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Volumn 63, Issue 9, 2011, Pages 1141-1155

Mechanisms of burst release from pH-responsive polymeric microparticles

Author keywords

burst release; Eudragit L100; hydrocortisone; microencapsulation; spray drying

Indexed keywords

EUDRAGIT; EUDRAGIT L100; HYDROCORTISONE; POLYMER; UNCLASSIFIED DRUG;

EID: 80051696582     PISSN: 00223573     EISSN: 20427158     Source Type: Journal    
DOI: 10.1111/j.2042-7158.2011.01322.x     Document Type: Article
Times cited : (22)

References (49)
  • 1
    • 11844259383 scopus 로고    scopus 로고
    • Microencapsulation by solvent extraction/evaporation: Reviewing the state of the art of microsphere preparation process technology
    • DOI 10.1016/j.jconrel.2004.10.015, PII S0168365904004845
    • Freitas S, et al,. Microencapsulation by solvent extraction/evaporation: reviewing the state of the art of microsphere preparation process technology. J Control Release 2005; 102: 313-332. (Pubitemid 40093756)
    • (2005) Journal of Controlled Release , vol.102 , Issue.2 , pp. 313-332
    • Freitas, S.1    Merkle, H.P.2    Gander, B.3
  • 2
    • 55649104973 scopus 로고    scopus 로고
    • Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles
    • Wischke C, Schwendeman SP,. Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles. Int J Pharm 2008; 364: 298-327.
    • (2008) Int J Pharm , vol.364 , pp. 298-327
    • Wischke, C.1    Schwendeman, S.P.2
  • 3
    • 33645034817 scopus 로고    scopus 로고
    • Methods for preparation of drug-loaded polymeric nanoparticles
    • Nanoencapsulation 1
    • Pinto Reis C, et al,. Nanoencapsulation 1. Methods for preparation of drug-loaded polymeric nanoparticles. Nanomed Nanotechnol Biol Med 2006; 2: 8-21.
    • (2006) Nanomed Nanotechnol Biol Med , vol.2 , pp. 8-21
    • Pinto Reis, C.1
  • 5
    • 33745585586 scopus 로고    scopus 로고
    • Preparation of roxithromycin-polymeric microspheres by the emulsion solvent diffusion method for taste masking
    • DOI 10.1016/j.ijpharm.2006.03.018, PII S0378517306002365
    • Gao Y, et al,. Preparation of roxithromycin-polymeric microspheres by the emulsion solvent diffusion method for taste masking. Int J Pharm 2006; 318: 62-69. (Pubitemid 43983049)
    • (2006) International Journal of Pharmaceutics , vol.318 , Issue.1-2 , pp. 62-69
    • Gao, Y.1    Cui, F.-d.2    Guan, Y.3    Yang, L.4    Wang, Y.-s.5    Zhang, L.-n.6
  • 6
    • 33750451927 scopus 로고    scopus 로고
    • Encapsulation of lipophilic drugs within enteric microparticles by a novel coacervation method
    • Dong W, Bodmeier R,. Encapsulation of lipophilic drugs within enteric microparticles by a novel coacervation method. Int J Pharm 2006; 326: 128.
    • (2006) Int J Pharm , vol.326 , pp. 128
    • Dong, W.1    Bodmeier, R.2
  • 7
    • 0023698042 scopus 로고
    • Preparation of biodegradable poly(±)lactide microparticles using a spray-drying technique
    • Bodmeier R, Chen H,. Preparation of biodegradable poly(±)lactide microparticles using a spray-drying technique. J Pharm Pharmacol 1988; 40: 754-757.
    • (1988) J Pharm Pharmacol , vol.40 , pp. 754-757
    • Bodmeier, R.1    Chen, H.2
  • 8
    • 0035083556 scopus 로고    scopus 로고
    • Spray-drying as a method for microparticulate controlled release systems preparation: Advantages and limits. I. Water-soluble drugs
    • Palmieri G, et al,. Spray-drying as a method for microparticulate controlled release systems preparation: Advantages and limits. I. Water-soluble drugs. Drug Dev Ind Pharm 2001; 27: 195.
    • (2001) Drug Dev Ind Pharm , vol.27 , pp. 195
    • Palmieri, G.1
  • 9
    • 0037151532 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of pyridostigmine bromide microparticles
