-
1
-
-
0030711065
-
Tacrolimus. An update of its pharmacology and clinical efficacy in the management of organ transplantation
-
Spencer, C. M., Goa, K. L. and Gillis, J. C.: Tacrolimus. An update of its pharmacology and clinical efficacy in the management of organ transplantation. Drugs, 54: 925-975 (1997).
-
(1997)
Drugs
, vol.54
, pp. 925-975
-
-
Spencer, C.M.1
Goa, K.L.2
Gillis, J.C.3
-
2
-
-
0029586398
-
Clinical pharmacokinetics of tacrolimus
-
Venkataramanan, R., Swaminathan, A., Prasad, T., Jain, A., Zuckerman, S., Warty, V., McMichael, J., Lever, J., Burckart, G. and Starzl, T.: Clinical pharmacokinetics of tacrolimus. Clin. Pharmacokinet., 29: 404-430 (1995).
-
(1995)
Clin. Pharmacokinet
, vol.29
, pp. 404-430
-
-
Venkataramanan, R.1
Swaminathan, A.2
Prasad, T.3
Jain, A.4
Zuckerman, S.5
Warty, V.6
McMichael, J.7
Lever, J.8
Burckart, G.9
Starzl, T.10
-
3
-
-
0026681640
-
In vitro metabolism of FK-506 in rat, rabbit, and human liver microsomes: Identification of a major metabolite and of cytochrome P450 3A as the major enzymes responsible for its metabolism
-
Vincent, S. H., Karanam, B. V., Painter, S. K. and Chiu, S. H.: In vitro metabolism of FK-506 in rat, rabbit, and human liver microsomes: identification of a major metabolite and of cytochrome P450 3A as the major enzymes responsible for its metabolism. Arch. Biochem. Biophys., 294: 454-460 (1992).
-
(1992)
Arch. Biochem. Biophys
, vol.294
, pp. 454-460
-
-
Vincent, S.H.1
Karanam, B.V.2
Painter, S.K.3
Chiu, S.H.4
-
4
-
-
23044476217
-
Contribution of CYP3A5 to the in vitro hepatic clearance of tacrolimus
-
Kamdem, L. K., Streit, F., Zanger, U. M., Brockmöller, J., Oellerich, M., Armstrong, V. W. and Wojnowski, L.: Contribution of CYP3A5 to the in vitro hepatic clearance of tacrolimus. Clin. Chem., 51: 1374-1381 (2005).
-
(2005)
Clin. Chem
, vol.51
, pp. 1374-1381
-
-
Kamdem, L.K.1
Streit, F.2
Zanger, U.M.3
Brockmöller, J.4
Oellerich, M.5
Armstrong, V.W.6
Wojnowski, L.7
-
5
-
-
0028295725
-
Metabolism of FK506, a potent immunosuppressive agent, by cytochrome P450 3A enzymes in rat, dog and human liver microsomes
-
Shiraga, T., Matsuda, H., Nagase, K., Iwasaki, K., Noda, K., Yamazaki, H., Shimada, T. and Funae, Y.: Metabolism of FK506, a potent immunosuppressive agent, by cytochrome P450 3A enzymes in rat, dog and human liver microsomes. Biochem. Pharmacol., 47: 727-735 (1994).
-
(1994)
Biochem. Pharmacol
, vol.47
, pp. 727-735
-
-
Shiraga, T.1
Matsuda, H.2
Nagase, K.3
Iwasaki, K.4
Noda, K.5
Yamazaki, H.6
Shimada, T.7
Funae, Y.8
-
6
-
-
0029560982
-
Metabolism of the immunosuppressant tacrolimus in the small intestine: Cytochrome P450, drug interactions, and interindividual variability
-
Lampen, A., Christians, U., Guengerich, F. P., Watkins, P. B., Kolars, J. C., Bader, A., Gonschior, A. K., Dralle, H., Hackbarth, I. and Sewing, K. F.: Metabolism of the immunosuppressant tacrolimus in the small intestine: cytochrome P450, drug interactions, and interindividual variability. Drug Metab. Dispos., 23: 1315-1324 (1995).
