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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 1, 2014, Pages 245-248

Novel pyrazole integrated 1,3,4-oxadiazoles: Synthesis, characterization and antimicrobial evaluation

(5) Ningaiah, Srikantamurthy a Bhadraiah, Umesha K a Doddaramappa, Shridevi D b Keshavamurthy, Shubakara a Javarasetty, Chethan b

a UNIVERSITY OF MYSORE (India)

b UNIVERSITY OF MYSORE (India)

Author keywords

1,3,4 Oxadiazoles; Antimicrobial activity; Chloramine T; Minimum inhibitory concentration (MIC); Pyrazole

Indexed keywords

1,3,4 OXADIAZOLE DERIVATIVE; ANTIINFECTIVE AGENT; HYDRAZONE DERIVATIVE; NYSTATIN; TETRACYCLINE; TOSYLCHLORAMIDE SODIUM; ANTIBIOTIC AGENT; ANTIFUNGAL AGENT; PYRAZOLE DERIVATIVE;

ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS FLAVUS; ASPERGILLUS NIGER; BACILLUS CEREUS; CARBON NUCLEAR MAGNETIC RESONANCE; CYCLIZATION; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; FUSARIUM OXYSPORUM; IN VITRO STUDY; INFRARED SPECTROSCOPY; KLEBSIELLA PNEUMONIAE; LIQUID CHROMATOGRAPHY; MASS SPECTROMETRY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; REACTION TIME; STAPHYLOCOCCUS AUREUS; FUSARIUM; FUSARIUM MONALIFORME; MINIMUM BACTERICIDAL CONCENTRATION;

FUNGI;

1,3,4-OXADIAZOLES; ANTIMICROBIAL ACTIVITY; CHLORAMINE-T; MINIMUM INHIBITORY CONCENTRATION (MIC); PYRAZOLE;

ANTI-BACTERIAL AGENTS; ANTIFUNGAL AGENTS; BACTERIA; DOSE-RESPONSE RELATIONSHIP, DRUG; FUNGI; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; OXADIAZOLES; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84891482892 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.11.029 Document Type: Article

Times cited : (79)

References (44)

1
- 0031579941
- L.F. Tietze, A. Steinmetz, and F. Balkenhohl Bioorg. Med. Chem. Lett. 7 1997 1303
- (1997) Bioorg. Med. Chem. Lett. , vol.7 , pp. 1303
- Tietze, L.F.¹ Steinmetz, A.² Balkenhohl, F.³

2
- 84891487309
- P. Grosche, A. Holtzel, T.B. Walk, A.W. Trautwein, and G. Jung Synthesis 1961 1999
- (1999) Synthesis , vol.1961
- Grosche, P.¹ Holtzel, A.² Walk, T.B.³ Trautwein, A.W.⁴ Jung, G.⁵

3
- 13444266910
- T.D. Penning, J.J. Talley, S.R. Bertenshaw, J.S. Carter, P.W. Collins, S. Docter, M.J. Graneto, L.F. Lee, J.W. Malecha, J.M. Miyashiro, R.S. Rogers, D.J. Rogier, S.S. Yu, G.D. Anderson, E.G. Burton, J.N. Cogburn, S.A. Gregory, C.M. Koboldt, W.E. Perkins, K. Seibert, A.W. Veenhuizen, Y.Y. Zhang, and P.C. Isakson J. Med. Chem. 40 1997 1347
- (1997) J. Med. Chem. , vol.40 , pp. 1347
- Penning, T.D.¹ Talley, J.J.² Bertenshaw, S.R.³ Carter, J.S.⁴ Collins, P.W.⁵ Docter, S.⁶ Graneto, M.J.⁷ Lee, L.F.⁸ Malecha, J.W.⁹ Miyashiro, J.M.¹⁰ Rogers, R.S.¹¹ Rogier, D.J.¹² Yu, S.S.¹³ Anderson, G.D.¹⁴ Burton, E.G.¹⁵ Cogburn, J.N.¹⁶ Gregory, S.A.¹⁷ Koboldt, C.M.¹⁸ Perkins, W.E.¹⁹ Seibert, K.²⁰ more..

