SCOPUS 정보 검색 플랫폼

Journal of Inorganic Biochemistry

Volumn 111, Issue , 2012, Pages 1-9

Novel estradiol based metal complexes of Tc-99m

(6) Neto, Carina a Oliveira, Maria Cristina a Gano, Lurdes a Marques, Fernanda a Thiemann, Thies b Santos, Isabel a

a INSTITUTO TECNOLÓGICO E NUCLEAR (Portugal)

b UNITED ARAB EMIRATES UNIVERSITY (United Arab Emirates)

Author keywords

Breast cancer; Estrogen receptor; Rhenium; SPECT imaging; Technetium; Tricarbonyl complexes

Indexed keywords

17ALPHA [2 (HYDROXYCARBONYLMETHYLAMINOMETHYL)PYRID 5 YL ETHYNYL]ESTRA 1,3,5(10) TRIENE 3,17BETA DIOL; 17ALPHA [[N [2 (3,5 DIMETHYL 1H PYRAZOL 1 YL)ETHYL]ETHANE 1,2 DIAMINE] 4 ETHYLPHENYL] ETHYNYL ESTRA 1,3,5(10) TRIENE 3,17BETA DIOL; ESTRADIOL; ESTROGEN RECEPTOR; ETHYL 2 [(5 BROMOPYRID 2 YL)METHYLAMINO]ACETATE; METAL COMPLEX; RHENIUM; TECHNETIUM 99M; TERT BUTYL 2 (4 BROMOETHYLPHENYL) [2 (3,5 DIMETHYL 1H PYRAZOL 1 YLETHYL)AMINE]ETHYLCARBAMATE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IRRADIATION; LIPOPHILICITY; MASS SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE; RADIOCHEMISTRY; RADIOCHROMATOGRAPHY; RECEPTOR BINDING; SUBSTITUTION REACTION;

BINDING, COMPETITIVE; BREAST NEOPLASMS; CELL LINE, TUMOR; ESTRADIOL; FEMALE; HUMANS; KINETICS; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MODELS, CHEMICAL; MOLECULAR STRUCTURE; ORGANOMETALLIC COMPOUNDS; RECEPTORS, ESTROGEN; RHENIUM; TECHNETIUM;

EID: 84860528917 PISSN: 01620134 EISSN: 18733344 Source Type: Journal
DOI: 10.1016/j.jinorgbio.2012.03.001 Document Type: Article

Times cited : (20)

References (45)

1
- 0034783960
- S. Nilsson, S. Mäkelä, E. Treuter, M. Tujague, J. Thomsen, G. Andersson, E. Enmark, K. Pettersson, M. Warner, J. Gustafsson, Physiol. Rev. 81 (2001) 1535-1565.
- (2001) Physiol. Rev. , vol.81 , pp. 1535-1565
- Nilsson, S.¹ Mäkelä, S.² Treuter, E.³ Tujague, M.⁴ Thomsen, J.⁵ Andersson, G.⁶ Enmark, E.⁷ Pettersson, K.⁸ Warner, M.⁹ Gustafsson, J.¹⁰

2
- 30944469849
- J.D. Yager, N.E. Davidson, N. Engl. J. Med. 354 (2006) 270-282.
- (2006) N. Engl. J. Med. , vol.354 , pp. 270-282
- Yager, J.D.¹ Davidson, N.E.²

3
- 0027230247
- C.H. Cummins, Steroids 58 (1993) 245-259.
- (1993) Steroids , vol.58 , pp. 245-259
- Cummins, C.H.¹

4
- 0033864602
- C. Van de Wiele, F. De Vos, G. Slegers, S. Van Belle, R.A. Dierckx, Eur. J. Nucl. Med. Mol. Imaging 27 (2000) 1421-1433.
- (2000) Eur. J. Nucl. Med. Mol. Imaging , vol.27 , pp. 1421-1433
- Van De Wiele, C.¹ De Vos, F.² Slegers, G.³ Van Belle, S.⁴ Dierckx, R.A.⁵

