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Volumn 690, Issue 1-3, 2012, Pages 115-118

Effects of intraperitoneal administration of the GABAB receptor positive allosteric modulator 2,6-di tert-butyl-4-(2-hydroxy-2,2-dimethyl- propyl)-phenol (CGP7930) on food intake in non-deprived rats

Author keywords

Baclofen; CGP7930; Feeding; Food intake; GABAB receptor; PAM; Positive allosteric modulator

Indexed keywords

2,6 DI TERT BUTYL 4 (3 HYDROXY 2,2 DIMETHYLPROPYL)PHENOL; BACLOFEN;

EID: 84864439929     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2012.05.021     Document Type: Article
Times cited : (12)

References (30)
  • 1
    • 3042546515 scopus 로고    scopus 로고
    • Molecular structure and physiological functions of the GABAB receptor
    • B. Bettler, K. Kaupmann, J. Mosbacher, and M. Gassmann Molecular structure and physiological functions of the GABAB receptor Physiol. Rev. 84 2004 835 867
    • (2004) Physiol. Rev. , vol.84 , pp. 835-867
    • Bettler, B.1    Kaupmann, K.2    Mosbacher, J.3    Gassmann, M.4
  • 2
    • 3142685557 scopus 로고    scopus 로고
    • The hepta-helical domain of GABAB2 is activated directly by CGP7930, a positive allosteric modulator of the GABAB receptor
    • V. Binet, C. Brajont, L. LeCorre, F. Archer, J.P. Pin, and L. Prezeau The hepta-helical domain of GABAB2 is activated directly by CGP7930, a positive allosteric modulator of the GABAB receptor J. Biol. Chem. 209 2004 29085 29091
    • (2004) J. Biol. Chem. , vol.209 , pp. 29085-29091
    • Binet, V.1    Brajont, C.2    Lecorre, L.3    Archer, F.4    Pin, J.P.5    Prezeau, L.6
  • 3
    • 58549112362 scopus 로고    scopus 로고
    • B receptor agonist, baclofen, and the positive allosteric modulator, CGP7930, inhibit visceral pain-related responses to colorectal distension in rats
    • B receptor agonist, baclofen, and the positive allosteric modulator, CGP7930, inhibit visceral pain-related responses to colorectal distension in rats Neuropharmacology 56 2009 362 367
    • (2009) Neuropharmacology , vol.56 , pp. 362-367
    • Brusberg, M.1    Ravnefjord, A.2    Martinsson, R.3    Larsson, H.4    Martinez, V.5    Lindstrom, E.6
  • 4
    • 24944563848 scopus 로고    scopus 로고
    • Baclofen reduced fat intake under binge-type conditions
    • A. Buda-Levin, F.H.E. Wojnicki, and R.L. Corwin Baclofen reduced fat intake under binge-type conditions Physiol. Behav. 86 2005 176 184
    • (2005) Physiol. Behav. , vol.86 , pp. 176-184
    • Buda-Levin, A.1    Wojnicki, F.H.E.2    Corwin, R.L.3
  • 5
    • 8444232545 scopus 로고    scopus 로고
    • In vivo effectiveness of CGP7930, a positive allosteric modulator of the GABAB receptor
    • M.A. Carai, G. Colombo, and G.L. Gessa In vivo effectiveness of CGP7930, a positive allosteric modulator of the GABAB receptor Eur. J. Pharmacol. 504 2004 213 216
    • (2004) Eur. J. Pharmacol. , vol.504 , pp. 213-216
    • Carai, M.A.1    Colombo, G.2    Gessa, G.L.3
  • 6
    • 78649937126 scopus 로고    scopus 로고
    • Effects of baclofen on liquid and solid gastric emptying in rats
    • E.F. Collares, and A.M. Vinagre Effects of baclofen on liquid and solid gastric emptying in rats. Arq Gastroentrol. 47 2010 290 296
    • (2010) Arq Gastroentrol. , vol.47 , pp. 290-296
    • Collares, E.F.1    Vinagre, A.M.2
  • 7
    • 0025613615 scopus 로고
    • The effect of intracerebroventricular administration of baclofen on food intake in rats
    • I.S. Ebenezer The effect of intracerebroventricular administration of baclofen on food intake in rats NeuroReport 1 1990 73 76
