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Volumn 43, Issue 3, 2008, Pages 456-463

Synthesis and biological evaluation of some thiazolyl and thiadiazolyl derivatives of 1H-pyrazole as anti-inflammatory antimicrobial agents

(5) Bekhit, Adnan A a Ashour, Hayam M A a Abdel Ghany, Yasser S a Bekhit, Alaa El Din A b Baraka, Azza c

a Alexandria University Faculty of Pharmacy (Egypt)

b LINCOLN UNIVERSITY (New Zealand)

c ALEXANDRIA UNIVERSITY (Egypt)

Author keywords

Acute toxicity; Anti inflammatory; Antimicrobial; Pyrazole; Ulcerogenic effect

Indexed keywords

4 BROMOPHENACYL BROMIDE; ACETIC ANHYDRIDE; AMPICILLIN; ANTIINFECTIVE AGENT; ANTIINFLAMMATORY AGENT; BENZENESULFONAMIDE DERIVATIVE; BROMOACETIC ACID; BROMOACETIC ACID ETHYL ESTER; CLOTRIMAZOLE; CYCLOOXYGENASE 2; FERRIC CHLORIDE; INDOMETACIN; PYRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; BIOASSAY; CANDIDA ALBICANS; CONTROLLED STUDY; CYCLIZATION; DRUG ACTIVITY; DRUG SAFETY; DRUG SYNTHESIS; ESCHERICHIA COLI; GRANULOMA; MALE; MOUSE; NONHUMAN; PAW EDEMA; RAT; STAPHYLOCOCCUS AUREUS; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION; ULCEROGENESIS;

ANIMALS; ANTI-INFECTIVE AGENTS; ANTI-INFLAMMATORY AGENTS; BACTERIA; CARRAGEENAN; CYCLOOXYGENASE 1; CYCLOOXYGENASE 2; DRUG DESIGN; EDEMA; FUNGI; GRANULOMA; HUMANS; MALE; MICROBIAL SENSITIVITY TESTS; PYRAZOLES; RATS; THIADIAZOLES; THIAZOLES; ULCER;

EID: 40049108415 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2007.03.030 Document Type: Article

Times cited : (315)

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