5
- 0025251173
- M.G. Pomper, H. VanBrocklin, A.M. Thieme, R.D. Thomas, D.O. Kiesewetter, K.E. Carlson, C.J. Mathias, M.J. Welch, J.A. Katzenellenbogen, J. Med. Chem. 33 (1990) 3143-3155.
- (1990) J. Med. Chem. , vol.33 , pp. 3143-3155
- Pomper, M.G.¹ VanBrocklin, H.² Thieme, A.M.³ Thomas, R.D.⁴ Kiesewetter, D.O.⁵ Carlson, K.E.⁶ Mathias, C.J.⁷ Welch, M.J.⁸ Katzenellenbogen, J.A.⁹

6
- 0021751581
- D.O. Kiesewetter, M.R. Kilbourn, S.W. Landvatter, D.F. Heiman, J.A. Katzenellenbogen, M.J. Welch, J. Nucl. Med. 25 (1984) 1212-1221.
- (1984) J. Nucl. Med. , vol.25 , pp. 1212-1221
- Kiesewetter, D.O.¹ Kilbourn, M.R.² Landvatter, S.W.³ Heiman, D.F.⁴ Katzenellenbogen, J.A.⁵ Welch, M.J.⁶

7
- 0027336501
- H.F. VanBrocklin, K.E. Carlson, J.A. Katzenellenbogen, M.J. Welch, J. Med. Chem. 36 (1993) 1619-1629.
- (1993) J. Med. Chem. , vol.36 , pp. 1619-1629
- VanBrocklin, H.F.¹ Carlson, K.E.² Katzenellenbogen, J.A.³ Welch, M.J.⁴

8
- 0028144460
- H.F. VanBrocklin, A. Liu, M.J. Welch, J.P. O'Neil, J.A. Katzenellenbogen, Steroids 59 (1994) 34-45.
- (1994) Steroids , vol.59 , pp. 34-45
- VanBrocklin, H.F.¹ Liu, A.² Welch, M.J.³ O'Neil, J.P.⁴ Katzenellenbogen, J.A.⁵

9
- 0035996627
- Y. Seimbille, J. Rousseau, F. Bénard, C. Morin, H. Ali, G. Avvakumov, G.L. Hammond, J.E. van Lier, Steroids 67 (2002) 765-775.
- (2002) Steroids , vol.67 , pp. 765-775
- Seimbille, Y.¹ Rousseau, J.² Bénard, F.³ Morin, C.⁴ Ali, H.⁵ Avvakumov, G.⁶ Hammond, G.L.⁷ Van Lier, J.E.⁸

10
- 77955923606
- L. Huang, H. Zhu, Y. Zhang, X. Xu, W. Cui, G. Yang, Y.-M. Shen, Steroids 75 (2010) 905-911.
- (2010) Steroids , vol.75 , pp. 905-911
- Huang, L.¹ Zhu, H.² Zhang, Y.³ Xu, X.⁴ Cui, W.⁵ Yang, G.⁶ Shen, Y.-M.⁷

11
- 33745545477
- H.M. Linden, S.A. Stekhova, J.M. Link, J.R. Gralow, R.B. Livingston, G.K. Ellis, P.H. Petra, L.M. Peterson, E.K. Schubert, L.K. Dunnwald, K.A. Krohn, D.A. Mankoff, J. Clin. Oncol. 24 (2006) 2793-2799.
- (2006) J. Clin. Oncol. , vol.24 , pp. 2793-2799
- Linden, H.M.¹ Stekhova, S.A.² Link, J.M.³ Gralow, J.R.⁴ Livingston, R.B.⁵ Ellis, G.K.⁶ Petra, P.H.⁷ Peterson, L.M.⁸ Schubert, E.K.⁹ Dunnwald, L.K.¹⁰ Krohn, K.A.¹¹ Mankoff, D.A.¹²