4
- 0037019275
- J. Regan, S. Breitfelder, P. Cirillo, T. Gilmore, A.G. Graham, E. Hickey, B. Klaus, J. Madwed, M. Moriak, N. Moss, C. Pargellis, S. Pav, A. Proto, A. Swinamer, L. Tang, and C. Torcellini J. Med. Chem. 45 2002 2994
- (2002) J. Med. Chem. , vol.45 , pp. 2994
- Regan, J.¹ Breitfelder, S.² Cirillo, P.³ Gilmore, T.⁴ Graham, A.G.⁵ Hickey, E.⁶ Klaus, B.⁷ Madwed, J.⁸ Moriak, M.⁹ Moss, N.¹⁰ Pargellis, C.¹¹ Pav, S.¹² Proto, A.¹³ Swinamer, A.¹⁴ Tang, L.¹⁵ Torcellini, C.¹⁶

5
- 2942522534
- P. Pevarello, M.G. Brasca, R. Amici, P. Orsini, G. Traquandi, L. Corti, C. Piutti, P. Sansonna, M. Villa, B.S. Pierce, M. Pulici, P. Giordano, K. Martina, E.L. Fritzen, R.A. Nugent, E. Casale, A. Cameron, M. Ciomei, F. Roletto, A. Isacchi, G. Fogliatto, E. Pesenti, W. Pastori, A. Marsiglio, K.L. Leach, P.M. Clare, F. Fiorentini, M. Varasi, A. Vulpetti, and M.A. Warpehoski J. Med. Chem. 47 2004 3367
- (2004) J. Med. Chem. , vol.47 , pp. 3367
- Pevarello, P.¹ Brasca, M.G.² Amici, R.³ Orsini, P.⁴ Traquandi, G.⁵ Corti, L.⁶ Piutti, C.⁷ Sansonna, P.⁸ Villa, M.⁹ Pierce, B.S.¹⁰ Pulici, M.¹¹ Giordano, P.¹² Martina, K.¹³ Fritzen, E.L.¹⁴ Nugent, R.A.¹⁵ Casale, E.¹⁶ Cameron, A.¹⁷ Ciomei, M.¹⁸ Roletto, F.¹⁹ Isacchi, A.²⁰ more..

6
- 0033661951
- C. Hansong, Zhengming Li, and H. Yufeng Agric. Food Chem. 48 2000 5312
- (2000) Agric. Food Chem. , vol.48 , pp. 5312
- Hansong, C.¹ Li, Z.² Yufeng, H.³

7
- 0030572496
- N.K. Terrett, A.S. Bell, D. Brown, and P. Ellis Bioorg. Med. Chem. Lett. 6 1996 1819
- (1996) Bioorg. Med. Chem. Lett. , vol.6 , pp. 1819
- Terrett, N.K.¹ Bell, A.S.² Brown, D.³ Ellis, P.⁴

8
- 79953196169
- S. Gang, L. Pengfei, and Yu Rao Org. Lett. 13 2011 1746
- (2011) Org. Lett. , vol.13 , pp. 1746
- Gang, S.¹ Pengfei, L.² Rao, Y.³

9
- 84918022463
- A. Strecker Justus Liebigs Ann. Chem. 75 1850 27
- (1850) Justus Liebigs Ann. Chem. , vol.75 , pp. 27
- Strecker, A.¹

10
- 68049140888
- A. Domling, and I. Ugi Angew. Chem., Int. Ed. 39 2000 3168
- (2000) Angew. Chem., Int. Ed. , vol.39 , pp. 3168
- Domling, A.¹ Ugi, I.²

11
- 0034518876
- C.O. Kappe Acc. Chem. Res. 33 2000 879
- (2000) Acc. Chem. Res. , vol.33 , pp. 879
- Kappe, C.O.¹

12
- 0021884383
- R. Benoit, and C. Daniel J. Heterocycl. Chem. 22 1985 287
- (1985) J. Heterocycl. Chem. , vol.22 , pp. 287
- Benoit, R.¹ Daniel, C.²

13
- 33745758352
- S.L. Gaonkar, K.M.L. Rai, and B. Prabhuswamy Eur. J. Med. Chem. 41 2006 841
- (2006) Eur. J. Med. Chem. , vol.41 , pp. 841
- Gaonkar, S.L.¹ Rai, K.M.L.² Prabhuswamy, B.³

