Solid-phase synthesis of polymer-bound β-ketoesters and their application in the synthesis of structurally diverse pyrazolones

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 10, 1997, Pages 1303-1306

  Tietze, Lutz F ^a   Steinmetz, Adrian ^a   Balkenhohl, Friedhelm ^b  

^a UNIVERSITY OF GÖTTINGEN   (Germany)

^b BASF SE   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

PYRAZOLONE DERIVATIVE;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; INFRARED SPECTROPHOTOMETRY; REACTION ANALYSIS; TECHNIQUE;

EID: 0031579941     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00209-6     Document Type: Article

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21. Polymer-bound acetoacetate was prepared according to .
22. All compounds were characterized by NMR and MS.
23. Purities were determined by NMR.