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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 12, 2012, Pages 4189-4192

Structure and property based design, synthesis and biological evaluation of γ-lactam based HDAC inhibitors: Part II

(9) Lee, Chulho a Choi, Eunhyun a Cho, Misun a Lee, Boah a Oh, Soo Jin b Park, Song Kyu c Lee, Kiho c Kim, Hwan Mook d Han, Gyoonhee a

a Yonsei University (South Korea)

b Korea Research Institute of Bioscience and Biotechnology (KRIBB) (South Korea)

c Korea University (South Korea)

d Gachon University College of Medicine (South Korea)

Author keywords

Docking; Histone deacetylases; Inhibitor; Optimization; Property

Indexed keywords

DEPSIPEPTIDE; GAMMA LACTAM DERIVATIVE; HISTONE DEACETYLASE INHIBITOR; ROMIDEPSIN; VORINOSTAT;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL; CANCER INHIBITION; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; HYDROGEN BOND; HYDROPHOBICITY; LIPOPHILICITY;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL SURVIVAL; DRUG DESIGN; DRUG SCREENING ASSAYS, ANTITUMOR; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HUMANS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; INHIBITORY CONCENTRATION 50; LACTAMS; MODELS, MOLECULAR; MOLECULAR WEIGHT; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84861571256 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.04.045 Document Type: Article

Times cited : (20)

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