    • (1990) NeuroReport , vol.1 , pp. 73-76
    • Ebenezer, I.S.1
  • 8
    • 0028961504 scopus 로고
    • Intraperitoneal administration of baclofen increases consumption of both solid and liquid diets in rats
    • I.S. Ebenezer Intraperitoneal administration of baclofen increases consumption of both solid and liquid diets in rats Eur. J. Pharmacol. 273 1995 183 185
    • (1995) Eur. J. Pharmacol. , vol.273 , pp. 183-185
    • Ebenezer, I.S.1
  • 9
    • 0029961348 scopus 로고    scopus 로고
    • The inhibitory effect of intraperitoneally administered cholecystokinin (CCK) on food intake in rats is attenuated by baclofen pretreatment
    • I.S. Ebenezer The inhibitory effect of intraperitoneally administered cholecystokinin (CCK) on food intake in rats is attenuated by baclofen pretreatment Brain Res. Bull. 41 1996 269 272
    • (1996) Brain Res. Bull. , vol.41 , pp. 269-272
    • Ebenezer, I.S.1
  • 10
    • 7444264978 scopus 로고    scopus 로고
    • B receptor agonists baclofen and 3-aminopropylphosphinic acid (3-APA) on food intake in rats
    • B receptor agonists baclofen and 3-aminopropylphosphinic acid (3-APA) on food intake in rats Methods Find. Exp. Clin. Pharmacol. 26 2004 627 630
    • (2004) Methods Find. Exp. Clin. Pharmacol. , vol.26 , pp. 627-630
    • Ebenezer, I.S.1    Patel, S.M.2
  • 11
    • 84855552005 scopus 로고    scopus 로고
    • B receptor agonist baclofen on food intake in rats measured under different feeding conditions
    • B receptor agonist baclofen on food intake in rats measured under different feeding conditions Eur. J. Pharmacol. 635 2011 129 134
    • (2011) Eur. J. Pharmacol. , vol.635 , pp. 129-134
    • Ebenezer, I.S.1    Patel, S.M.2
  • 12
    • 0026530493 scopus 로고
    • The effects of systemic administration of baclofen on food intake in rats
    • I.S. Ebenezer, and A.K. Pringle The effects of systemic administration of baclofen on food intake in rats Neuropharmacology 31 1992 39 42
    • (1992) Neuropharmacology , vol.31 , pp. 39-42
    • Ebenezer, I.S.1    Pringle, A.K.2
  • 13
    • 0347132600 scopus 로고    scopus 로고
    • Effects of gepirone on food intake in rats may depend on their motivation to eat
    • I.S. Ebenezer, and R.M. Tite Effects of gepirone on food intake in rats may depend on their motivation to eat Methods Find. Exp. Clin. Pharmacol. 25 2003 727 731
    • (2003) Methods Find. Exp. Clin. Pharmacol. , vol.25 , pp. 727-731
    • Ebenezer, I.S.1    Tite, R.M.2
  • 14
    • 78651515998 scopus 로고    scopus 로고
    • Baclofen fails to alter highly palatable food intake in hindbrain lesioned rats
    • (Abstr.)
    • G.L. Edwards, and K.G. Freeman Baclofen fails to alter highly palatable food intake in hindbrain lesioned rats Appetite 44 2005 348 (Abstr.)
    • (2005) Appetite , vol.44 , pp. 348
    • Edwards, G.L.1    Freeman, K.G.2
  • 16
    • 34548600129 scopus 로고    scopus 로고
    • Effects of GABAB receptor agents on cocaine priming, discrete contextual cue and food induced relapses
    • M. Filip, and M. Frankowska Effects of GABAB receptor agents on cocaine priming, discrete contextual cue and food induced relapses Eur. J. Pharmacol. 571 2007 166 173
    • (2007) Eur. J. Pharmacol. , vol.571 , pp. 166-173
    • Filip, M.1    Frankowska, M.2
  • 18
    • 33645236729 scopus 로고    scopus 로고
    • The GABA(B) receptor allosteric modulator CGP7930, like baclofen, reduces operant self-administration of ethanol in alcohol-preferring rats
