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Volumn 22, Issue 1, 2014, Pages 393-397

From NMDA receptor antagonists to discovery of selective σ2 receptor ligands

(9) Gitto, Rosaria a De Luca, Laura a Ferro, Stefania a Scala, Angela b Ronsisvalle, Simone c Parenti, Carmela c Prezzavento, Orazio c Buemi, Maria Rosa a Chimirri, Alba a

a UNIVERSITY OF MESSINA (Italy)

b Dipartimento di Scienze della Terra (Italy)

c UNIVERSITY OF CATANIA (Italy)

Author keywords

GluN2B NMDA; Glutamate; Ifenprodil; Indoles; Sigma receptor

Indexed keywords

1 (5 HYDROXY 1H INDOL 3 YL) 2 (4 HYDROXY 4 PHENYLPIPERIDIN 1 YL)ETHANONE; 1 (5 HYDROXY 1H INDOL 3 YL) 2 (4 PHENYLPIPERIDIN 1 YL)ETHANONE; 1 (5 METHOXY 1H INDOL 3 YL) 2 (4 PHENYLPIPERIDIN 1 YL)ETHANONE; 1 [2 (5 HYDROXY 1H INDOL 3 YL) 2 OXOETHYL] 4 PHENYLPIPERIDINE 4 CARBONITRILE; 1 [2 (5 METHOXY 1H INDOL 3 YL) 2 OXOETHYL] 4 PHENYLPIPERIDINE 4 CARBONITRILE; 2 (4 ACETYL 4 PHENYLPIPERIDIN 1 YL) 1 (5 METHOXY 1H INDOLE 3 YL)ETHANONE; 2 (4 ACETYL 4 PHENYLPIPERIDINE 1 YL) 1 (5 HYDROXY 1H INDOL 3YL)ETHANONE; 2 (4 HYDROXY 4 PHENYLPIPERIDIN 1 YL) 1 (5 METHOXY 1H INDOL 3 YL)ETHANONE; 2 [4 (4 BROMOPHENYL) 4 HYDROXYPIPERIDIN 1 YL] 1 (5 HYDROXY 1H INDOL 3YL)ETHANONE; 2 [4 (4 BROMOPHENYL) 4 HYDROXYPIPERIDIN 1 YL] 1 (5 METHOXY 1H INDOL 3 YL)ETHANONE; 2 [4 (4 CHLOROPHENYL) 4 HYDROXYPIPERIDIN 1 YL] 1 (5 HYDROXY 1H INDOL 3YL)ETHANONE; 2 [4 (4 CHLOROPHENYL) 4 HYDROXYPIPERIDIN 1 YL] 1 (5 METHOXY 1H INDOL 3 YL)ETHANONE; 2 CHLORO 1 (5 HYDROXY 1H INDOL 3 YL)ETHANONE; 2 CHLORO 1 (5 METHOXY 1H INDOL 3 YL)ETHANONE; IFENPRODIL; INDOLE DERIVATIVE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR 2B; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; SIGMA OPIATE RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; LIGAND BINDING; RADIOASSAY; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

GLUN2B/NMDA; GLUTAMATE; IFENPRODIL; INDOLES; SIGMA RECEPTOR;

BINDING SITES; GLUTAMIC ACID; RECEPTORS, N-METHYL-D-ASPARTATE; RECEPTORS, SIGMA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84891493554 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2013.11.014 Document Type: Article

Times cited : (13)

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