SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 1, 2013, Pages 112-116

Synthesis, antimalarial activity and cytotoxic potential of new monocarbonyl analogues of curcumin

(10) Manohar, Sunny a Khan, Shabana I b Kandi, Shamseer Kulangara a Raj, Kranthi a Sun, Guojing c Yang, Xiaochuan c Calderon Molina, Angie D c Ni, Nanting c Wang, Binghe c Rawat, Diwan S a

a UNIVERSITY OF DELHI (India)

b UNIVERSITY OF MISSISSIPPI (United States)

c GEORGIA STATE UNIVERSITY (United States)

Author keywords

Anticancer; Antimalarial; Curcumin; Cytotoxicity; HeLa cell line

Indexed keywords

ANTIMALARIAL AGENT; ANTINEOPLASTIC AGENT; CURCUMIN; DOXORUBICIN;

ANTIMALARIAL ACTIVITY; ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CONTROLLED STUDY; CYTOTOXICITY; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; PLASMODIUM FALCIPARUM;

ANTIMALARIALS; ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL SURVIVAL; CURCUMIN; DRUG DESIGN; HELA CELLS; HUMANS; PLASMODIUM FALCIPARUM; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP;

PLASMODIUM FALCIPARUM;

EID: 84870984106 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.11.004 Document Type: Article

Times cited : (63)

References (56)

1
- 42949160050
- D.J. Newman J. Med. Chem. 51 2008 2589
- (2008) J. Med. Chem. , vol.51 , pp. 2589
- Newman, D.J.¹

2
- 55949084512
- P. Anand, S.G. Thomas, A.B. Kunnumakkara, C. Sundaram, K.B. Harikumar, B. Sung, S.T. Tharakan, K. Misra, I.K. Priyadarsini, K.N. Rajasekharan, and B.B. Aggarwal Biochem. Pharmacol. 76 2008 1590
- (2008) Biochem. Pharmacol. , vol.76 , pp. 1590
- Anand, P.¹ Thomas, S.G.² Kunnumakkara, A.B.³ Sundaram, C.⁴ Harikumar, K.B.⁵ Sung, B.⁶ Tharakan, S.T.⁷ Misra, K.⁸ Priyadarsini, I.K.⁹ Rajasekharan, K.N.¹⁰ Aggarwal, B.B.¹¹

3
- 0026093041
- H.P. Ammon, and M.A. Wahl Planta Med. 57 1991 1
- (1991) Planta Med. , vol.57 , pp. 1
- Ammon, H.P.¹ Wahl, M.A.²

4
- 44749093175
- H. Hatcher, R. Planalp, J. Cho, F.M. Torti, and S.V. Torti Cell. Mol. Life Sci. 65 2008 1631
- (2008) Cell. Mol. Life Sci. , vol.65 , pp. 1631
- Hatcher, H.¹ Planalp, R.² Cho, J.³ Torti, F.M.⁴ Torti, S.V.⁵

5
- 0037236792
- B.B. Aggarwal, A. Kumar, and A.C. Bharti Anticancer Res. 23 2003 363
- (2003) Anticancer Res. , vol.23 , pp. 363
- Aggarwal, B.B.¹ Kumar, A.² Bharti, A.C.³

6
- 0142166328
- Y.J. Surh Nat. Rev. Cancer 3 2003 768
- (2003) Nat. Rev. Cancer , vol.3 , pp. 768
- Surh, Y.J.¹

7
- 84870996036
- O.P. Sharma Biochem. Pharmacol. 1976 1811 25
- (1811) Biochem. Pharmacol. , vol.1976 , pp. 25
- Sharma, O.P.¹

8
- 0029648973
- A.J. Ruby, G. Kuttan, K.D. Babu, K.N. Rajasekharan, and R. Kuttan Cancer Lett. 94 1995 79
- (1995) Cancer Lett. , vol.94 , pp. 79
- Ruby, A.J.¹ Kuttan, G.² Babu, K.D.³ Rajasekharan, K.N.⁴ Kuttan, R.⁵

9
- 0029979805
- Y. Sugiyama, S. Kawakishi, and T. Osawa Biochem. Pharmacol. 52 1996 519
- (1996) Biochem. Pharmacol. , vol.52 , pp. 519
- Sugiyama, Y.¹ Kawakishi, S.² Osawa, T.³

10
- 0015785965
- R.C. Srimal, and B.N. Dhawan J. Pharm. Pharmacol. 25 1973 447
- (1973) J. Pharm. Pharmacol. , vol.25 , pp. 447
- Srimal, R.C.¹ Dhawan, B.N.²