    • Hegazy N, et al,. Preparation and in vitro evaluation of pyridostigmine bromide microparticles. Int J Pharm 2002; 242: 171.
    • (2002) Int J Pharm , vol.242 , pp. 171
    • Hegazy, N.1
  • 10
    • 44749090403 scopus 로고    scopus 로고
    • Taste masking microspheres for orally disintegrating tablets
    • Xu J, et al,. Taste masking microspheres for orally disintegrating tablets. Int J Pharm 2008; 359: 63-69.
    • (2008) Int J Pharm , vol.359 , pp. 63-69
    • Xu, J.1
  • 11
    • 0037124468 scopus 로고    scopus 로고
    • Sustained release of etanidazole from spray dried microspheres prepared by non-halogenated solvents
    • DOI 10.1016/S0168-3659(02)00066-4, PII S0168365902000664
    • Wang F-J, Wang C-H,. Sustained release of etanidazole from spray dried microspheres prepared by non-halogenated solvents. J Control Release 2002; 81: 263-280. (Pubitemid 34607147)
    • (2002) Journal of Controlled Release , vol.81 , Issue.3 , pp. 263-280
    • Wang, F.-J.1    Wang, C.-H.2
  • 12
    • 62949197149 scopus 로고    scopus 로고
    • PH-Sensitive nanospheres for colon-specific drug delivery in experimentally induced colitis rat model
    • Makhlof A, et al,. pH-Sensitive nanospheres for colon-specific drug delivery in experimentally induced colitis rat model. Eur J Pharm Biopharm 2009; 72: 1-8.
    • (2009) Eur J Pharm Biopharm , vol.72 , pp. 1-8
    • Makhlof, A.1
  • 13
    • 0032801932 scopus 로고    scopus 로고
    • Solvent influence on spray-dried biodegradable microspheres
    • DOI 10.1080/026520499288915
    • Bain DF, et al,. Solvent influence on spray-dried biodegradable microspheres. J Microencapsul 1999; 16: 453-474. (Pubitemid 29332733)
    • (1999) Journal of Microencapsulation , vol.16 , Issue.4 , pp. 453-474
    • Bain, D.F.1    Munday, D.L.2    Smith, A.3
  • 14
    • 42049094490 scopus 로고    scopus 로고
    • Pharmaceutical particle engineering via spray drying
    • Vehring R,. Pharmaceutical particle engineering via spray drying. Pharm Res 2008; 25: 999-1022.
    • (2008) Pharm Res , vol.25 , pp. 999-1022
    • Vehring, R.1
  • 16
    • 0031881636 scopus 로고    scopus 로고
    • PDLLA microspheres containing steroids: Spray-drying, o/w and w/o/w emulsifications as preparation methods
    • Giunchedi P, et al,. PDLLA microspheres containing steroids: spray drying, o/w and w/o/w emulsification as preparation methods. J Microencapsul 1998; 15: 185-195. (Pubitemid 28105134)
    • (1998) Journal of Microencapsulation , vol.15 , Issue.2 , pp. 185-195
    • Giunchedi, P.1    Alpar, H.O.2    Conte, U.3
  • 17
    • 80054738031 scopus 로고    scopus 로고
    • Using pH abnormalities in diseased skin to trigger and target topical therapy
    • (in press)
    • Rizi K, et al,. Using pH abnormalities in diseased skin to trigger and target topical therapy. Pharm Res 2011 (in press).
    • (2011) Pharm Res
    • Rizi, K.1
  • 18
    • 0032752533 scopus 로고    scopus 로고
    • Cutaneous pH in children affected by atopic dermatitis and in healthy children: A multicenter study
    • DOI 10.1111/j.1600-0846.1999.tb00134.x
    • Sparavigna A, et al,. Cutaneous pH in children affected by atopic dermatitis and in healthy children: a multicenter study. Skin Res Technol 1999; 5: 221-227. (Pubitemid 29504971)
    • (1999) Skin Research and Technology , vol.5 , Issue.4 , pp. 221-227
    • Sparavigna, A.1    Setaro, M.2    Gualandri, V.3
  • 19
    • 67349281689 scopus 로고    scopus 로고
    • Fabrication and in vivo evaluation of highly pH-responsive acrylic microparticles for targeted gastrointestinal delivery
    • Kendall RA, et al,. Fabrication and in vivo evaluation of highly pH-responsive acrylic microparticles for targeted gastrointestinal delivery. Eur J Pharm Sci 2009; 37: 284-290.
    • (2009) Eur J Pharm Sci , vol.37 , pp. 284-290
