Inhibition of vinblastine efflux mediated by P-glycoprotein by grapefruit juice components in Caco-2 cells

Biological and Pharmaceutical Bulletin

Volumn 21, Issue 10, 1998, Pages 1062-1066

  Takanaga, Hitomi ^a   Ohnishi, Ayako ^a   Matsuo, Hirotami ^a   Sawada, Yasufumi ^a  

^a KYUSHU UNIVERSITY   (Japan)

Author keywords

Caco 2 cell; Grapefruit juice; P glycoprotein; Vinblastine

Indexed keywords

ACETIC ACID ETHYL ESTER; AURANTIIN; CYCLOSPORIN A; DICHLOROMETHANE; ETHER; GLYCOPROTEIN P; NARINGENIN; VINBLASTINE;

ARTICLE; CELL STRAIN CACO 2; CONTROLLED STUDY; DOSE RESPONSE; DRUG METABOLISM; DRUG UPTAKE; FRUIT JUICE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; PERMEABILITY; STEADY STATE;

EID: 0031790854     PISSN: 09186158     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb.21.1062     Document Type: Article

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