11
- 33846624650
- L. Cui, J. Miao, and L. Cui Antimicrob. Agents Chemother. 51 2007 488
- (2007) Antimicrob. Agents Chemother. , vol.51 , pp. 488
- Cui, L.¹ Miao, J.² Cui, L.³

12
- 0021033789
- Y. Kiso, Y. Suzuki, N. Watanabe, Y. Oshima, and H. Hikino Planta Med. 49 1983 185
- (1983) Planta Med. , vol.49 , pp. 185
- Kiso, Y.¹ Suzuki, Y.² Watanabe, N.³ Oshima, Y.⁴ Hikino, H.⁵

13
- 0033979590
- N. Venkatesan, D. Punithavathi, and V. Arumugam Br. J. Pharmacol. 129 2000 231
- (2000) Br. J. Pharmacol. , vol.129 , pp. 231
- Venkatesan, N.¹ Punithavathi, D.² Arumugam, V.³

14
- 0022401146
- R. Srivastava, M. Dikshit, R.C. Srimal, and B.N. Dhawan Thromb. Res. 40 1985 413
- (1985) Thromb. Res. , vol.40 , pp. 413
- Srivastava, R.¹ Dikshit, M.² Srimal, R.C.³ Dhawan, B.N.⁴

15
- 0028887709
- M. Dikshit, L. Rastogi, R. Shukla, and R.C. Srimal Indian J. Med. Res. 101 1995 31
- (1995) Indian J. Med. Res. , vol.101 , pp. 31
- Dikshit, M.¹ Rastogi, L.² Shukla, R.³ Srimal, R.C.⁴

16
- 0030002254
- C. Nirmala, and R. Puvanakrishnan Mol. Cell. Biochem. 159 1996 85
- (1996) Mol. Cell. Biochem. , vol.159 , pp. 85
- Nirmala, C.¹ Puvanakrishnan, R.²

17
- 0030045859
- C. Nirmala, and R. Puvanakrishnan Biochem. Pharmacol. 51 1996 47
- (1996) Biochem. Pharmacol. , vol.51 , pp. 47
- Nirmala, C.¹ Puvanakrishnan, R.²

18
- 0015319846
- M. Srinivasan Indian. J. Med. Sci. 26 1972 269
- (1972) Indian. J. Med. Sci. , vol.26 , pp. 269
- Srinivasan, M.¹

19
- 0028807262
- P.S. Babu, and K. Srinivasan Mol. Cell. Biochem. 152 1995 13
- (1995) Mol. Cell. Biochem. , vol.152 , pp. 13
- Babu, P.S.¹ Srinivasan, K.²

20
- 8044223405
- P.S. Babu, and K. Srinivasan Mol. Cell. Biochem. 166 1997 169
- (1997) Mol. Cell. Biochem. , vol.166 , pp. 169
- Babu, P.S.¹ Srinivasan, K.²

21
- 0036007614
- N. Arun, and N. Nalini Plant Foods Hum. Nutr. 57 2002 41
- (2002) Plant Foods Hum. Nutr. , vol.57 , pp. 41
- Arun, N.¹ Nalini, N.²

22
- 0018887037
- S.D. Deodhar, R. Sethi, and R.C. Srimal Indian J. Med. Res. 71 1980 632
- (1980) Indian J. Med. Res. , vol.71 , pp. 632
- Deodhar, S.D.¹ Sethi, R.² Srimal, R.C.³

23
- 0035174504
- A.L. Cheng, C.H. Hsu, J.K. Lin, M.M. Hsu, Y.F. Ho, T.S. Shen, J.Y. Ko, J.T. Lin, B.R. Lin, W. Ming-Shiang, H.S. Yu, S.H. Jee, G.S. Chen, T.M. Chen, C.A. Chen, M.K. Lai, Y.S. Pu, M.H. Pan, Y.J. Wang, C.C. Tsai, and C.Y. Hsieh Anticancer Res. 21 2001 2895
- (2001) Anticancer Res. , vol.21 , pp. 2895
- Cheng, A.L.¹ Hsu, C.H.² Lin, J.K.³ Hsu, M.M.⁴ Ho, Y.F.⁵ Shen, T.S.⁶ Ko, J.Y.⁷ Lin, J.T.⁸ Lin, B.R.⁹ Ming-Shiang, W.¹⁰ Yu, H.S.¹¹ Jee, S.H.¹² Chen, G.S.¹³ Chen, T.M.¹⁴ Chen, C.A.¹⁵ Lai, M.K.¹⁶ Pu, Y.S.¹⁷ Pan, M.H.¹⁸ Wang, Y.J.¹⁹ Tsai, C.C.²⁰ Hsieh, C.Y.²¹ more..