-
(1995)
Drug Metab. Dispos
, vol.23
, pp. 1315-1324
-
-
Lampen, A.1
Christians, U.2
Guengerich, F.P.3
Watkins, P.B.4
Kolars, J.C.5
Bader, A.6
Gonschior, A.K.7
Dralle, H.8
Hackbarth, I.9
Sewing, K.F.10
-
7
-
-
0027418815
-
Human P-glycoprotein transports cyclosporin A and FK506
-
Saeki, T., Ueda, K., Tanigawara, Y., Hori, R. and Komano, T.: Human P-glycoprotein transports cyclosporin A and FK506. J. Biol. Chem., 268: 6077-6080 (1993).
-
(1993)
J. Biol. Chem
, vol.268
, pp. 6077-6080
-
-
Saeki, T.1
Ueda, K.2
Tanigawara, Y.3
Hori, R.4
Komano, T.5
-
8
-
-
26444597593
-
Concomitant clotrimazole therapy more than doubles the relative oral bioavailability of tacrolimus
-
Vasquez, E. M., Shin, G. P., Sifontis, N. and Benedetti, E.: Concomitant clotrimazole therapy more than doubles the relative oral bioavailability of tacrolimus. Ther. Drug Monit., 27: 587-591 (2005).
-
(2005)
Ther. Drug Monit
, vol.27
, pp. 587-591
-
-
Vasquez, E.M.1
Shin, G.P.2
Sifontis, N.3
Benedetti, E.4
-
9
-
-
0035093640
-
Clotrimazole increases tacrolimus blood levels: A drug interaction in kidney transplant patients
-
Vasquez, E. M., Pollak, R. and Benedetti, E.: Clotrimazole increases tacrolimus blood levels: a drug interaction in kidney transplant patients. Clin. Transplant., 15: 95-99 (2001).
-
(2001)
Clin. Transplant
, vol.15
, pp. 95-99
-
-
Vasquez, E.M.1
Pollak, R.2
Benedetti, E.3
-
10
-
-
0345700744
-
Pomelo-induced increase in the blood level of tacrolimus in a renal transplant patient
-
Egashira, K., Fukuda, E., Onga, T., Yogi, Y., Matsuya, F., Koyabu, N., Ohtani, H. and Sawada, Y.: Pomelo-induced increase in the blood level of tacrolimus in a renal transplant patient. Transplantation, 75: 1057 (2003).
-
(2003)
Transplantation
, vol.75
, pp. 1057
-
-
Egashira, K.1
Fukuda, E.2
Onga, T.3
Yogi, Y.4
Matsuya, F.5
Koyabu, N.6
Ohtani, H.7
Sawada, Y.8
-
11
-
-
3242699473
-
Inhibitory effects of pomelo on the metabolism of tacrolimus and the activities of CYP3A4 and P-glycoprotein
-
Egashira, K., Ohtani, H., Itoh, S., Koyabu, N., Tsujimoto, M., Murakami, H. and Sawada, Y.: Inhibitory effects of pomelo on the metabolism of tacrolimus and the activities of CYP3A4 and P-glycoprotein. Drug Metab. Dispos., 32: 828-833 (2004).
-
(2004)
Drug Metab. Dispos
, vol.32
, pp. 828-833
-
-
Egashira, K.1
Ohtani, H.2
Itoh, S.3
Koyabu, N.4
Tsujimoto, M.5
Murakami, H.6
Sawada, Y.7
-
12
-
-
78751550662
-
Effects of mace and nutmeg on human cytochrome P450 3A4 and 2C9 activity
-
Kimura, Y., Ito, H. and Hatano, T.: Effects of mace and nutmeg on human cytochrome P450 3A4 and 2C9 activity. Biol. Pharm. Bull., 33: 1977-1982 (2010).
