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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 23, 2011, Pages 7166-7169

Synthesis of GSK3β mimetic inhibitors of Akt featuring a novel extended dipeptide surrogate

(2) Ranatunga, Sujeewa a,b Del Valle, Juan R a

a H LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE (United States)

b NEW MEXICO STATE UNIVERSITY (United States)

Author keywords

Strand; Akt; GSK3; Peptidomimetics; Protein protein interactions

Indexed keywords

DIPEPTIDE; GLYCOGEN SYNTHASE KINASE 3BETA; PEPTIDOMIMETIC AGENT; PROTEIN KINASE B; PROTEIN KINASE B INHIBITOR;

ARTICLE; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG CONFORMATION; DRUG DESIGN; DRUG SYNTHESIS; ENZYME SUBSTRATE; IC 50; MOLECULAR MODEL; STEREOCHEMISTRY; X RAY CRYSTALLOGRAPHY; X RAY DIFFRACTION;

DIPEPTIDES; DRUG DESIGN; ENZYME ACTIVATION; ENZYME INHIBITORS; GLYCOGEN SYNTHASE KINASE 3; INHIBITORY CONCENTRATION 50; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PEPTIDOMIMETICS; PROTO-ONCOGENE PROTEINS C-AKT;

EID: 80255127455 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.09.079 Document Type: Article

Times cited : (7)

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