Modulation of particle size and molecular interactions by sonoprecipitation method for enhancing dissolution rate of poorly water-soluble drug

Ultrasonics Sonochemistry

Volumn 24, Issue , 2015, Pages 256-263

  Tran, Thao Truong Dinh ^a   Tran, Kiet Anh ^a   Tran, Phuong Ha Lien ^a  

^a INTERNATIONAL UNIVERSITY   (Viet Nam)

Author keywords

Crystallinity; Curcumin; Molecular interactions; Polymeric nanoparticles; Ultrasonication

Indexed keywords

CONTROLLED DRUG DELIVERY; DISSOLUTION; MOLECULAR INTERACTIONS; MOLECULAR STRUCTURE; NANOPARTICLES; PARTICLE SIZE; POLYMERS;

CRYSTALLINITIES; CURCUMIN; DISSOLUTION RATES; DRUG DISSOLUTION RATES; DRUG-POLYMER INTERACTION; POLYMERIC NANOPARTICLES; POORLY WATER-SOLUBLE DRUGS; ULTRA-SONICATION;

DRUG INTERACTIONS;

CURCUMIN; HYDROXYL GROUP; NANOPARTICLE; POLYMER; DRUG CARRIER;

ARTICLE; CRYSTALLIZATION; DRUG DELIVERY SYSTEM; DRUG RELEASE; DRUG SOLUBILITY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HYDROGEN BOND; INFRARED SPECTROSCOPY; MODULATION; MOLECULAR INTERACTION; MOLECULAR WEIGHT; NANOENCAPSULATION; PARTICLE SIZE; PHYSICAL CHEMISTRY; POLYMERIZATION; PRECIPITATION; PRIORITY JOURNAL; SONOPRECIPITATION METHOD; TRANSMISSION ELECTRON MICROSCOPY; ULTRASOUND; X RAY POWDER DIFFRACTION; CHEMISTRY; PROCEDURES; SOLUBILITY;

CHEMICAL PRECIPITATION; CURCUMIN; DRUG CARRIERS; DRUG LIBERATION; NANOPARTICLES; PARTICLE SIZE; SOLUBILITY; SONICATION;

EID: 84921528029     PISSN: 13504177     EISSN: 18732828     Source Type: Journal    
DOI: 10.1016/j.ultsonch.2014.11.020     Document Type: Article

References (29)