-
(2010)
Biol. Pharm. Bull
, vol.33
, pp. 1977-1982
-
-
Kimura, Y.1
Ito, H.2
Hatano, T.3
-
13
-
-
0021077291
-
A nonlinear least squares program based on differential equations, MULTI (RUNGE), for microcomputers
-
Yamaoka, K. and Nakagawa, T.: A nonlinear least squares program based on differential equations, MULTI (RUNGE), for microcomputers. J. Pharmacobiodyn., 6: 595-606 (1983).
-
(1983)
J. Pharmacobiodyn
, vol.6
, pp. 595-606
-
-
Yamaoka, K.1
Nakagawa, T.2
-
14
-
-
0018111355
-
Statistical moments in pharmacokinetics
-
Yamaoka, K., Nakagawa, T. and Uno, T.: Statistical moments in pharmacokinetics. J. Pharmacokinet. Biopharm., 6: 547-558 (1978).
-
(1978)
J. Pharmacokinet. Biopharm
, vol.6
, pp. 547-558
-
-
Yamaoka, K.1
Nakagawa, T.2
Uno, T.3
-
15
-
-
0043128579
-
Time course of recovery of cytochrome p450 3A function after single doses of grapefruit juice
-
Greenblatt, D. J., von Moltke, L. L., Harmatz, J. S., Chen, G., Weemhoff, J. L., Jen, C., Kelley, C. J., LeDuc, B. W. and Zinny, M. A.: Time course of recovery of cytochrome p450 3A function after single doses of grapefruit juice. Clin. Pharmacol. Ther., 74: 121-129 (2003).
-
(2003)
Clin. Pharmacol. Ther
, vol.74
, pp. 121-129
-
-
Greenblatt, D.J.1
von Moltke, L.L.2
Harmatz, J.S.3
Chen, G.4
Weemhoff, J.L.5
Jen, C.6
Kelley, C.J.7
Leduc, B.W.8
Zinny, M.A.9
-
16
-
-
0026099498
-
Interaction of citrus juices with felodipine and nifedipine
-
Bailey, D. G., Spence, J. D., Munoz, C. and Arnold, J. M.: Interaction of citrus juices with felodipine and nifedipine. Lancet, 337: 268-269 (1991).
-
(1991)
Lancet
, vol.337
, pp. 268-269
-
-
Bailey, D.G.1
Spence, J.D.2
Munoz, C.3
Arnold, J.M.4
-
17
-
-
0034468612
-
Effects of grapefruit juice on the stereoselective disposition of nicardipine in humans: Evidence for dominant presystemic elimination at the gut site
-
Uno, T., Ohkubo, T., Sugawara, K., Higashiyama, A., Motomura, S. and Ishizaki, T.: Effects of grapefruit juice on the stereoselective disposition of nicardipine in humans: evidence for dominant presystemic elimination at the gut site. Eur. J. Clin. Pharmacol., 56: 643-649 (2000).
-
(2000)
Eur. J. Clin. Pharmacol
, vol.56
, pp. 643-649
-
-
Uno, T.1
Ohkubo, T.2
Sugawara, K.3
Higashiyama, A.4
Motomura, S.5
Ishizaki, T.6
-
18
-
-
0033736174
-
Duration of effect of grapefruit juice on the pharmacokinetics of the CYP3A4 substrate simvastatin
-
Lilja, J. J., Kivistö, K. T. and Neuvonen, P. J.: Duration of effect of grapefruit juice on the pharmacokinetics of the CYP3A4 substrate simvastatin. Clin. Pharmacol. Ther., 68: 384-390 (2000).
