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ChemMedChem

Volumn 8, Issue 3, 2013, Pages 385-395

Carboxylic Acid (Bio)Isosteres in Drug Design

(3) Ballatore, Carlo a Huryn, Donna M a Smith III, Amos B a

a UNIVERSITY OF PENNSYLVANIA (United States)

Author keywords

Bioisosteres; Carboxylic acids; Drug design; Isosteric replacement

Indexed keywords

1,2,4 OXADIAZOLE DERIVATIVE; 1,2,4 THIADIAZOLE DERIVATIVE; 2,4 THIAZOLIDINEDIONE DERIVATIVE; 3 HYDROXYQUINOLIN 2 ONE DERIVATIVE; 4 AMINOBUTYRIC ACID B RECEPTOR BLOCKING AGENT; 4 HYDROXYQUINOLIN 2 ONE DERIVATIVE; 5 OXO 1,2,4 OXADIAZOLE DERIVATIVE; 5 OXO 1,2,4 THIADIAZOLE DERIVATIVE; 5 THIOXO 1,2,4 OXADIAZOLE DERIVATIVE; CARBOXYLIC ACID; CARBOXYLIC ACID BIOISOSTERE DERIVATIVE; CHOLECYSTOKININ B RECEPTOR ANTAGONIST; CYCLOPENTANE 1,3 DIONE DERIVATIVE; CYCLOPENTANE DERIVATIVE; DIFLUOROPHENOL DERIVATIVE; FUNCTIONAL GROUP; HYDROXAMIC ACID; ISOTHIAZOLE DERIVATIVE; OXAZOLIDINEDIONE DERIVATIVE; PHENOL DERIVATIVE; QUINOLINE DERIVATIVE; SQUARIC ACID DERIVATIVE; SULFINIC ACID DERIVATIVE; SULFONAMIDE; SULFONIC ACID DERIVATIVE; SULFONYLUREA DERIVATIVE; TETRAMIC ACID DERIVATIVE; TETRAZOLE DERIVATIVE; TETRONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ARTICLE; DRUG DESIGN; DRUG DIFFUSION; DRUG RECEPTOR BINDING; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; MEMBRANE PERMEABILITY; NONHUMAN; PASSIVE TRANSPORT; PATENT; PHARMACOPHORE; PRIORITY JOURNAL; PROTON TRANSPORT; TAUTOMERIZATION;

AZOLES; CARBOXYLIC ACIDS; DRUG DESIGN; FURANS; HYDROXAMIC ACIDS; KETONES; KINETICS; PHOSPHOROUS ACIDS; SULFONAMIDES; SULFONIC ACIDS;

EID: 84874353612 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201200585 Document Type: Article

Times cited : (384)

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