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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 16, 2013, Pages 4547-4551

1,2,4-Triazole derivatives as transient inactivators of kallikreins involved in skin diseases

(6) Tan, Xiao a Furio, Laetitia b Reboud Ravaux, Michèle a Villoutreix, Bruno O b Hovnanian, Alain b El Amri, Chahrazade a

a SORBONNE UNIVERSITÉ (France)

b UNIVERSITÉ PARIS DESCARTES (France)

Author keywords

Acyl enzymes; Inhibitors; Kallikreins; Matriptase; Netherton syndrome; Transient inactivators

Indexed keywords

1,2,4 TRIAZOLE DERIVATIVE; ENZYME; KALLIKREIN; MATRIPTASE;

ARTICLE; ENZYME STRUCTURE; HUMAN; KERATINOCYTE; MOLECULAR WEIGHT; NETHERTON DISEASE; NONHUMAN; PROTEIN DEGRADATION; PROTEIN TARGETING; SKIN DISEASE;

3-AMINO-7-METHYL-COUMARIN; ACYL-ENZYMES; AMC; DIMETHYL SULFOXIDE; DMSO; HIGH THROUGHPUT SCREENING; HK; HTS; HUMAN KALLIKREIN; INHIBITORS; KALLIKREINS; LEKTI; LYMPHO-EPITHELIAL KAZAL-TYPE INHIBITOR; MATRIPTASE; NETHERTON SYNDROME; TRANSIENT INACTIVATORS;

CELL SURVIVAL; ENZYME ACTIVATION; ENZYME INHIBITORS; HUMANS; KALLIKREINS; KERATINOCYTES; SKIN DISEASES; TRIAZOLES;

EID: 84880580104 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.06.039 Document Type: Article

Times cited : (29)

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