12
- 0029979129
- J.E. Mortimer, F. Dehdashti, B.A. Siegel, J.A. Katzenellenbogen, P. Fracasso, M.J. Welch, Clin. Cancer Res. 2 (1996) 933-939.
- (1996) Clin. Cancer Res. , vol.2 , pp. 933-939
- Mortimer, J.E.¹ Dehdashti, F.² Siegel, B.A.³ Katzenellenbogen, J.A.⁴ Fracasso, P.⁵ Welch, M.J.⁶

13
- 34848825649
- L. Sundararajan, H.M. Linden, J.M. Link, K.A. Krohn, D.A. Mankoff, Semin. Nucl. Med. 37 (2007) 470-476.
- (2007) Semin. Nucl. Med. , vol.37 , pp. 470-476
- Sundararajan, L.¹ Linden, H.M.² Link, J.M.³ Krohn, K.A.⁴ Mankoff, D.A.⁵

14
- 0344760800
- M.J. Welch, C.S. Redvanly (Eds.), John Wiley & Sons, Ltd., Chichester, UK
- J.A. Katzenellenbogen, in: M.J. Welch, C.S. Redvanly (Eds.), Receptor Imaging of Tumors (Non-peptide), Handbook of Radiopharmaceuticals Radiochemistry and Applications, Vol. 25, John Wiley & Sons, Ltd., Chichester, UK, 2003, pp. 715-730.
- (2003) Receptor Imaging of Tumors (Non-peptide), Handbook of Radiopharmaceuticals Radiochemistry and Applications , vol.25 , pp. 715-730
- Katzenellenbogen, J.A.¹

15
- 0025686948
- E.J. Pavlik, K.Nelson, H.H. Gallion, J.R. vanNagell, E.S. Donaldson, W.J. Shih, J.A. Spicer, D.F. Preston, R.J. Baranczuk, D.E. Kenady, Cancer Res. 50 (1990) 7799-7805.
- (1990) Cancer Res. , vol.50 , pp. 7799-7805
- Pavlik, E.J.¹ Nelson, K.² Gallion, H.H.³ VanNagell, J.R.⁴ Donaldson, E.S.⁵ Shih, W.J.⁶ Spicer, J.A.⁷ Preston, D.F.⁸ Baranczuk, R.J.⁹ Kenady, D.E.¹⁰

16
- 50749135432
- M.J. Ribeiro-Barras, C. Foulon, J.L. Baulieu, D. Guilloteau, P. Bougnoux, J. Lansac, J.C. Besnard, Nucl. Med. Biol. 19 (1992) 263-267.
- (1992) Nucl. Med. Biol. , vol.19 , pp. 263-267
- Ribeiro-Barras, M.J.¹ Foulon, C.² Baulieu, J.L.³ Guilloteau, D.⁴ Bougnoux, P.⁵ Lansac, J.⁶ Besnard, J.C.⁷

17
- 0029664612
- L.J.M. Rijks, G.J. Boer, E. Endert, K. Bruin, J.C. Bos, P.A.P.M. Doremalen, W.G.E.J. Schoonen, A.G.M. Janssen, E.A. Royen, Eur. J. Nucl. Med. Mol. Imaging 23 (1996) 295-307.
- (1996) Eur. J. Nucl. Med. Mol. Imaging , vol.23 , pp. 295-307
- Rijks, L.J.M.¹ Boer, G.J.² Endert, E.³ Bruin, K.⁴ Bos, J.C.⁵ Doremalen, P.A.P.M.⁶ Schoonen, W.G.E.J.⁷ Janssen, A.G.M.⁸ Royen, E.A.⁹

18
- 0030907782
- L.J.M. Rijks, G.J. Boer, E. Endert, K. de Bruin, A.G.M. Janssen, E.A. van Royen, Nucl. Med. Biol. 24 (1997) 65-75.
- (1997) Nucl. Med. Biol. , vol.24 , pp. 65-75
- Rijks, L.J.M.¹ Boer, G.J.² Endert, E.³ De Bruin, K.⁴ Janssen, A.G.M.⁵ Van Royen, E.A.⁶

