SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 15, 2012, Pages 4955-4961

Discovery of ITX 4520: A highly potent orally bioavailable hepatitis C virus entry inhibitor

(12) Mittapalli, Gopi Kumar a Zhao, Fang a Jackson, Andrew a Gao, Hongfeng a Lee, Haekyung a Chow, Stephine a Kaur, Maninder Pal a Nguyen, Natalie a Zamboni, Robert a McKelvy, Jeffrey a Wong Staal, Flossie a MacDonald, James E a

a iTherX Pharmaceuticals Inc (United States)

Author keywords

Bioisostere; Entry inhibitors; Hepatitis C virus; Oral bioavailability; Scavenger receptor B 1

Indexed keywords

ANTIVIRUS AGENT; ITX 4520; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; DRUG BIOAVAILABILITY; DRUG EFFECT; DRUG EFFICACY; DRUG HALF LIFE; DRUG IDENTIFICATION; DRUG MECHANISM; DRUG POTENCY; DRUG TOLERABILITY; HEPATITIS C VIRUS; NONHUMAN; RAT; VIRUS ENTRY;

ADMINISTRATION, ORAL; ANIMALS; ANTIVIRAL AGENTS; BIOLOGICAL AVAILABILITY; CARBAZOLES; DOGS; DRUG EVALUATION, PRECLINICAL; HALF-LIFE; HEPACIVIRUS; HUMANS; MICROSOMES; OXADIAZOLES; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS INTERNALIZATION;

CANIS FAMILIARIS; HEPATITIS C VIRUS; RATTUS;

EID: 84863981346 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.06.038 Document Type: Article

Times cited : (21)

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