24
- 84871016195
- H. Inano, M. Onoda, N. Inafuku, M. Kubota, Y. Kamada, T. Osawa, H. Kobayashi, and K. Wakabayashi Carcinogenesis 1011 1999 20
- (1999) Carcinogenesis , vol.1011 , pp. 20
- Inano, H.¹ Onoda, M.² Inafuku, N.³ Kubota, M.⁴ Kamada, Y.⁵ Osawa, T.⁶ Kobayashi, H.⁷ Wakabayashi, K.⁸

25
- 0029947057
- M.A. Ereira, C.J. Grubbs, L.H. Barnes, H. Li, G.R. Olson, I. Eto, M. Juliana, L.M. Whitaker, G.J. Kelloff, V.E. Steele, and R.A. Lubet Carcinogenesis 17 1996 1305
- (1996) Carcinogenesis , vol.17 , pp. 1305
- Ereira, M.A.¹ Grubbs, C.J.² Barnes, L.H.³ Li, H.⁴ Olson, G.R.⁵ Eto, I.⁶ Juliana, M.⁷ Whitaker, L.M.⁸ Kelloff, G.J.⁹ Steele, V.E.¹⁰ Lubet, R.A.¹¹

26
- 72549087782
- C. Schaaf, B. Shan, M. Buchfelder, M. Losa, J. Kreutzer, W. Rachinger, G.K. Stalla, T. Schilling, E. Arzt, M.J. Perone, and U. Renner Endocr. Relat. Cancer 16 2009 1339
- (2009) Endocr. Relat. Cancer , vol.16 , pp. 1339
- Schaaf, C.¹ Shan, B.² Buchfelder, M.³ Losa, M.⁴ Kreutzer, J.⁵ Rachinger, W.⁶ Stalla, G.K.⁷ Schilling, T.⁸ Arzt, E.⁹ Perone, M.J.¹⁰ Renner, U.¹¹

27
- 84870975931
- T.J. Somers-Edgar, M.J. Scandlyn, E.C. Stuart, M.J. Le Nedelec, S.P. Valentine, and R.J. Rosengren Int. J. Cancer 2008 1966 122
- (1966) Int. J. Cancer , vol.2008 , pp. 122
- Somers-Edgar, T.J.¹ Scandlyn, M.J.² Stuart, E.C.³ Le Nedelec, M.J.⁴ Valentine, S.P.⁵ Rosengren, R.J.⁶

28
- 33344461738
- A.R. Hussain, M. Al-Rasheed, P.S. Manogaran, K.A. Al-Hussein, L.C. Platanias, K. Al Kuraya, and S. Uddin Apoptosis 11 2006 245
- (2006) Apoptosis , vol.11 , pp. 245
- Hussain, A.R.¹ Al-Rasheed, M.² Manogaran, P.S.³ Al-Hussein, K.A.⁴ Platanias, L.C.⁵ Al Kuraya, K.⁶ Uddin, S.⁷

29
- 33745918631
- C.S. Beevers, F. Li, L. Liu, and S. Huang Int. J. Cancer 119 2006 757
- (2006) Int. J. Cancer , vol.119 , pp. 757
- Beevers, C.S.¹ Li, F.² Liu, L.³ Huang, S.⁴

30
- 68549083507
- S.M. Johnson, P. Gulhati, I. Arrieta, X. Wang, T. Uchida, T. Gao, and B.M. Evers Anticancer Res. 29 2009 3185
- (2009) Anticancer Res. , vol.29 , pp. 3185
- Johnson, S.M.¹ Gulhati, P.² Arrieta, I.³ Wang, X.⁴ Uchida, T.⁵ Gao, T.⁶ Evers, B.M.⁷

31
- 36448981749
- S. Shankar, Q. Chen, K. Sarva, I. Siddiqui, and R.K. Srivastava J. Mol. Signal. 2 2007 10
- (2007) J. Mol. Signal. , vol.2 , pp. 10
- Shankar, S.¹ Chen, Q.² Sarva, K.³ Siddiqui, I.⁴ Srivastava, R.K.⁵

32
- 68849083504
- C.P. Prasad, G. Rath, S. Mathur, D. Bhatnagar, and R. Ralhan Chem. Biol. Interact. 181 2009 263
- (2009) Chem. Biol. Interact. , vol.181 , pp. 263
- Prasad, C.P.¹ Rath, G.² Mathur, S.³ Bhatnagar, D.⁴ Ralhan, R.⁵

