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Bioorganic and Medicinal Chemistry

Volumn 21, Issue 22, 2013, Pages 7210-7215

Structural study of interaction between brinzolamide and dorzolamide inhibition of human carbonic anhydrases

(5) Pinard, Melissa A a Boone, Christopher D a Rife, Brittany D a Supuran, Claudiu T b McKenna, Robert a

a UNIVERSITY OF FLORIDA COLLEGE OF MEDICINE (United States)

b UNIVERSITY OF FLORENCE (Italy)

Author keywords

Brinzolamide; Dorzolamide; Human carbonic anhydrase

Indexed keywords

BRINZOLAMIDE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE IX; DORZOLAMIDE;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG BINDING; DRUG BINDING SITE; ENZYME ACTIVE SITE; ENZYME INHIBITION; MOLECULAR DOCKING; SITE DIRECTED MUTAGENESIS; STRUCTURE ANALYSIS; X RAY CRYSTALLOGRAPHY;

BRINZOLAMIDE; BRZ; CA; CA II; CA IX; CARBONIC ANHYDRASE; DORZOLAMIDE; DRZ; HUMAN CARBONIC ANHYDRASE; HUMAN CARBONIC ANHYDRASE II; HUMAN CARBONIC ANHYDRASE IX;

ANTIGENS, NEOPLASM; BINDING SITES; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; CATALYTIC DOMAIN; CRYSTALLOGRAPHY, X-RAY; HUMANS; KINETICS; MOLECULAR DOCKING SIMULATION; MUTAGENESIS, SITE-DIRECTED; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; THERMODYNAMICS; THIAZINES; THIOPHENES;

EID: 84885838420 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2013.08.033 Document Type: Article

Times cited : (89)

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