19
- 0034877612
- R.J. Bennink, L.J. Rijks, G. van Tienhoven, L.A. Noorduyn, A.G. Janssen, G.W. Sloof, Radiology 220 (2001) 774-779.
- (2001) Radiology , vol.220 , pp. 774-779
- Bennink, R.J.¹ Rijks, L.J.² Van Tienhoven, G.³ Noorduyn, L.A.⁴ Janssen, A.G.⁵ Sloof, G.W.⁶

20
- 0030808619
- R.K. Hom, J.A. Katzenellenbogen, Nucl. Med. Biol. 24 (1997) 485-498.
- (1997) Nucl. Med. Biol. , vol.24 , pp. 485-498
- Hom, R.K.¹ Katzenellenbogen, J.A.²

21
- 0343184053
- M.B. Skaddan, F.R. Wüst, S. Jonson, R. Syhre, M.J. Welch, H. Spies, J.A. Katzenellenbogen, Nucl. Med. Biol. 27 (2000) 269-278.
- (2000) Nucl. Med. Biol. , vol.27 , pp. 269-278
- Skaddan, M.B.¹ Wüst, F.R.² Jonson, S.³ Syhre, R.⁴ Welch, M.J.⁵ Spies, H.⁶ Katzenellenbogen, J.A.⁷

22
- 0041336761
- J.B. Arterburn, C. Corona, K.V. Rao, K.E. Carlson, J.A. Katzenellenbogen, J. Org. Chem. 68 (2003) 7063-7070.
- (2003) J. Org. Chem. , vol.68 , pp. 7063-7070
- Arterburn, J.B.¹ Corona, C.² Rao, K.V.³ Carlson, K.E.⁴ Katzenellenbogen, J.A.⁵

23
- 0242266521
- L.G. Luyt, H.M. Bigott, M.J. Welch, J.A. Katzenellenbogen, Bioorg. Med. Chem. 11 (2003) 4977-4989.
- (2003) Bioorg. Med. Chem. , vol.11 , pp. 4977-4989
- Luyt, L.G.¹ Bigott, H.M.² Welch, M.J.³ Katzenellenbogen, J.A.⁴

24
- 0026706764
- H. El Amouri, A. Vessieres, D. Vichard, S. Top, M. Gruselle, G. Jaouen, J. Med. Chem. 35 (1992) 3130-3135.
- (1992) J. Med. Chem. , vol.35 , pp. 3130-3135
- El Amouri, H.¹ Vessieres, A.² Vichard, D.³ Top, S.⁴ Gruselle, M.⁵ Jaouen, G.⁶

25
- 0039272909
- G. Jaouen, A. Vessieres, I.S. Butler, Acc. Chem. Res. 26 (1993) 361-369.
- (1993) Acc. Chem. Res. , vol.26 , pp. 361-369
- Jaouen, G.¹ Vessieres, A.² Butler, I.S.³

26
- 0029145533
- S. Top, H. El Hafa, A. Vessieres, J. Quivy, J. Vaissermann, D.W. Hughes, M.J. McGlinchey, J.-P. Mornon, E. Thoreau, G. Jaouen, J. Am. Chem. Soc. 117 (1995) 8372-8380.
- (1995) J. Am. Chem. Soc. , vol.117 , pp. 8372-8380
- Top, S.¹ El Hafa, H.² Vessieres, A.³ Quivy, J.⁴ Vaissermann, J.⁵ Hughes, D.W.⁶ McGlinchey, M.J.⁷ Mornon, J.-P.⁸ Thoreau, E.⁹ Jaouen, G.¹⁰

27
- 0039710691
- F. Wüst, K.E. Carlson, J.A. Katzenellenbogen, H. Spies, B. Johannsen, Steroids 63 (1998) 665-671.
- (1998) Steroids , vol.63 , pp. 665-671
- Wüst, F.¹ Carlson, K.E.² Katzenellenbogen, J.A.³ Spies, H.⁴ Johannsen, B.⁵