1. T. Vasconcelos, B. Sarmento, P. Costa, Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs, Drug Discov. Today 12 (2007) 1068-1075.
2. N. Ahuja, O.P. Katare, B. Singh, Studies on dissolution enhancement and mathematical modeling of drug release of a poorly water-soluble drug using water-soluble carriers, Eur. J. Pharm. Biopharm. 65 (2007) 26-38.
3. N.S. Ha, T.T.-D. Tran, P.H.-L. Tran, J.-B. Park, B.-J. Lee, Dissolution-enhancing mechanism of alkalizers in poloxamer-based solid dispersions and physical mixtures containing poorly water-soluble valsartan, Chem. Pharm. Bull. 59 (2011) 844-850.
4. P.H.L. Tran, T.T.D. Tran, J.B. Park, B.-J. Lee, Controlled release systems containing solid dispersions: strategies and mechanisms, Pharm. Res. 28 (2011) 2353-2378.
5. P.H.L. Tran, T.T.-D. Tran, K.H. Lee, D.J. Kim, B.J. Lee, Dissolution-modulating mechanism of pH modifiers in solid dispersion containing weakly acidic or basic drugs with poor water solubility, Expert Opin. Drug Deliv. 7 (2010) 647-661.
6. D. Liu, H. Xu, B. Tian, K. Yuan, H. Pan, S. Ma, X. Yang, W. Pan, Fabrication of carvedilol nanosuspensions through the anti-solvent precipitation-ultrasonication method for the improvement of dissolution rate and oral bioavailability, AAPS PharmSciTech 13 (2012) 295-304.
7. T.T.-D. Tran, P.H.-L. Tran, B.-J. Lee, Dissolution-modulating mechanism of alkalizers and polymers in a nanoemulsifying solid dispersion containing ionizable and poorly water-soluble drug, Eur. J. Pharm. Biopharm. 72 (2009) 83-90.
8. T.T.-D. Tran, P.H.L. Tran, J. Lim, J.B. Park, S.K. Choi, B.J. Lee, Physicochemical principles of controlled release solid dispersion containing a poorly water-soluble drug, Ther. Deliv. 1 (2010) 51-62.
9. P.H.-L. Tran, T.T.-D. Tran, B.-J. Lee, Enhanced solubility and modified release of poorly water-soluble drugs via self-assembled gelatin-oleic acid nanoparticles, Int. J. Pharm. 455 (2013) 235-240.
10. A.A. Thorat, S.V. Dalvi, Liquid antisolvent precipitation and stabilization of nanoparticles of poorly water soluble drugs in aqueous suspensions: recent developments and future perspective, Chem. Eng. J. 181-182 (2012) 1-34.
11. R.S. Dhumal, S.V. Biradar, S. Yamamura, A.R. Paradkar, P. York, Preparation of amorphous cefuroxime axetil nanoparticles by sonoprecipitation for enhancement of bioavailability, Eur. J. Pharm. Biopharm. 70 (2008) 109-115.
12. S.V. Dalvi, R.N. Dave, Analysis of nucleation kinetics of poorly water-soluble drugs in presence of ultrasound and hydroxypropyl methyl cellulose during antisolvent precipitation, Int. J. Pharm. 387 (2010) 172-179.
13. S.V. Dalvi, R.N. Dave, Controlling particle size of a poorly water-soluble drug using ultrasound and stabilizers in antisolvent precipitation, Ind. Eng. Chem. Res. 48 (2009) 7581-7593.
14. D. Xia, P. Quan, H. Piao, H. Piao, S. Sun, Y. Yin, F. Cui, Preparation of stable nitrendipine nanosuspensions using the precipitation-ultrasonication method for enhancement of dissolution and oral bioavailability, Eur. J. Pharm. Sci. 40 (2010) 325-334.
15. T.T.-D. Tran, P.H.-L. Tran, M.N.U. Nguyen, K.T.M. Tran, M.N. Pham, P.C. Tran, T.V. Vo, Amorphous isradipine nanosuspension by the sonoprecipitation method, Int. J. Pharm. 474 (2014) 146-150.
16. P.H.L. Tran, H.T.T. Tran, B.-J. Lee, Modulation of microenvironmental pH and crystallinity of ionizable telmisartan using alkalizers in solid dispersions for controlled release, J. Control. Release 129 (2008) 59-65.
17. T.T.-D. Tran, P.H.-L. Tran, H.-G. Choi, H.-K. Han, B.-J. Lee, The roles of acidifiers in solid dispersions and physical mixtures, Int. J. Pharm. 384 (2010) 60-66.
18. T.T.-D. Tran, P.H.-L. Tran, T.N. Khanh, T.V. Van, B.-J. Lee, Solubilization of poorly water-soluble drugs using solid dispersions, Recent Pat. Drug Delivery Formulation 7 (2013) 122-133.
19. M.H. Ucisik, S. Küpcü, B. Schuster, U.B. Sleytr, Characterization of CurcuEmulsomes: nanoformulation for enhanced solubility and delivery of curcumin, J. Nanobiotechnol. 11 (2013) 1-13.
20. Z. Zheng, X. Zhang, D. Carbo, C. Clark, C. Nathan, Y. Lvov, Sonication-assisted synthesis of polyelectrolyte-coated curcumin nanoparticles, Langmuir 26 (2010) 7679-7681.
21. C. Moorthi, K. Kathiresan, Fabrication of highly stable sonication assisted curcumin nanocrystals by nanoprecipitation method, Drug Invention Today 5 (2013) 66-69.
22. Y. Dong, W.K. Ng, S. Shen, S. Kim, R.B. Tan, Preparation and characterization of spironolactone nanoparticles by antisolvent precipitation, Int. J. Pharm. 375 (2009) 84-88.
23. J. Hu, K.P. Johnston, R.O. Williams Iii, Spray freezing into liquid (SFL) particle engineering technology to enhance dissolution of poorly water soluble drugs: organic solvent versus organic/aqueous co-solvent systems, Eur. J. Pharm. Sci. 20 (2003) 295-303.
24. S.M. Wong, I.W. Kellaway, S. Murdan, Enhancement of the dissolution rate and oral absorption of a poorly water soluble drug by formation of surfactant-containing microparticles, Int. J. Pharm. 317 (2006) 61-68.
25. V. Teeranachaideekul, V.B. Junyaprasert, E.B. Souto, R.H. Müller, Development of ascorbyl palmitate nanocrystals applying the nanosuspension technology, Int. J. Pharm. 354 (2008) 227-234.
26. B. Li, S. Konecke, L.A. Wegiel, L.S. Taylor, K.J. Edgar, Both solubility and chemical stability of curcumin are enhanced by solid dispersion in cellulose derivative matrices, Carbohydr. Polym. 98 (2013) 1108-1116.
27. M.K. Modasiya, V.M. Patel, Studies on solubility of curcumin, Int. J. Pharm. Life Sci. 3 (2012) 1490-1497.
28. P.R.K. Mohan, G. Sreelakshmi, C.V. Muraleedharan, R. Joseph, Water soluble complexes of curcumin with cyclodextrins: characterization by FT-Raman spectroscopy, Vib. Spectrosc. 62 (2012) 77-84.
29. N. Kaewnopparat, S. Kaewnopparat, A. Jangwang, D. Maneenaun, T. Chuchome, P. Panichayupakaranant, Increased solubility, dissolution and physicochemical studies of curcuminpolyvinylpyrrolidone K-30 solid dispersions world academy of science, Eng. Technol. 31 (2009) 225-230.