osawa, and S. Yamashita A new formulation for orally disintegrating tablets using a suspension spray-coating method Int. J. Pharm. 382 2009 80 87
17. Y. Okuda, Y. Irisawa, K. Okimoto, T. Osawa, and S. Yamashita Further improvement of orally disintegrating tablets using micronized ethylcellulose Int. J. Pharm. 423 2012 351 359
18. Y. Okuda, Y. Okamoto, Y. Irisawa, K. Okimoto, T. Osawa, and S. Yamashita Formulation design for orally disintegrating tablets containing enteric-coated particles Chem. Pharm. Bull. 62 2014 407 414
19. M. Pein, C. Eckert, M. Preis, and J. Breitkreutz New protocol for αAstree electronic tongue enabling full performance qualification according to ICH Q2 J. Pharm. Biomed. Anal. 83 2013 157 163
20. O. Rachid, F.E. Simons, M. Rawas-Qalaji, and K.J. Simons An electronic tongue: evaluation of the masking efficacy of sweetening and/or flavoring agents on the bitter taste of epinephrine AAPS PharmSciTech 11 2010 550 557
21. G. Sandri, M.C. Bonferoni, F. Ferrari, S. Rossi, and C. Camella Differentiating factors between oral fast-dissolving technologies Am. J. Drug Deriv. 4 2006 249 262
22. B.A. Shishu, and T. Singh Preparation of tablets rapidly disintegrating in saliva containing bitter taste-masked granules by compression method Indian J. Pharm. Sci. 69 2007 80 84
23. J. Sjovall, A. Fogh, B. Huitfeldt, G. Karlsson, and O. Nylen Methods for evaluating the taste of paediatric formulations in children: a comparison between the facial hedonic method and the patients' own spontaneous verbal judgement Eur. J. Pediatr. 141 1984 243 247
24. T. Sugiura, S. Uchida, and N. Namiki Taste-masking effect of physical and organoleptic methods on peppermint-scented orally disintegrating tablet of famotidine based on suspension spray-coating method Chem. Pharm. Bull. 60 2012 315 319
25. H. Suzuki, H. Onishi, Y. Takahashi, M. Iwata, and Y. Machida Development of oral acetaminophen chewable tablets with inhibited bitter taste Int. J. Pharm. 251 2003 123 132
26. E. Tokuyama, C. Matsunaga, K. Yoshida, J. Mifsud, T. Irie, M. Yoshida, and T. Uchida Famotidine orally disintegrating tablets bitterness comparison of original and generic products Chem. Pharm. Bull. 57 2009 382 387
27. M.E. Wewers, and N.K. Lowe A critical review of visual analogue scales in the measurement of clinical phenomena Res. Nurs. Health 13 1990 227 236
28. R.P. William, and K.G. Tapash Orally disintegrating tablets Pharm. Technol. 2005
29. K. Woertz, C. Tissen, P. Kleinebudde, and J. Breitkreutz Performance qualification of an electronic tongue based on ICH guideline Q2 J. Pharm. Biomed. Anal. 51 2010 497 506
30. K. Woertz, C. Tissen, P. Kleinebudde, and J. Breitkreutz A comparative study on two electronic tongues for pharmaceutical formulation development J. Pharm. Biomed. Anal. 55 2011 272 281
31. K. Woertz, C. Tissen, P. Kleinebudde, and J. Breitkreutz Taste sensing systems (electronic tongues) for pharmaceutical applications Int. J. Pharm. 417 2011 256 271
32. J.Y. Zheng, and M.P. Keeney Taste masking analysis in pharmaceutical formulation development using an electronic tongue Int. J. Pharm. 310 2006 118 124