-
(2000)
Clin. Pharmacol. Ther
, vol.68
, pp. 384-390
-
-
Lilja, J.J.1
Kivistö, K.T.2
Neuvonen, P.J.3
-
19
-
-
27444434929
-
Effects of grapefruit juice on the pharmacokinetics of pitavastatin and atorvastatin
-
Ando, H., Tsuruoka, S., Yanagihara, H., Sugimoto, K., Miyata, M., Yamazoe, Y., Takamura, T., Kaneko, S. and Fujimura, A.: Effects of grapefruit juice on the pharmacokinetics of pitavastatin and atorvastatin. Br. J. Clin. Pharmacol., 60: 494-497 (2005).
-
(2005)
Br. J. Clin. Pharmacol
, vol.60
, pp. 494-497
-
-
Ando, H.1
Tsuruoka, S.2
Yanagihara, H.3
Sugimoto, K.4
Miyata, M.5
Yamazoe, Y.6
Takamura, T.7
Kaneko, S.8
Fujimura, A.9
-
20
-
-
0034464046
-
The effects of grapefruit juice on the pharmacokinetics of erythromycin
-
Kanazawa, S., Ohkubo, T. and Sugawara, K.: The effects of grapefruit juice on the pharmacokinetics of erythromycin. Eur. J. Clin. Pharmacol., 56: 799-803 (2001).
-
(2001)
Eur. J. Clin. Pharmacol
, vol.56
, pp. 799-803
-
-
Kanazawa, S.1
Ohkubo, T.2
Sugawara, K.3
-
21
-
-
0031908050
-
Grapefruit juice enhances the bioavailability of the HIV protease inhibitor saquinavir in man
-
Kupferschmidt, H. H., Fattinger, K. E., Ha, H. R., Follath, F. and Krähenbühl, S.: Grapefruit juice enhances the bioavailability of the HIV protease inhibitor saquinavir in man. Br. J. Clin. Pharmacol., 45: 355-359 (1998).
-
(1998)
Br. J. Clin. Pharmacol
, vol.45
, pp. 355-359
-
-
Kupferschmidt, H.H.1
Fattinger, K.E.2
Ha, H.R.3
Follath, F.4
Krähenbühl, S.5
-
22
-
-
69249230842
-
Co-administration of grapefruit juice increases bioavailability of tacrolimus in liver transplant patients: A prospective study
-
Liu, C., Shang, Y. F., Zhang, X. F., Zhang, X. G., Wang, B., Wu, Z., Liu, X. M., Yu, L., Ma, F. and Lv, Y.: Co-administration of grapefruit juice increases bioavailability of tacrolimus in liver transplant patients: a prospective study. Eur. J. Clin. Pharmacol., 65: 881-885 (2009).
-
(2009)
Eur. J. Clin. Pharmacol
, vol.65
, pp. 881-885
-
-
Liu, C.1
Shang, Y.F.2
Zhang, X.F.3
Zhang, X.G.4
Wang, B.5
Wu, Z.6
Liu, X.M.7
Yu, L.8
Ma, F.9
Lv, Y.10
-
23
-
-
0029055363
-
Disposition of intravenous and oral cyclosporine after administration with grapefruit juice
-
Ducharme, M. P., Warbasse, L. H. and Edwards, D. J.: Disposition of intravenous and oral cyclosporine after administration with grapefruit juice. Clin. Pharmacol. Ther., 57: 485-491 (1995).
-
(1995)
Clin. Pharmacol. Ther
, vol.57
, pp. 485-491
-
-
Ducharme, M.P.1
Warbasse, L.H.2
Edwards, D.J.3
-
24
-
-
0031790854
-
Inhibition of vinblastine efflux mediated by P-glycoprotein by grapefruit juice components in caco-2 cells
-
Takanaga, H., Ohnishi, A., Matsuo, H. and Sawada, Y.: Inhibition of vinblastine efflux mediated by P-glycoprotein by grapefruit juice components in caco-2 cells. Biol. Pharm. Bull., 21: 1062-1066 (1998).