14
- 0001230973
- J.J. Bhatt, B.R. Shah, H.P. Shah, P.B. Trivedi, N.K. Undavia, and N.C. Desai J. Indian Chem. 33B 1994 189
- (1994) J. Indian Chem. , vol.33 B , pp. 189
- Bhatt, J.J.¹ Shah, B.R.² Shah, H.P.³ Trivedi, P.B.⁴ Undavia, N.K.⁵ Desai, N.C.⁶

15
- 33745208794
- T.M. Tan, Y. Chen, K.H. Kong, J. Bai, Y. Li, S.G. Lim, T.H. Ang, and Y. Lam Antiviral Res. 71 2006 7
- (2006) Antiviral Res. , vol.71 , pp. 7
- Tan, T.M.¹ Chen, Y.² Kong, K.H.³ Bai, J.⁴ Li, Y.⁵ Lim, S.G.⁶ Ang, T.H.⁷ Lam, Y.⁸

16
- 30344436995
- A.S. Aboraia, H.M.A. Rahman, N.M. Mahfouz, and M.A. Gendy Bioorg. Med. Chem. Lett. 14 2006 1236
- (2006) Bioorg. Med. Chem. Lett. , vol.14 , pp. 1236
- Aboraia, A.S.¹ Rahman, H.M.A.² Mahfouz, N.M.³ Gendy, M.A.⁴

17
- 84861642773
- J.P. Namita Soni, A.K. Barthwal, K.P. Saxena, and S.S. Bhargava J. Heterocycl. Chem. 19 2009 29
- (2009) J. Heterocycl. Chem. , vol.19 , pp. 29
- Namita Soni, J.P.¹ Barthwal, A.K.² Saxena, K.P.³ Bhargava, S.S.⁴

18
- 17444374605
- M.T.H. Khan, M.I. Choudhary, K.M. Khan, M. Rani, and Atta-ur-Rahman Bioorg. Med. Chem. 13 2005 3385
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 3385
- Khan, M.T.H.¹ Choudhary, M.I.² Khan, K.M.³ Rani, M.⁴ Atta-Ur-Rahman⁵

19
- 29044438582
- C.R.W. Guimaraes, D.L. Boger, and W.L. Jorgensen J. Am. Chem. Soc. 127 2005 17377
- (2005) J. Am. Chem. Soc. , vol.127 , pp. 17377
- Guimaraes, C.R.W.¹ Boger, D.L.² Jorgensen, W.L.³

20
- 13444302530
- V.P.M. Rahman, S. Mukhtar, W.H. Ansari, and G. Lemiere Eur. J. Med. Chem. 40 2005 173
- (2005) Eur. J. Med. Chem. , vol.40 , pp. 173
- Rahman, V.P.M.¹ Mukhtar, S.² Ansari, W.H.³ Lemiere, G.⁴

21
- 0036828026
- S. Peara, and T.F. Patterson Clin. Infect. Dis. 35 2002 1073
- (2002) Clin. Infect. Dis. , vol.35 , pp. 1073
- Peara, S.¹ Patterson, T.F.²

22
- 4544354404
- M. Giulia, M. Luisa, F. Paola, S. Silvia, R. Angelo, M. Luisa, B. Francesco, L. Roberta, M. Chiara, M. Valeria, L.C. Paolo, and T. Elena Bioorg. Med. Chem. 12 2004 5465
- (2004) Bioorg. Med. Chem. , vol.12 , pp. 5465
- Giulia, M.¹ Luisa, M.² Paola, F.³ Silvia, S.⁴ Angelo, R.⁵ Luisa, M.⁶ Francesco, B.⁷ Roberta, L.⁸ Chiara, M.⁹ Valeria, M.¹⁰ Paolo, L.C.¹¹ Elena, T.¹²

23
- 48249125036
- T.A. Vincent J. Antimicrob. Chemother. 44 1999 151
- (1999) J. Antimicrob. Chemother. , vol.44 , pp. 151
- Vincent, T.A.¹

