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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 22, 2011, Pages 6852-6855

Discovery of highly potent small molecule Hepatitis C Virus entry inhibitors

(8) Mittapalli, Gopi Kumar a Jackson, Andrew a Zhao, Fang a Lee, Haekyung a Chow, Stephine a McKelvy, Jeffrey a Wong Staal, Flossie a MacDonald, James E a

a iTherX Pharmaceuticals Inc (United States)

Author keywords

Entry inhibitors; HCVcc; Hepatitis C Virus; Pharmacokinetics; Tetrahydrocarbazoles

Indexed keywords

1,2,3,4 TETRAHYDROCARBAZOLE DERIVATIVE; 2 AMINO PYRIMIDINE; 4,6 DIMETHOXY 2 AMINO PYRIMIDINE; ANTIVIRUS AGENT; CARBOXYLIC ACID; IMIDAZOLE; MORPHOLINE; PIPERIDINE DERIVATIVE; PURINE; PYRIMIDINE DERIVATIVE; RIMCAZOLE; SULFONAMIDE; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; DRUG BIOAVAILABILITY; DRUG CLEARANCE; DRUG HALF LIFE; DRUG POTENCY; DRUG SCREENING; DRUG STABILITY; GENOTYPE; HEPATITIS C VIRUS; IC 50; MASS SPECTROMETRY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; VIRUS ENTRY;

ANIMALS; ANTIVIRAL AGENTS; DRUG DISCOVERY; HEPACIVIRUS; HEPATITIS C; HUMANS; INHIBITORY CONCENTRATION 50; RATS; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS INTERNALIZATION;

HEPATITIS C VIRUS;

EID: 80054741500 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.09.019 Document Type: Article

Times cited : (21)

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