Pharmacological profiling of the TRPV3 channel in recombinant and native assays

British Journal of Pharmacology

Volumn 171, Issue 10, 2014, Pages 2631-2644

  Grubisha, Olivera ^a   Mogg, Adrian J ^a   Sorge, Jessica L ^a   Ball, Laura Jayne ^a   Sanger, Helen ^a   Ruble, Cara L A ^a   Folly, Elizabeth A ^a   Ursu, Daniel ^a   Broad, Lisa M ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

FLIPR; Mouse 308 keratinocytes; TRP channel; TRPV3

Indexed keywords

ARACHIDONIC ACID; LINOLEIC ACID; VANILLOID RECEPTOR 3; AGENTS AFFECTING WATER, MOLECULE OR ION TRANSPORT; LIGAND; RECOMBINANT PROTEIN; TRPV3 PROTEIN, HUMAN; TRPV3 PROTEIN, MOUSE; TRPV3 PROTEIN, RAT; VANILLOID RECEPTOR;

ANIMAL CELL; ARTICLE; CALCIUM SIGNALING; CELL ASSAY; CONTROLLED STUDY; EMBRYO; FLUORESCENCE IMAGING; HUMAN; HUMAN CELL; KERATINOCYTE; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROCESS DEVELOPMENT; PROTEIN DETERMINATION; PROTEIN FUNCTION; SEQUENCE ANALYSIS; ANIMAL; COMPARATIVE STUDY; DOSE RESPONSE; DRUG EFFECTS; GENETIC TRANSFECTION; GENETICS; HEK293 CELL LINE; METABOLISM; RAT;

ANIMALS; CALCIUM SIGNALING; DOSE-RESPONSE RELATIONSHIP, DRUG; HEK293 CELLS; HUMANS; LIGANDS; MEMBRANE TRANSPORT MODULATORS; MICE; RATS; RECOMBINANT PROTEINS; TRANSFECTION; TRPV CATION CHANNELS;

EID: 84900824791     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/bph.12303     Document Type: Article

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