Discovery of a potent and selective GPR120 agonist

Journal of Medicinal Chemistry

Volumn 55, Issue 9, 2012, Pages 4511-4515

  Shimpukade, Bharat ^a   Hudson, Brian D ^b   Hovgaard, Christine Kiel ^a   Milligan, Graeme ^b   Ulven, Trond ^a  

^a UNIVERSITY OF SOUTHERN DENMARK   (Denmark)

^b UNIVERSITY OF GLASGOW   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

AGENTS INTERACTING WITH TRANSMITTER, HORMONE OR DRUG RECEPTORS; FATTY ACID; FREE FATTY ACID 1; G PROTEIN COUPLED RECEPTOR 120; GW 9508; LINOLENIC ACID; NCG 21; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; PROCESS OPTIMIZATION;

CELL SURVIVAL; CINNAMATES; DIABETES MELLITUS, TYPE 2; GLUCAGON-LIKE PEPTIDE 1; HEK293 CELLS; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MOLECULAR STRUCTURE; RECEPTORS, G-PROTEIN-COUPLED; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84861066914     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm300215x     Document Type: Article

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