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European Journal of Medicinal Chemistry

Volumn 62, Issue , 2013, Pages 270-279

Synthesis of some new 2-(3-pyridyl)-4,5-disubstituted thiazoles as potent antimicrobial agents

(3) Bondock, Samir a,b Naser, Tamer b,c Ammar, Yousry A b,d

a Mansoura University (Egypt)

b KING KHALID UNIVERSITY (Saudi Arabia)

c Helwan (Egypt)

d AL AZHAR UNIVERSITY (Egypt)

Author keywords

Antimicrobial activity; Chalcone; Pyrazoline; Pyridine; Thiazole

Indexed keywords

1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) 3 (2 NITROPHENYL) PROPENONE; 1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) 3 PHENYLPROPENONE; 1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) ETHANONE; 3 (2 PYRIDIN 3 YL THIAZOL 4 YL) CHROMEN 2 ONE; 3 (2,4 DIFLUOROPHENYL) 1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) PROPENONE; 3 (4 CHLOROPHENYL) 1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) PROPENONE; 3 (4 METHOXYPHENYL) 1 (4 METHYL 2 PYRIDIN 3 YL THIAZOL 5 YL) PROPENONE; 3 (4 METHYLTHIAZOL 2 YL) PYRIDINE; 3 [4 METHYL 5 (5 PHENYL 4,5 DIHYDRO 1H PYRAZOL 3 YL)THIAZOL 2 YL] PYRIDINE; 3 [4 METHYL 5 [5 (2 NITROPHENYL) 4,5 DIHYDRO 1H PYRAZOL 3 YL]THIAZOL 2 YL] PYRIDINE; 3 [5 [5 (2,4 DIFLUOROPHENYL) 4,5 DIHYDRO 1H PYRAZOL 3 YL] 4 METHYL THIAZOL 2 YL] PYRIDINE; 3 [5 [5 (4 CHLOROPHENYL) 4,5 DIHYDRO 1H PYRAZOL 3 YL] 4 METHYL THIAZOL 2 YL] PYRIDINE; 3 [5 [5 (4 METHOXYPHENYL) 4,5 DIHYDRO 1H PYRAZOL 3 YL] 4 METHYL THIAZOL 2 YL] PYRIDINE; 5 ACETYL 4 METHYL 2 (3 PYRIDYL)THIAZOLE; AMPHOTERICIN B; AMPICILLIN; ANTIBIOTIC AGENT; ANTIFUNGAL AGENT; N [4 (2 PYRIDIN 3 YL THIAZOL 4 YL) PHENYL] ACETAMIDE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS CLAVATUS; ASPERGILLUS FUMIGATUS; BACILLUS SUBTILIS; BACTERIAL STRAIN; CANDIDA ALBICANS; CONTROLLED STUDY; DISK DIFFUSION; DRUG SCREENING; DRUG SYNTHESIS; ENTEROCOCCUS FAECALIS; FUNGAL STRAIN; GEOTRICHUM; GROWTH INHIBITION; IN VITRO STUDY; KLEBSIELLA PNEUMONIAE; NEISSERIA GONORRHOEAE; NONHUMAN; PENICILLIUM MARNEFFEI; PROTEUS VULGARIS; PSEUDOMONAS AERUGINOSA; SHIGELLA FLEXNERI; SPECTROSCOPY; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS; STREPTOCOCCUS PYOGENES; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; ANTIFUNGAL AGENTS; BACTERIA; DOSE-RESPONSE RELATIONSHIP, DRUG; FUNGI; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 84873022161 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2012.12.050 Document Type: Article

Times cited : (120)

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