    • Kendall, R.A.1
  • 20
    • 48149092612 scopus 로고    scopus 로고
    • Characterisation of excipient-free nanoporous microparticles (NPMPs) of bendroflumethiazide
    • Healy AM, et al,. Characterisation of excipient-free nanoporous microparticles (NPMPs) of bendroflumethiazide. Eur J Pharm Biopharm 2008; 69: 1182-1186.
    • (2008) Eur J Pharm Biopharm , vol.69 , pp. 1182-1186
    • Healy, A.M.1
  • 21
    • 62949241990 scopus 로고    scopus 로고
    • Physical characteristics and aerosol performance of naringin dry powders for pulmonary delivery prepared by spray-drying
    • Sansone F, et al,. Physical characteristics and aerosol performance of naringin dry powders for pulmonary delivery prepared by spray-drying. Eur J Pharm Biopharm 2009; 72: 206-213.
    • (2009) Eur J Pharm Biopharm , vol.72 , pp. 206-213
    • Sansone, F.1
  • 22
    • 80051700283 scopus 로고
    • ed. New York: Academic Press,: Analytical profiles of drug substances; No. 1
    • Florey K, ed. Triamcinolone. New York: Academic Press, 1977: Analytical profiles of drug substances; No. 1.
    • (1977) Triamcinolone
    • Florey, K.1
  • 23
    • 1542332529 scopus 로고    scopus 로고
    • Penciclovir solubility in Eudragit films: A comparison of X-ray, thermal, microscopic and release rate techniques
    • DOI 10.1016/j.jpba.2003.11.018, PII S0731708503006940
    • Ahmed A, et al,. Penciclovir solubility in Eudragit films: a comparison of X-ray, thermal, microscopic and release rate techniques. J Pharm Biomed Anal 2004; 34: 945-956. (Pubitemid 38296397)
    • (2004) Journal of Pharmaceutical and Biomedical Analysis , vol.34 , Issue.5 , pp. 945-956
    • Ahmed, A.1    Barry, B.W.2    Williams, A.C.3    Davis, A.F.4
  • 24
    • 78650543899 scopus 로고    scopus 로고
    • Production of pH-responsive microparticles by spray drying: Investigation of experimental parameter effects on morphological and release properties
    • Rizi K, et al,. Production of pH-responsive microparticles by spray drying: investigation of experimental parameter effects on morphological and release properties. J Pharm Sci 2010; 100: 566-579.
    • (2010) J Pharm Sci , vol.100 , pp. 566-579
    • Rizi, K.1
  • 25
    • 64649100465 scopus 로고    scopus 로고
    • Hydroxypropyl methylcellulose acetate succinate-based spray-dried dispersions: An overview
    • Friesen DT, et al,. Hydroxypropyl methylcellulose acetate succinate-based spray-dried dispersions: an overview. Mol Pharm 2008; 5: 1003-1019.
    • (2008) Mol Pharm , vol.5 , pp. 1003-1019
    • Friesen, D.T.1
  • 26
    • 80051678920 scopus 로고    scopus 로고
    • Technical bulletin: Shin-Estu AQOAT: Shin-Estu Chemical Co.Ltd 2006
    • Technical bulletin: Shin-Estu AQOAT: Shin-Estu Chemical Co.Ltd. 2006.
  • 29
    • 33646772174 scopus 로고    scopus 로고
    • Nanoparticles in inflammatory bowel disease: Particle targeting versus pH-sensitive delivery
    • DOI 10.1016/j.ijpharm.2006.01.032, PII S0378517306000834
    • Meissner Y, et al,. Nanoparticles in inflammatory bowel disease: particles targeting versus pH-sensitive delivery. Int J Pharm 2006; 316: 138-143. (Pubitemid 43765696)
    • (2006) International Journal of Pharmaceutics , vol.316 , Issue.1-2 , pp. 138-143
    • Meissner, Y.1    Pellequer, Y.2    Lamprecht, A.3
  • 31
    • 3042854242 scopus 로고    scopus 로고
    • pH-sensitive microsphere delivery increases oral bioavailability of calcitonin
    • DOI 10.1016/j.jconrel.2004.02.001, PII S0168365904000616
    • Lamprecht A, et al,. pH-sensitive microsphere delivery increases oral bioavailability of calcitonin. J Control Release 2004; 98: 1-9. (Pubitemid 38881602)
    • (2004) Journal of Controlled Release , vol.98 , Issue.1 , pp. 1-9
    • Lamprecht, A.1    Yamamoto, H.2    Takeuchi, H.3    Kawashima, Y.4