28
- 0028025435
- M. Wenzel, C. Klinge, J. Label. Compd. Radiopharm. 34 (1994) 981-987.
- (1994) J. Label. Compd. Radiopharm. , vol.34 , pp. 981-987
- Wenzel, M.¹ Klinge, C.²

29
- 0035973694
- A. Jackson, J. Davis, R.J. Pither, A. Rodger, M.J. Hannon, Inorg. Chem. 40 (2001) 3964-3973.
- (2001) Inorg. Chem. , vol.40 , pp. 3964-3973
- Jackson, A.¹ Davis, J.² Pither, R.J.³ Rodger, A.⁴ Hannon, M.J.⁵

30
- 0345440144
- M.B. Skaddan, F.R.Wust, J.A. Katzenellenbogen, J. Org. Chem. 64 (1999) 8108-8121.
- (1999) J. Org. Chem. , vol.64 , pp. 8108-8121
- Skaddan, M.B.¹ Wust, F.R.² Katzenellenbogen, J.A.³

31
- 33751004697
- C. Ramesh, B. Bryant, T. Nayak, C.M. Revankar, T. Anderson, K.E. Carlson, J.A. Katzenellenbogen, L.A. Sklar, J.P. Norenberg, E.R. Prossnitz, J.B. Arterburn, J. Am. Chem. Soc. 128 (2006) 14476-14477.
- (2006) J. Am. Chem. Soc. , vol.128 , pp. 14476-14477
- Ramesh, C.¹ Bryant, B.² Nayak, T.³ Revankar, C.M.⁴ Anderson, T.⁵ Carlson, K.E.⁶ Katzenellenbogen, J.A.⁷ Sklar, L.A.⁸ Norenberg, J.P.⁹ Prossnitz, E.R.¹⁰ Arterburn, J.B.¹¹

32
- 44849115355
- T.K. Nayak, H.J. Hathaway, C. Ramesh, J.B. Arterburn, D. Dai, L.A. Sklar, J.P. Norenberg, E.R. Prossnitz, J. Nucl. Med. 49 (2008) 978-986.
- (2008) J. Nucl. Med. , vol.49 , pp. 978-986
- Nayak, T.K.¹ Hathaway, H.J.² Ramesh, C.³ Arterburn, J.B.⁴ Dai, D.⁵ Sklar, L.A.⁶ Norenberg, J.P.⁷ Prossnitz, E.R.⁸

33
- 4544281766
- N. Lazarova, S. James, J. Babich, J. Zubieta, Inorg. Chem. Commun. 7 (2004) 1023-1026.
- (2004) Inorg. Chem. Commun. , vol.7 , pp. 1023-1026
- Lazarova, N.¹ James, S.² Babich, J.³ Zubieta, J.⁴

34
- 0021445407
- D.E. Troutner, W.A. Volkert, T.J. Hoffman, R.A. Holmes, Appl. Radiat. Isot. 35 (1984) 467-470.
- (1984) Appl. Radiat. Isot. , vol.35 , pp. 467-470
- Troutner, D.E.¹ Volkert, W.A.² Hoffman, T.J.³ Holmes, R.A.⁴

35
- 33646048615
- X.-R. Jiang, J. Walter Sowell, B.T. Zhu, Steroids 71 (2006) 334-342.
- (2006) Steroids , vol.71 , pp. 334-342
- Jiang, X.-R.¹ Walter Sowell, J.² Zhu, B.T.³

36
- 0018826511
- R.B. Hochberg, W. Rosner, Proc. Natl. Acad. Sci. U. S. A. 77 (1980) 328-332.
- (1980) Proc. Natl. Acad. Sci. U. S. A. , vol.77 , pp. 328-332
- Hochberg, R.B.¹ Rosner, W.²