24
- 0033762894
- E. Aiello, S. Aiello, F. Mingoia, A. Bacchi, G. Pelizzi, C. Musiu, M.G. Setzu, A. Pani, P. La Colla, and M.E. Marongiu Bioorg. Med. Chem. 8 2000 2719
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 2719
- Aiello, E.¹ Aiello, S.² Mingoia, F.³ Bacchi, A.⁴ Pelizzi, G.⁵ Musiu, C.⁶ Setzu, M.G.⁷ Pani, A.⁸ La Colla, P.⁹ Marongiu, M.E.¹⁰

25
- 0034706932
- M.S.A. El-Gaby, A.A. Atalla, A.M. Gaber, and K.A. Abd Al-Wahab Farmaco 55 2000 596
- (2000) Farmaco , vol.55 , pp. 596
- El-Gaby, M.S.A.¹ Atalla, A.A.² Gaber, A.M.³ Abd Al-Wahab, K.A.⁴

26
- 0037019175
- B.K. Kaymakcioglu, and S. Rollas Farmaco 57 2002 595
- (2002) Farmaco , vol.57 , pp. 595
- Kaymakcioglu, B.K.¹ Rollas, S.²

27
- 2342485135
- A. Tanitame, Y. Oyamada, K. Ofuji, Y. Kyoya, K. Suziki, H. Ito, M. Kawasaki, K. Nagai, M. Wachi, and J. Yamagishi Bioorg. Med. Chem. Lett. 14 2004 2857
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 2857
- Tanitame, A.¹ Oyamada, Y.² Ofuji, K.³ Kyoya, Y.⁴ Suziki, K.⁵ Ito, H.⁶ Kawasaki, M.⁷ Nagai, K.⁸ Wachi, M.⁹ Yamagishi, J.¹⁰

28
- 2342467510
- A. Tanitame, Y. Oyamada, K. Ofuji, K. Suziki, H. Ito, M. Kawasaki, M. Wachi, and J. Yamagishi Bioorg. Med. Chem. Lett. 14 2004 2863
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 2863
- Tanitame, A.¹ Oyamada, Y.² Ofuji, K.³ Suziki, K.⁴ Ito, H.⁵ Kawasaki, M.⁶ Wachi, M.⁷ Yamagishi, J.⁸

29
- 3042552189
- A. Tanitame, Y. Oyamada, K. Ofuji, M. Fujimoto, N. Iwai, Y. Hiyama, K. Suziki, H. Ito, H. Terauchi, M. Kawasaki, K. Nagai, M. Wachi, and J. Yamagishi J. Med. Chem. 47 2004 3693
- (2004) J. Med. Chem. , vol.47 , pp. 3693
- Tanitame, A.¹ Oyamada, Y.² Ofuji, K.³ Fujimoto, M.⁴ Iwai, N.⁵ Hiyama, Y.⁶ Suziki, K.⁷ Ito, H.⁸ Terauchi, H.⁹ Kawasaki, M.¹⁰ Nagai, K.¹¹ Wachi, M.¹² Yamagishi, J.¹³

30
- 75849162554
- R. Venkat Ragavan, V. Vijayakumar, and N. Suchetha Kumari Eur. J. Med. Chem. 45 2010 1173
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 1173
- Venkat Ragavan, R.¹ Vijayakumar, V.² Suchetha Kumari, N.³

31
- 40049108415
- A.A. Bekhit, H.M.A. Ashour, Y.S.A. Ghany, A.E.D.A. Bekhit, and A. Baraka Eur. J. Med. Chem. 43 2008 456
- (2008) Eur. J. Med. Chem. , vol.43 , pp. 456
- Bekhit, A.A.¹ Ashour, H.M.A.² Ghany, Y.S.A.³ Bekhit, A.E.D.A.⁴ Baraka, A.⁵

32
- 84857921808
- V. Ines, P.R. Andrea, M.M. Kata, B. Karmen, and B. Branimir Bioorg. Med. Chem. 20 2012 2101
- (2012) Bioorg. Med. Chem. , vol.20 , pp. 2101
- Ines, V.¹ Andrea, P.R.² Kata, M.M.³ Karmen, B.⁴ Branimir, B.⁵

