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Volumn 1, Issue 3, 2010, Pages 233-238

Discovery of potent, proteolytically stable, and cell permeable human sirtuin peptidomimetic inhibitors containing Nε-thioacetyl- lysine

(5) Hirsch, Brett M a Gallo, Caroline A a Du, Zhanwen b Wang, Zhenghe b Zheng, Weiping a

a UNIVERSITY OF AKRON (United States)

b CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AGK 2; EX 527; HYDROLASE INHIBITOR; LYSINE DERIVATIVE; N EPSILON THIOACETYLLYSINE; PEPTIDOMIMETIC AGENT; SIRTUIN 1; SIRTUIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CELL MEMBRANE PERMEABILITY; DRUG IDENTIFICATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; IN VITRO STUDY; IN VIVO STUDY; MOLECULAR WEIGHT; PRIORITY JOURNAL; PROTEIN DEGRADATION; STRUCTURE ACTIVITY RELATION;

EID: 78650107007 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c0md00089b Document Type: Article

Times cited : (21)

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