37
- 33745866583
- S. Alves, J.D.G. Correia, I. Santos, B. Veerendra, G.L. Sieckman, T.J. Hoffman, T.L. Rold, S.D. Figueroa, L. Retzloff, J. McCrate, A. Prasanphanich, C.J. Smith, Nucl. Med. Biol. 33 (2006) 625-634.
- (2006) Nucl. Med. Biol. , vol.33 , pp. 625-634
- Alves, S.¹ Correia, J.D.G.² Santos, I.³ Veerendra, B.⁴ Sieckman, G.L.⁵ Hoffman, T.J.⁶ Rold, T.L.⁷ Figueroa, S.D.⁸ Retzloff, L.⁹ McCrate, J.¹⁰ Prasanphanich, A.¹¹ Smith, C.J.¹²

38
- 0037153792
- S. Alves, A. Paulo, J.D.G. Correia, A. Domingos, I. Santos, J. Chem. Soc. Dalton Trans. 24 (2002) 4714-4719.
- (2002) J. Chem. Soc. Dalton Trans. , vol.24 , pp. 4714-4719
- Alves, S.¹ Paulo, A.² Correia, J.D.G.³ Domingos, A.⁴ Santos, I.⁵

39
- 0038143208
- A. Stichelberger, R. Waibel, C. Dumas, P.A. Schubiger, R. Schibli, Nucl. Med. Biol. 30 (2003) 465-470.
- (2003) Nucl. Med. Biol. , vol.30 , pp. 465-470
- Stichelberger, A.¹ Waibel, R.² Dumas, C.³ Schubiger, P.A.⁴ Schibli, R.⁵

40
- 0344026346
- P. López, C.G. Seipelt, P. Merkling, L. Sturz, J. Álvarez, A. Dölle, M.D. Zeidler, S. Cerdán, P. Ballesteros, Bioorg. Med. Chem. 7 (1999) 517-527.
- (1999) Bioorg. Med. Chem. , vol.7 , pp. 517-527
- López, P.¹ Seipelt, C.G.² Merkling, P.³ Sturz, L.⁴ Álvarez, J.⁵ Dölle, A.⁶ Zeidler, M.D.⁷ Cerdán, S.⁸ Ballesteros, P.⁹

41
- 33947727055
- R. Chinchilla, C. Näjera, Chem. Rev. 107 (2007) 874-922.
- (2007) Chem. Rev. , vol.107 , pp. 874-922
- Chinchilla, R.¹ Näjera, C.²

42
- 0038038606
- F.R. Wüst, T. Kniess, J. Label. Compd. Radiopharm. 46 (2003) 699-713.
- (2003) J. Label. Compd. Radiopharm. , vol.46 , pp. 699-713
- Wüst, F.R.¹ Kniess, T.²

43
- 0034030754
- R. Schibli, R. Bella, R. Alberto, E. Garcia-Garayoa, K. Ortner, U. Abram, P.A. Schubiger, Bioconjug. Chem. 11 (2000) 345-351.
- (2000) Bioconjug. Chem. , vol.11 , pp. 345-351
- Schibli, R.¹ Bella, R.² Alberto, R.³ Garcia-Garayoa, E.⁴ Ortner, K.⁵ Abram, U.⁶ Schubiger, P.A.⁷

44
- 15244347266
- S. Alves, A. Paulo, J.D.G. Correia, L. Gano, C.J. Smith, T.J. Hoffman, I. Santos, Bioconjug. Chem. 16 (2005) 438-449.
- (2005) Bioconjug. Chem. , vol.16 , pp. 438-449
- Alves, S.¹ Paulo, A.² Correia, J.D.G.³ Gano, L.⁴ Smith, C.J.⁵ Hoffman, T.J.⁶ Santos, I.⁷

45
- 79955572936
- L. Gano, F. Mendes, S. Cunha, C. Fernandes, A. Paulo, I. Santos, Q. J. Nucl. Med. Mol. Imaging 54 (2010) 10-11.
- (2010) Q. J. Nucl. Med. Mol. Imaging , vol.54 , pp. 10-11
- Gano, L.¹ Mendes, F.² Cunha, S.³ Fernandes, C.⁴ Paulo, A.⁵ Santos, I.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.