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Volumn 4, Issue 6, 2013, Pages 1034-1041

Introduction of methionine mimics on 3-arylthiophene: Influence on protein farnesyltransferase inhibition and on antiparasitic activity

(6) Bosc, Damien a Mouray, Elisabeth b Grellier, Philippe b Cojean, Sandrine c Loiseau, Philippe M c Dubois, Joëlle a

a CNRS (France)

b MUSÉUM NATIONAL D'HISTOIRE NATURELLE (France)

c UNIVERSITÉ PARIS SACLAY (France)

Author keywords

[No Author keywords available]

Indexed keywords

3 ARYLTHIOPHENE DERIVATIVE; ANTIPARASITIC AGENT; CHLOROQUINE; METHIONINE; PROTEIN FARNESYLTRANSFERASE; PROTEIN FARNESYLTRANSFERASE INHIBITOR; UNCLASSIFIED DRUG;

ANTIPROTOZOAL ACTIVITY; ARTICLE; CHEMICAL MODIFICATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; LEISHMANIA DONOVANI; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; TRYPANOSOMA BRUCEI; TRYPANOSOMA CRUZI;

LEISHMANIA DONOVANI; PLASMODIUM FALCIPARUM; PROTOZOA; TRYPANOSOMA BRUCEI; TRYPANOSOMA BRUCEI BRUCEI; TRYPANOSOMA CRUZI;

EID: 84878773852 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c3md00065f Document Type: Article

Times cited : (8)

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