-
(1998)
Biol. Pharm. Bull
, vol.21
, pp. 1062-1066
-
-
Takanaga, H.1
Ohnishi, A.2
Matsuo, H.3
Sawada, Y.4
-
25
-
-
0033913305
-
Effect of furanocoumarin derivatives in grapefruit juice on the uptake of vinblastine by Caco-2 cells and on the activity of cytochrome P450 3A4
-
Ohnishi, A., Matsuo, H., Yamada, S., Takanaga, H., Morimoto, S., Shoyama, Y., Ohtani, H. and Sawada, Y.: Effect of furanocoumarin derivatives in grapefruit juice on the uptake of vinblastine by Caco-2 cells and on the activity of cytochrome P450 3A4. Br. J. Pharmacol., 130: 1369-1377 (2000).
-
(2000)
Br. J. Pharmacol
, vol.130
, pp. 1369-1377
-
-
Ohnishi, A.1
Matsuo, H.2
Yamada, S.3
Takanaga, H.4
Morimoto, S.5
Shoyama, Y.6
Ohtani, H.7
Sawada, Y.8
-
26
-
-
0031001463
-
Effects of grapefruit juice ingestion-pharmacokinetics and haemodynamics of intravenously and orally administered felodipine in healthy men
-
Lundahl, J., Regårdh, C. G., Edgar, B. and Johnsson, G.: Effects of grapefruit juice ingestion-pharmacokinetics and haemodynamics of intravenously and orally administered felodipine in healthy men. Eur. J. Clin. Pharmacol., 52: 139-145 (1997).
-
(1997)
Eur. J. Clin. Pharmacol
, vol.52
, pp. 139-145
-
-
Lundahl, J.1
Regårdh, C.G.2
Edgar, B.3
Johnsson, G.4
-
27
-
-
0031830305
-
Grapefruit juice-drug interactions
-
Bailey, D. G., Malcolm, J., Arnold, O. and Spence, J. D.: Grapefruit juice-drug interactions. Br. J. Clin. Pharmacol., 46: 101-110 (1998).
-
(1998)
Br. J. Clin. Pharmacol
, vol.46
, pp. 101-110
-
-
Bailey, D.G.1
Malcolm, J.2
Arnold, O.3
Spence, J.D.4
-
28
-
-
0342868292
-
Role of furanocoumarin derivatives on grapefruit juice-mediated inhibition of human CYP3A activity
-
Guo, L. Q., Fukuda, K., Ohta, T. and Yamazoe, Y.: Role of furanocoumarin derivatives on grapefruit juice-mediated inhibition of human CYP3A activity. Drug Metab. Dispos., 28: 766-771 (2000).
-
(2000)
Drug Metab. Dispos
, vol.28
, pp. 766-771
-
-
Guo, L.Q.1
Fukuda, K.2
Ohta, T.3
Yamazoe, Y.4
-
29
-
-
0030482468
-
Identification of 6',7'-dihydroxybergamottin, a cytochrome P450 inhibitor, in grapefruit juice
-
Edwards, D. J., Bellevue, F. H., 3rd and Woster, P. M.: Identification of 6',7'-dihydroxybergamottin, a cytochrome P450 inhibitor, in grapefruit juice. Drug Metab. Dispos., 24: 1287-1290 (1996).
-
(1996)
Drug Metab. Dispos
, vol.24
, pp. 1287-1290
-
-
Edwards, D.J.1
Bellevue 3rd., F.H.2
Woster, P.M.3
-
30
-
-
33749430489
-
Does a kampo medicine containing schisandra fruit affect pharmacokinetics of nifedipine like grapefruit juice?
-
Makino, T., Mizuno, F. and Mizukami, H.: Does a kampo medicine containing schisandra fruit affect pharmacokinetics of nifedipine like grapefruit juice? Biol. Pharm. Bull., 29: 2065-2069 (2006).
