Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 10, 2012, Pages 3535-3539

  Ortar, Giorgio ^a   Morera, Ludovica ^a   Schiano Moriello, Aniello ^b   Morera, Enrico ^a   Nalli, Marianna ^a   Di Marzo, Vincenzo ^c   De Petrocellis, Luciano ^b  

^a SAPIENZA UNIVERSITY OF ROME   (Italy)

^b CNR   (Italy)

^c CNR   (Italy)

Author keywords

3 Amino p cymene derivatives; p Cymene 3 carboxylic acid derivatives; Thermo TRP channels; TRPA1; TRPM8; TRPV3; Tymol derivatives

Indexed keywords

3 AMINO 4 CYMENE DERIVATIVE; 4 CYMENE 3 CARBOXYLIC ACID DERIVATIVE; BORNEOL; CAMPHOR; CARVACROL; CARVEOL; CINEOLE; GERANIOL; LIGAND; LINALOOL; MENTHOL; RECEPTOR SUBTYPE; TERPENE DERIVATIVE; THERMO TRANSIENT RECEPTOR POTENTIAL CHANNEL; THYMOL; THYMOL DERIVATIVE; TRANSIENT RECEPTOR POTENTIAL CHANNEL; UNCLASSIFIED DRUG; VANILLOID RECEPTOR 1; VANILLOID RECEPTOR 3;

ANIMAL CELL; ARTICLE; CELL STRAIN HEK293; CHEMICAL STRUCTURE; DRUG SELECTIVITY; HUMAN; NONHUMAN; OREGANO; RAT; SYNTHESIS; THYME;

ANIMALS; CELL LINE; HUMANS; RATS; THYMOL; TRANSIENT RECEPTOR POTENTIAL CHANNELS;

EID: 84860478788     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.03.055     Document Type: Article

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