Proteoliposomes as tool for assaying membrane transporter functions and interactions with xenobiotics

Pharmaceutics

Volumn 5, Issue 3, 2013, Pages 472-497

  Scalise, Mariafrancesca ^a   Pochini, Lorena ^a   Giangregorio, Nicola ^b   Tonazzi, Annamaria ^b   Indiveri, Cesare ^a,b  

^a UNIVERSITY OF CALABRIA   (Italy)

^b CNR   (Italy)

Author keywords

Drug discovery; Drugs; Proteoliposomes; Reconstitution; Transport; Xenobiotics

Indexed keywords

ABC TRANSPORTER; AMINO ACID TRANSPORTER; AMPICILLIN; BETA LACTAM ANTIBIOTIC; CARNITINE ACYLCARNITINE TRANSPORTER; CEFONICID; CITRULLINE; MELDONIUM; OMEPRAZOLE; ORGANIC ANION TRANSPORTER 1; ORGANIC CATION TRANSPORTER 1; ORGANIC CATION TRANSPORTER 2; ORNITHINE; ORNITHINE CITRULLINE TRANSPORTER; PROTEOLIPOSOME; SODIUM GLUCOSE COTRANSPORTER 1; UNCLASSIFIED DRUG; XENOBIOTIC AGENT;

ABSORPTION; ARTICLE; BINDING AFFINITY; BINDING SITE; CARDIOMYOPATHY; CATALYSIS; CELL MEMBRANE; DRUG ACTIVITY; DRUG MEGADOSE; DRUG PROTEIN BINDING; DRUG SAFETY; DRUG STRUCTURE; ELECTROCHEMISTRY; ENDOPLASMIC RETICULUM; ENZYME KINETICS; FATTY ACID OXIDATION; FATTY LIVER; GENE EXPRESSION PROFILING; GENE SEQUENCE; GLYCOSYLATION; HOMEOSTASIS; HUMAN; HYDROPHILICITY; HYDROPHOBICITY; MEMBRANE RECONSTITUTION; MOLECULAR DYNAMICS; NONHUMAN; PHOSPHOLIPID BILAYER; PROTEIN BINDING; PROTEIN LOCALIZATION; PROTEIN METABOLISM; PROTEIN MODIFICATION; PROTEIN MOTIF; PROTEIN PURIFICATION; PROTEIN SECONDARY STRUCTURE; PROTEIN TRANSPORT; SEQUENCE HOMOLOGY; SITE DIRECTED MUTAGENESIS; STRUCTURAL HOMOLOGY;

EID: 84884741685     PISSN: None     EISSN: 19994923     Source Type: Journal    
DOI: 10.3390/pharmaceutics5030472     Document Type: Article

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