33
- 70350225860
- F.H. Sarkar, and Y. Li Cancer Treat. Rev. 35 2009 597
- (2009) Cancer Treat. Rev. , vol.35 , pp. 597
- Sarkar, F.H.¹ Li, Y.²

34
- 37549051274
- P. Anand, A.B. Kunnumakkara, R.A. Newman, and B.B. Aggarwal Mol. Pharm. 4 2007 807
- (2007) Mol. Pharm. , vol.4 , pp. 807
- Anand, P.¹ Kunnumakkara, A.B.² Newman, R.A.³ Aggarwal, B.B.⁴

35
- 77449124082
- E. Burgos-Moron, J.M. Calderon-Montano, J. Salvador, A. Robles, and M. Lopez-Lazaro Int. J. Cancer 126 2010 1771
- (2010) Int. J. Cancer , vol.126 , pp. 1771
- Burgos-Moron, E.¹ Calderon-Montano, J.M.² Salvador, J.³ Robles, A.⁴ Lopez-Lazaro, M.⁵

36
- 1542286600
- M.J. Rosemond, L. St John-Williams, T. Yamaguchi, T. Fujishita, and J.S. Walsh Chem. Biol. Interact. 147 2004 129
- (2004) Chem. Biol. Interact. , vol.147 , pp. 129
- Rosemond, M.J.¹ St John-Williams, L.² Yamaguchi, T.³ Fujishita, T.⁴ Walsh, J.S.⁵

37
- 77956340070
- B. Yadav, S. Taurin, R.J. Rosengren, M. Schumacher, M. Diederich, T.J. Somers-Edgar, and L. Larsen Bioorg. Med. Chem. 18 2010 6701
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 6701
- Yadav, B.¹ Taurin, S.² Rosengren, R.J.³ Schumacher, M.⁴ Diederich, M.⁵ Somers-Edgar, T.J.⁶ Larsen, L.⁷

38
- 84871000767
- U. Das, R.K. Sharma, and J.R. Dimmock Curr. Med. Chem. 2009 2001 16
- (2001) Curr. Med. Chem. , vol.2009 , pp. 16
- Das, U.¹ Sharma, R.K.² Dimmock, J.R.³

39
- 2942726181
- B.K. Adams, E.M. Ferstl, M.C. Davis, M. Herold, S. Kurtkaya, R.F. Camalier, M.G. Hollingshead, G. Kaur, E.A. Sausville, F.R. Rickles, J.P. Snyder, D.C. Liotta, and M. Shoji Bioorg. Med. Chem. 12 2004 3871
- (2004) Bioorg. Med. Chem. , vol.12 , pp. 3871
- Adams, B.K.¹ Ferstl, E.M.² Davis, M.C.³ Herold, M.⁴ Kurtkaya, S.⁵ Camalier, R.F.⁶ Hollingshead, M.G.⁷ Kaur, G.⁸ Sausville, E.A.⁹ Rickles, F.R.¹⁰ Snyder, J.P.¹¹ Liotta, D.C.¹² Shoji, M.¹³

40
- 70349138396
- P. Lagisetty, D.R. Powell, and V. Awasthi J. Mol. Struct. 936 2009 23
- (2009) J. Mol. Struct. , vol.936 , pp. 23
- Lagisetty, P.¹ Powell, D.R.² Awasthi, V.³

41
- 79957443191
- A.M. Katsori, M. Chatzopoulou, K. Dimas, C. Kontogiorgis, A. Patsilinakos, T. Trangas, and D. Hadjipavlou-Litina Eur. J. Med. Chem. 46 2011 2722
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 2722
- Katsori, A.M.¹ Chatzopoulou, M.² Dimas, K.³ Kontogiorgis, C.⁴ Patsilinakos, A.⁵ Trangas, T.⁶ Hadjipavlou-Litina, D.⁷

42
- 77955471499
- P. Lagisetty, P. Vilekar, K. Sahoo, S. Anant, and V. Awasthi Bioorg. Med. Chem. 18 2010 6109
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 6109
- Lagisetty, P.¹ Vilekar, P.² Sahoo, K.³ Anant, S.⁴ Awasthi, V.⁵

43
- 75849164993
- M.V. Makarov, E.S. Leonova, E.Y. Rybalkina, P. Tongwa, V.N. Khrustalev, T.V. Timofeeva, and I.L. Odinets Eur. J. Med. Chem. 45 2010 992
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 992
- Makarov, M.V.¹ Leonova, E.S.² Rybalkina, E.Y.³ Tongwa, P.⁴ Khrustalev, V.N.⁵ Timofeeva, T.V.⁶ Odinets, I.L.⁷