-
(2006)
Biol. Pharm. Bull
, vol.29
, pp. 2065-2069
-
-
Makino, T.1
Mizuno, F.2
Mizukami, H.3
-
31
-
-
0035076745
-
Ginger for nausea and vomiting in pregnancy: Randomized, double-masked, placebocontrolled trial
-
Vutyavanich, T., Kraisarin, T. and Ruangsri, R.: Ginger for nausea and vomiting in pregnancy: randomized, double-masked, placebocontrolled trial. Obstet. Gynecol., 97: 577-582 (2001).
-
(2001)
Obstet. Gynecol
, vol.97
, pp. 577-582
-
-
Vutyavanich, T.1
Kraisarin, T.2
Ruangsri, R.3
-
32
-
-
0037371099
-
Effects of ginger on motion sickness and gastric slow-wave dysrhythmias induced by circular vection
-
Lien, H. C., Sun, W. M., Chen, Y. H., Kim, H., Hasler, W. and Owyang, C.: Effects of ginger on motion sickness and gastric slow-wave dysrhythmias induced by circular vection. Am. J. Physiol. Gastrointest. Liver Physiol., 284: G481-G489 (2003).
-
(2003)
Am. J. Physiol. Gastrointest. Liver Physiol
, vol.284
-
-
Lien, H.C.1
Sun, W.M.2
Chen, Y.H.3
Kim, H.4
Hasler, W.5
Owyang, C.6
-
33
-
-
0037103569
-
Modulation of P-glycoprotein expression and function by curcumin in multidrug-resistant human KB cells
-
Anuchapreeda, S., Leechanachai, P., Smith, M. M., Ambudkar, S. V. and Limtrakul, P. N.: Modulation of P-glycoprotein expression and function by curcumin in multidrug-resistant human KB cells. Biochem. Pharmacol., 64: 573-582 (2002).
-
(2002)
Biochem. Pharmacol
, vol.64
, pp. 573-582
-
-
Anuchapreeda, S.1
Leechanachai, P.2
Smith, M.M.3
Ambudkar, S.V.4
Limtrakul, P.N.5
-
34
-
-
46449099725
-
Effects of spice constituents on P-glycoprotein-mediated transport and CYP3A4-mediated metabolism in vitro
-
Zhang, W. and Lim, L. Y.: Effects of spice constituents on P-glycoprotein-mediated transport and CYP3A4-mediated metabolism in vitro. Drug Metab. Dispos., 36: 1283-1290 (2008).
-
(2008)
Drug Metab. Dispos
, vol.36
, pp. 1283-1290
-
-
Zhang, W.1
Lim, L.Y.2
-
35
-
-
33845937786
-
Impact of curcumininduced changes in P-glycoprotein and CYP3A expression on the pharmacokinetics of peroral celiprolol and midazolam in rats
-
Zhang, W., Tan, T. M. and Lim, L. Y.: Impact of curcumininduced changes in P-glycoprotein and CYP3A expression on the pharmacokinetics of peroral celiprolol and midazolam in rats. Drug Metab. Dispos., 35: 110-115 (2007).
-
(2007)
Drug Metab. Dispos
, vol.35
, pp. 110-115
-
-
Zhang, W.1
Tan, T.M.2
Lim, L.Y.3
-
36
-
-
70350635146
-
Species-dependent hepatic metabolism of immunosuppressive agent tacrolimus (FK-506)
-
Tata, P. N., Subbotina, N., Burckart, G. J., Muddiman, D. C., Gusev, A. I., Hercules, D. M., Starzl, T. E. and Venkataramanan, R.: Species-dependent hepatic metabolism of immunosuppressive agent tacrolimus (FK-506). Xenobiotica, 39: 757-765 (2009).
-
(2009)
Xenobiotica
, vol.39
, pp. 757-765
-
-
Tata, P.N.1
Subbotina, N.2
Burckart, G.J.3
Muddiman, D.C.4
Gusev, A.I.5
Hercules, D.M.6
Starzl, T.E.7
Venkataramanan, R.8
|