Human SIRT3 tripeptidic inhibitors containing Nε-thioacetyl-lysine

Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 17, 2015, Pages 3481-3487

  Chen, Bing ^a   Wang, Juan ^a   Huang, Yajun ^a   Zheng, Weiping ^a  

^a JIANGSU UNIVERSITY   (China)

Author keywords

Deacetylation; Deacylation; Inhibitor; N thioacetyl lysine; SIRT3; Sirtuin

Indexed keywords

HYDROLASE INHIBITOR; LYSINE DERIVATIVE; N EPSILON THIOACETYL LYSINE; SIRTUIN 1; SIRTUIN 2; SIRTUIN 3; UNCLASSIFIED DRUG; LYSINE; N(EPSILON)-THIOACETYLLYSINE; SIRT3 PROTEIN, HUMAN; SIRTUIN;

ARTICLE; CATALYSIS; DEACETYLATION; DEACYLATION; ENZYME INHIBITION; ENZYME SPECIFICITY; HUMAN; MASS SPECTROMETRY; PEPTIDE SYNTHESIS; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; SOLID PHASE PEPTIDE SYNTHESIS; ANALOGS AND DERIVATIVES; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; GENETICS; METABOLISM;

CATALYSIS; HUMANS; LYSINE; MODELS, MOLECULAR; SIRTUIN 3; SIRTUINS;

EID: 84938289896     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2015.07.008     Document Type: Article

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