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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 10, 2015, Pages 2100-2105

Benzo-fused lactams from a diversity-oriented synthesis (DOS) library as inhibitors of scavenger receptor BI (SR-BI)-mediated lipid uptake

(14) Dockendorff, Chris a,b Faloon, Patrick W a Pu, Jun a Yu, Miao c Johnston, Stephen a Bennion, Melissa a Penman, Marsha c Nieland, Thomas J F c Dandapani, Sivaraman a Perez, José R a Munoz, Benito a Palmer, Michelle A a Schreiber, Stuart L a,d Krieger, Monty c

a BROAD INSTITUTE OF MIT AND HARVARD (United States)

b Marquette University (United States)

c MASSACHUSETTS INSTITUTE OF TECHNOLOGY (United States)

d HOWARD HUGHES MEDICAL INSTITUTE (United States)

Author keywords

Cholesterol transport; DOS macrocycle; HDL receptor; ML312; SR BI inhibitor

Indexed keywords

CD36 ANTIGEN; LACTAM;

ANIMAL; ANTAGONISTS AND INHIBITORS; CHEMISTRY; HUMAN; LIPID METABOLISM; PHYSIOLOGY; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIGENS, CD36; HUMANS; LACTAMS; LIPID METABOLISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84930004990 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.03.073 Document Type: Article

Times cited : (14)

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