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Bioorganic and Medicinal Chemistry

Volumn 22, Issue 15, 2014, Pages 3989-3993

Potential C-terminal-domain inhibitors of heat shock protein 90 derived from a C-terminal peptide helix

(3) Gavenonis, Jason a Jonas, Nicholas E a Kritzer, Joshua A a

a TUFTS UNIVERSITY (United States)

Author keywords

Hsp90; Molecular chaperones; Peptides; Protein protein interactions; Stapled helices

Indexed keywords

COUMAMYCIN A1; GELDANAMYCIN; HEAT SHOCK PROTEIN 90; HEAT SHOCK PROTEIN 90 INHIBITOR; NOVOBIOCIN; ADENOSINE TRIPHOSPHATE; PEPTIDE; PROTEIN BINDING;

AMINO ACID SUBSTITUTION; AMINO TERMINAL SEQUENCE; ARTICLE; BINDING SITE; CARBOXY TERMINAL SEQUENCE; CELL DISRUPTION; CELL MEMBRANE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG EFFECT; HUMAN; HUMAN CELL; IC 50; LC 50; POLARIZATION; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN DOMAIN; PROTEIN SYNTHESIS INHIBITION; STRUCTURE ACTIVITY RELATION; AMINO ACID SEQUENCE; ANTAGONISTS AND INHIBITORS; CHEMISTRY; METABOLISM; MOLECULAR GENETICS; PROTEIN SECONDARY STRUCTURE; SYNTHESIS;

ADENOSINE TRIPHOSPHATE; AMINO ACID SEQUENCE; BINDING SITES; HSP90 HEAT-SHOCK PROTEINS; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEIN BINDING; PROTEIN STRUCTURE, SECONDARY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84905111138 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2014.06.006 Document Type: Article

Times cited : (14)

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