33
- 84873048069
- A.M. Vijesh, A.M. Isloor, P. Shetty, S. Sundershan, and H.K. Fun Eur. J. Med. Chem. 62 2013 410
- (2013) Eur. J. Med. Chem. , vol.62 , pp. 410
- Vijesh, A.M.¹ Isloor, A.M.² Shetty, P.³ Sundershan, S.⁴ Fun, H.K.⁵

34
- 70349779197
- N.P. Rai, V.K. Narayanaswamy, S. Shashikanth, and P.N. Arunachalam Eur. J. Med. Chem. 44 2009 4522
- (2009) Eur. J. Med. Chem. , vol.44 , pp. 4522
- Rai, N.P.¹ Narayanaswamy, V.K.² Shashikanth, S.³ Arunachalam, P.N.⁴

35
- 77955553690
- O. Prakash, M. Kumar, R. Kumar, C. Sharma, and K.R. Aneja Eur. J. Med. Chem. 45 2010 4252
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 4252
- Prakash, O.¹ Kumar, M.² Kumar, R.³ Sharma, C.⁴ Aneja, K.R.⁵

36
- 84861622667
- P. Puthiyapurayil, B. Poojary, C. Chikkanna, and S.K. Buridipad Eur. J. Med. Chem. 53 2012 203
- (2012) Eur. J. Med. Chem. , vol.53 , pp. 203
- Puthiyapurayil, P.¹ Poojary, B.² Chikkanna, C.³ Buridipad, S.K.⁴

37
- 78650514875
- M.A. Abu-Zaied, E.M. El-Telbani, G.H. Elgemeie, and G.A.M. Nawwar Eur. J. Med. Chem. 46 2011 229
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 229
- Abu-Zaied, M.A.¹ El-Telbani, E.M.² Elgemeie, G.H.³ Nawwar, G.A.M.⁴

38
- 84880122996
- L. Hong-Shui, Z. Bao-Xiang, L. Ji-Kun, X. Young, L. Song, L. Wei-Young, and G. Zhong-Liang Dyes Pigm. 86 2010 25
- (2010) Dyes Pigm. , vol.86 , pp. 25
- Hong-Shui, L.¹ Bao-Xiang, Z.² Ji-Kun, L.³ Young, X.⁴ Song, L.⁵ Wei-Young, L.⁶ Zhong-Liang, G.⁷

39
- 80053384991
- L. Hong-Shui, X. Yong-Sheng, L. Wei-Yong, Gong Zhong-Liang, and Zhao Bao-Xiang J. Fluoresc. 21 2011 1797
- (2011) J. Fluoresc. , vol.21 , pp. 1797
- Hong-Shui, L.¹ Yong-Sheng, X.² Wei-Yong, L.³ Zhong-Liang, G.⁴ Bao-Xiang, Z.⁵

40
- 84880117082
- P. Horrocks, M.R. Pickard, H. Parekh, S.P. Patel, and B.P. Ravindra Org. Biomol. Chem. 11 2013 4891
- (2013) Org. Biomol. Chem. , vol.11 , pp. 4891
- Horrocks, P.¹ Pickard, M.R.² Parekh, H.³ Patel, S.P.⁴ Ravindra, B.P.⁵

41
- 84880625434
- S. Ningaiah, U.K. Bhadraiah, S. Keshavamurthy, and C. Javarasetty Bioorg. Med. Chem. Lett. 23 2013 4532
- (2013) Bioorg. Med. Chem. Lett. , vol.23 , pp. 4532
- Ningaiah, S.¹ Bhadraiah, U.K.² Keshavamurthy, S.³ Javarasetty, C.⁴

42
- 77954082016
- K.B. Umesha, and K.M.L. Rai Bulg. Chem. Commun. 42 2010 11
- (2010) Bulg. Chem. Commun. , vol.42 , pp. 11
- Umesha, K.B.¹ Rai, K.M.L.²

43
- 47249132185
- J.M. Andrews J. Antimicrob. Chemother. 62 2008 256
- (2008) J. Antimicrob. Chemother. , vol.62 , pp. 256
- Andrews, J.M.¹

44
- 0034828307
- J.R. Zgoda, and J.R. Porter Pharm. Biology. 39 2001 221
- (2001) Pharm. Biology. , vol.39 , pp. 221
- Zgoda, J.R.¹ Porter, J.R.²

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