TRPM8 ion channel ligands for new therapeutic applications and as probes to study menthol pharmacology

Life Sciences

Volumn 92, Issue 8-9, 2013, Pages 425-437

  Journigan, V Blair ^a   Zaveri, Nurulain T ^a  

^a Astraea Therapeutics Inc   (Spain)

Author keywords

Addiction; Agonist; Antagonist; Menthol; Nicotine; TRPM8

Indexed keywords

'PBMC'; 1 (2 HYDROXYPHENYL) 4 (3 NITROPHENYL) 1,2,3,6 TETRAHYDROPYRIMIDIN 2 ONE; 4 BENZYLOXYBENZOIC ACID AMIDE DERIVATIVE; 4-BENZYLOXY BENZYLOXYPHENYLMETHYLAMIDE DERIVATIVE; AMTB; BENZYLOXY PHENYLMETHYLCARBAMATE DERIVATIVE; BENZYLOXYPHENYLMETHYLUREA DERIVATIVE; D 3263; JNJ 39267631; MENTHOL; TETRAHYDROISOQUINOLINE; TRANSIENT RECEPTOR POTENTIAL CHANNEL AFFECTING AGENT; TRANSIENT RECEPTOR POTENTIAL CHANNEL M8; UNCLASSIFIED DRUG;

COLD SENSITIVITY; CONFERENCE PAPER; DRUG EFFICACY; DRUG METABOLISM; HUMAN; INFLAMMATORY PAIN; INTERSTITIAL CYSTITIS; NEUROPATHIC PAIN; NONHUMAN; OVERACTIVE BLADDER; PROSTATE CANCER; PROSTATE HYPERTROPHY; SMOKING; TOBACCO DEPENDENCE; URINARY TRACT DISEASE;

ANIMALS; ANTINEOPLASTIC AGENTS; COLD TEMPERATURE; FEMALE; HUMANS; INFLAMMATION; LIGANDS; MALE; MENTHOL; NEURALGIA; PROSTATIC HYPERPLASIA; PROSTATIC NEOPLASMS; SENSORY RECEPTOR CELLS; SMOKING; THERMOSENSING; TRPM CATION CHANNELS; UROLOGIC DISEASES;

EID: 84874650819     PISSN: 00243205     EISSN: 18790631     Source Type: Journal    
DOI: 10.1016/j.lfs.2012.10.032     Document Type: Conference Paper

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