    • J.H. Liang, F. Chen, E. Krstew, M.S. Cowen, F.Y. Carroll, D. Crawford, P.M. Beart, and A.J. Lawrence The GABA(B) receptor allosteric modulator CGP7930, like baclofen, reduces operant self-administration of ethanol in alcohol-preferring rats Neuropharmacology 50 2006 632 639
    • (2006) Neuropharmacology , vol.50 , pp. 632-639
    • Liang, J.H.1    Chen, F.2    Krstew, E.3    Cowen, M.S.4    Carroll, F.Y.5    Crawford, D.6    Beart, P.M.7    Lawrence, A.J.8
  • 19
    • 79958809012 scopus 로고    scopus 로고
    • Central regulation of feeding behavior during social isolation of rat: Evidence for the role of endogenous CART system
    • K.T. Nakhate, D.M. Kokare, P.S. Singru, and N.K. Subhedar Central regulation of feeding behavior during social isolation of rat: evidence for the role of endogenous CART system Int. J. Obes. 35 2011 773 784
    • (2011) Int. J. Obes. , vol.35 , pp. 773-784
    • Nakhate, K.T.1    Kokare, D.M.2    Singru, P.S.3    Subhedar, N.K.4
  • 20
    • 7444267899 scopus 로고    scopus 로고
    • B receptor antagonist CGP 35348 on food intake in rats
    • B receptor antagonist CGP 35348 on food intake in rats Eur. J. Pharmacol. 503 2004 89 93
    • (2004) Eur. J. Pharmacol. , vol.503 , pp. 89-93
    • Patel, S.M.1    Ebenezer, I.S.2
  • 21
    • 56949095727 scopus 로고    scopus 로고
    • B receptor agonist baclofen on food intake in rats
    • B receptor agonist baclofen on food intake in rats Eur. J. Pharmacol. 601 2008 106 110
    • (2008) Eur. J. Pharmacol. , vol.601 , pp. 106-110
    • Patel, S.1    Ebenezer, I.S.2
  • 22
    • 49849086006 scopus 로고    scopus 로고
    • B receptor agonist baclofen on food intake in rats
    • B receptor agonist baclofen on food intake in rats Eur. J. Pharmacol. 593 2008 68 72
    • (2008) Eur. J. Pharmacol. , vol.593 , pp. 68-72
    • Patel, S.1    Ebenezer, I.S.2
  • 23
    • 77952312468 scopus 로고    scopus 로고
    • B receptor agonist baclofen on food intake and body weight in rats
    • B receptor agonist baclofen on food intake and body weight in rats Eur. J. Pharmacol. 635 2010 129 134
    • (2010) Eur. J. Pharmacol. , vol.635 , pp. 129-134
    • Patel, S.M.1    Ebenezer, I.S.2
  • 24
    • 45749130575 scopus 로고    scopus 로고
    • Positive modulation of GABA(B) receptors decreased nicotine self-administration and conteracted nicotine-induced enhancement of brain reward function in rats
    • N.E. Patterson, S. Vlachou, S. Guery, W. Froestl, and A. Markou Positive modulation of GABA(B) receptors decreased nicotine self-administration and conteracted nicotine-induced enhancement of brain reward function in rats J. Pharmacol. Exp. Ther. 326 2008 306 314
    • (2008) J. Pharmacol. Exp. Ther. , vol.326 , pp. 306-314
    • Patterson, N.E.1    Vlachou, S.2    Guery, S.3    Froestl, W.4    Markou, A.5
  • 29
    • 13844275284 scopus 로고    scopus 로고
    • Mechanisms of allosteric modulation of GABAB receptors by CGP7930 and GS39783: Effects on affinities and efficacies of orthosteric ligands with distinct intrinsic properties
    • S. Urwyler, T. Gjoni, J. Koljatic, and D.S. Dupuis Mechanisms of allosteric modulation of GABAB receptors by CGP7930 and GS39783: effects on affinities and efficacies of orthosteric ligands with distinct intrinsic properties Neuropharmacology 38 2005 343 353
    • (2005) Neuropharmacology , vol.38 , pp. 343-353
    • Urwyler, S.1    Gjoni, T.2    Koljatic, J.3    Dupuis, D.S.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.