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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 20, 2011, Pages 6139-6142

The structural requirements of histone deacetylase inhibitors: Suberoylanilide hydroxamic acid analogs modified at the C3 position display isoform selectivity

(3) Choi, Sun Ea a Weerasinghe, Sujith V W a Pflum, Mary Kay H a

a WAYNE STATE UNIVERSITY (United States)

Author keywords

HDAC inhibitors; Histone deaceylases; Isoform selectivity; Vorinostat

Indexed keywords

ANTINEOPLASTIC AGENT; ENTINOSTAT; HISTONE DEACETYLASE; HISTONE DEACETYLASE 1; HISTONE DEACETYLASE 3; HISTONE DEACETYLASE 6; HISTONE DEACETYLASE INHIBITOR; ISOENZYME; VORINOSTAT;

ARTICLE; DRUG SELECTIVITY; ENZYME INHIBITION; HUMAN; HUMAN CELL; IC 50; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; HELA CELLS; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HUMANS; HYDROXAMIC ACIDS; NEOPLASMS; PROTEIN ISOFORMS;

EID: 80052925413 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.08.027 Document Type: Article

Times cited : (25)

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