SCOPUS 정보 검색 플랫폼

Volumn 7, Issue 1, 2012, Pages 159-170

Development of improved PPARβ/δ inhibitors

(7) Toth, Philipp M a Naruhn, Simone a Pape, Veronika F S a Dörr, Stefanie M A a Klebe, Gerhard a Müller, Rolf a Diederich, Wibke E a

a PHILIPPS UNIVERSITY MARBURG (Germany)

Author keywords

GSK0660; Inhibitors; NR1C2; Nuclear receptors; PPAR ; Structure activity relationships

Indexed keywords

GSK 0660; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ANTAGONIST; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA INHIBITOR; TERTIARY AMINE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CELL ASSAY; DRUG DESIGN; DRUG SYNTHESIS; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMAN; LIGAND BINDING; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELL LINE; ENZYME INHIBITORS; HUMANS; PPAR DELTA; PPAR-BETA; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONES; THIOPHENES;

EID: 84555186674 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100408 Document Type: Article

Times cited : (26)

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