PET Imaging of CXCR4 Receptors in Cancer by a New Optimized Ligand

ChemMedChem

Volumn 6, Issue 10, 2011, Pages 1789-1791

  Demmer, Oliver ^a   Gourni, Eleni ^a   Schumacher, Udo ^b   Kessler, Horst ^a,c   Wester, Hans Jürgen ^a  

^a TECHNICAL UNIVERSITY OF MUNICH   (Germany)

^b UNIVERSITY MEDICAL CENTER HAMBURG EPPENDORF   (Germany)

^c KING ABDULAZIZ UNIVERSITY   (Saudi Arabia)

Author keywords

CXCR4; DOTA; Imaging agents; Peptides; Positron emission tomography; Tracers

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; ARGININE; BENZOIC ACID; CHEMOKINE RECEPTOR CXCR4; GALLIUM 68; INDIUM; PLERIXAFOR;

AMINO ACID SUBSTITUTION; ARTICLE; B CELL LYMPHOMA; BINDING AFFINITY; BREAST CANCER; CANCER DIAGNOSIS; CELL MIGRATION; COMPUTER ASSISTED EMISSION TOMOGRAPHY; DRUG DISTRIBUTION; ENZYME ACTIVITY; GLIOMA; HYDROPHILICITY; IN VIVO STUDY; ISOTOPE LABELING; LIGAND BINDING; LIPOPHILICITY; LUNG SMALL CELL CANCER; MELANOMA; METASTASIS; NEUROBLASTOMA; NONHUMAN; NUCLEAR MAGNETIC RESONANCE IMAGING; PRIMARY TUMOR; PRIORITY JOURNAL; PROSTATE CANCER; PROTEIN ANALYSIS; PROTEIN BINDING; PROTEIN EXPRESSION; RADIOIODINATION; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; TUMOR GROWTH; UTERINE CERVIX CARCINOMA; XENOGRAFT;

ANIMALS; CELL LINE, TUMOR; CONTRAST MEDIA; COORDINATION COMPLEXES; GALLIUM RADIOISOTOPES; HETEROCYCLIC COMPOUNDS, 1-RING; HUMANS; LIGANDS; MICE; MICE, NUDE; NEOPLASMS; POSITRON-EMISSION TOMOGRAPHY; RECEPTORS, CXCR4; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION; TRANSPLANTATION, HETEROLOGOUS;

EID: 80053432658     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.201100320     Document Type: Article

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