Applications of supercritical fluids to enhance the dissolution behaviors of Furosemide by generation of microparticles and solid dispersions

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 81, Issue 1, 2012, Pages 131-141

  De Zordi, Nicola ^a   Moneghini, Mariarosa ^a   Kikic, Ireneo ^a   Grassi, Mario ^a   Del Rio Castillo, Antonio Esau ^a   Solinas, Dario ^a   Bolger, Michael B ^b  

^a UNIVERSITY OF TRIESTE   (Italy)

^b Simulations Plus Inc   (United States)

Author keywords

Crospovidone; Furosemide; Mathematical modeling; Micronization; Solid dispersions; Supercritical antisolvent technology

Indexed keywords

ACETONE; ALCOHOL; CARBON DIOXIDE; CROSPOVIDONE; FUROSEMIDE; METHANOL;

ARTICLE; DISPERSION; DRUG BIOAVAILABILITY; DRUG SOLUBILITY; EVAPORATION; HYDROPHILICITY; IN VITRO STUDY; IN VIVO STUDY; MATHEMATICAL MODEL; PARTICLE SIZE; PH; PHYSICAL CHEMISTRY; PRESSURE; RAMAN SPECTROMETRY; STOMACH JUICE; SUPERCRITICAL FLUID; TEMPERATURE; X RAY POWDER DIFFRACTION;

BIOLOGICAL AVAILABILITY; CARBON DIOXIDE; CRYSTALLIZATION; DIURETICS; DRUG STABILITY; FUROSEMIDE; GASTRIC JUICE; HYDROGEN-ION CONCENTRATION; MICROSPHERES; MODELS, THEORETICAL; PARTICLE SIZE; POVIDONE; SOLUBILITY; SOLVENTS; TECHNOLOGY, PHARMACEUTICAL; TIME FACTORS;

EID: 84861092432     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2012.01.002     Document Type: Article

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