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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 23, 2012, Pages 7084-7086

The structural requirements of histone deacetylase inhibitors: Suberoylanilide hydroxamic acid analogs modified at the C6 position

(2) Choi, Sun Ea a Pflum, Mary Kay H a

a WAYNE STATE UNIVERSITY (United States)

Author keywords

HDAC inhibitor; Histone deacetylase; Isoform selectivity; Vorinostat

Indexed keywords

ENTINOSTAT; HISTONE DEACETYLASE; VORINOSTAT;

ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS;

ANTINEOPLASTIC AGENTS; CARBON; HELA CELLS; HISTONE DEACETYLASE 1; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HUMANS; HYDROXAMIC ACIDS; PROTEIN BINDING;

EID: 84869085767 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.09.093 Document Type: Article

Times cited : (21)

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