44
- 62149086696
- G. Liang, L. Shao, Y. Wang, C. Zhao, Y. Chu, J. Xiao, Y. Zhao, X. Li, and S. Yang Bioorg. Med. Chem. 17 2009 2623
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 2623
- Liang, G.¹ Shao, L.² Wang, Y.³ Zhao, C.⁴ Chu, Y.⁵ Xiao, J.⁶ Zhao, Y.⁷ Li, X.⁸ Yang, S.⁹

45
- 57649240265
- M.W. Amolins, L.B. Peterson, and B.S. Blagg Bioorg. Med. Chem. 17 2009 360
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 360
- Amolins, M.W.¹ Peterson, L.B.² Blagg, B.S.³

46
- 70349333806
- N. Aggarwal, R. Kumar, P. Dureja, and D.S. Rawat J. Agric. Food Chem. 57 2009 8520
- (2009) J. Agric. Food Chem. , vol.57 , pp. 8520
- Aggarwal, N.¹ Kumar, R.² Dureja, P.³ Rawat, D.S.⁴

47
- 72049117615
- S. Manohar, S.I. Khan, and D.S. Rawat Bioorg. Med. Chem. Lett. 20 2010 322
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 322
- Manohar, S.¹ Khan, S.I.² Rawat, D.S.³

48
- 80052421210
- M. Sharma, M.C. Joshi, V. Kumar, S.V. Malhotra, and D.S. Rawat Arch. Pharm. 344 2011 567
- (2011) Arch. Pharm. , vol.344 , pp. 567
- Sharma, M.¹ Joshi, M.C.² Kumar, V.³ Malhotra, S.V.⁴ Rawat, D.S.⁵

49
- 79958808891
- S. Manohar, S.I. Khan, and D.S. Rawat Chem. Biol. Drug Des. 78 2011 124
- (2011) Chem. Biol. Drug Des. , vol.78 , pp. 124
- Manohar, S.¹ Khan, S.I.² Rawat, D.S.³

50
- 79151483153
- M. Sharma, P. Joshi, N. Kumar, S. Joshi, R.K. Rohilla, N. Roy, and D.S. Rawat Eur. J. Med. Chem. 46 2011 480
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 480
- Sharma, M.¹ Joshi, P.² Kumar, N.³ Joshi, S.⁴ Rohilla, R.K.⁵ Roy, N.⁶ Rawat, D.S.⁷

51
- 79957461484
- N. Kumar, S.I. Khan, H. Atheaya, R. Mamgain, and D.S. Rawat Eur. J. Med. Chem. 46 2011 2816
- (2011) Eur. J. Med. Chem. , vol.46 , pp. 2816
- Kumar, N.¹ Khan, S.I.² Atheaya, H.³ Mamgain, R.⁴ Rawat, D.S.⁵

52
- 84863812396
- S. Manohar, U.C. Rajesh, S.I. Khan, B.L. Tekwani, and D.S. Rawat ACS Med. Chem. Lett. 3 2012 555
- (2012) ACS Med. Chem. Lett. , vol.3 , pp. 555
- Manohar, S.¹ Rajesh, U.C.² Khan, S.I.³ Tekwani, B.L.⁴ Rawat, D.S.⁵

53
- 34248195594
- M.C. Joshi, G.S. Bisht, and D.S. Rawat Bioorg. Med. Chem. Lett. 17 2007 3226
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 3226
- Joshi, M.C.¹ Bisht, G.S.² Rawat, D.S.³

54
- 34347396940
- G.S. Bisht, D.S. Rawat, A. Kumar, R. Kumar, and S. Pasha Bioorg. Med. Chem. Lett. 17 2007 4343
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 4343
- Bisht, G.S.¹ Rawat, D.S.² Kumar, A.³ Kumar, R.⁴ Pasha, S.⁵

55
- 60449113949
- N. Beena Kumar, R.K. Rohilla, N. Roy, and D.S. Rawat Bioorg. Med. Chem. Lett. 19 2009 1396
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 1396
- Beena Kumar, N.¹ Rohilla, R.K.² Roy, N.³ Rawat, D.S.⁴

56
- 38949142635
- H. Atheaya, S.I. Khan, R. Mamgain, and D.S. Rawat Bioorg. Med. Chem. Lett. 18 2008 1446
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 1446
- Atheaya, H.¹ Khan, S.I.² Mamgain, R.³ Rawat, D.S.⁴

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.