  • 33
    • 3242688832 scopus 로고    scopus 로고
    • A novel pH-dependent gradient-release delivery system for nitrendipine: I. Manufacturing, evaluation in vitro and bioavailability in healthy dogs
    • DOI 10.1016/j.jconrel.2004.04.022, PII S0168365904002184
    • Yang M, et al,. A novel pH-dependent gradient-release delivery system for nitrendipine: I. Manufacturing, evaluation in vitro and bioavailability in healthy dogs. J Control Release 2004; 98: 219-229. (Pubitemid 38950732)
    • (2004) Journal of Controlled Release , vol.98 , Issue.2 , pp. 219-229
    • Yang, M.1    Cui, F.2    You, B.3    You, J.4    Wang, L.5    Zhang, L.6    Kawashima, Y.7
  • 34
    • 11144249850 scopus 로고    scopus 로고
    • A novel formulation design about water-insoluble oily drug: Preparation of zedoary turmeric oil microspheres with self-emulsifying ability and evaluation in rabbits
    • DOI 10.1016/j.ijpharm.2004.10.005, PII S0378517304005988
    • You J, et al,. A novel formulation design about water-insoluble oily drug: preparation of zedoary turmeric oil microspheres with self-emulsifying ability and evaluation in rabbits. Int J Pharm 2005; 288: 315-323. (Pubitemid 40038585)
    • (2005) International Journal of Pharmaceutics , vol.288 , Issue.2 , pp. 315-323
    • You, J.1    Cui, F.-D.2    Li, Q.-P.3    Han, X.4    Yu, Y.-W.5    Yang, M.-S.6
  • 35
    • 0038061601 scopus 로고    scopus 로고
    • Physicochemical properties to determine the buoyancy of hollow microspheres (microballoons) prepared by the emulsion solvent diffusion method
    • DOI 10.1016/S0939-6411(03)00003-1
    • Sato Y, et al,. Physicochemical properties to determine the buoyancy of hollow microparticles (microballons) prepared by the emulsion solvent diffusion method. Eur J Pharm Biopharm 2003; 55: 297-304. (Pubitemid 36561556)
    • (2003) European Journal of Pharmaceutics and Biopharmaceutics , vol.55 , Issue.3 , pp. 297-304
    • Sato, Y.1    Kawashima, Y.2    Takeuchi, H.3    Yamamoto, H.4
  • 37
    • 1842421289 scopus 로고    scopus 로고
    • Effect of the size of biodegradable microparticles on drug release: Experiment and theory
    • DOI 10.1016/j.jconrel.2004.01.011, PII S0168365904000379
    • Siepmann J, et al,. Effect of the size of biodegradable microparticles on drug release: experiment and theory. J Control Release 2004; 96: 123-134. (Pubitemid 38438495)
    • (2004) Journal of Controlled Release , vol.96 , Issue.1 , pp. 123-134
    • Siepmann, J.1    Faisant, N.2    Akiki, J.3    Richard, J.4    Benoit, J.P.5
  • 38
    • 10044282200 scopus 로고    scopus 로고
    • On the mechanisms of surface formation and the surface compositions of industrial milk powders
    • Kim EH-J, et al,. On the mechanisms of surface formation and the surface compositions of industrial milk powders. Drying Technol 2003; 21: 265-278.
    • (2003) Drying Technol , vol.21 , pp. 265-278
    • Kim, E.-J.1
  • 39
    • 68649120071 scopus 로고    scopus 로고
    • Drug distribution in enteric microparticles
    • Nilkumhang S, et al,. Drug distribution in enteric microparticles. Int J Pharm 2009; 379: 1-8.
    • (2009) Int J Pharm , vol.379 , pp. 1-8
    • Nilkumhang, S.1
  • 40
    • 0032734092 scopus 로고    scopus 로고
    • Formation and physical characterisation of large porous particles for inhalation
    • Vanber R,. Formation and physical characterisation of large porous particles for inhalation. Pharm Res 1999; 16: 1735-1742.
    • (1999) Pharm Res , vol.16 , pp. 1735-1742
    • Vanber, R.1
  • 41
    • 67649645083 scopus 로고    scopus 로고
    • The robustness and flexibility of an emulsion solvent evaporation method to prepare pH-responsive microparticles
    • Nilkumhang S, Basit AW,. The robustness and flexibility of an emulsion solvent evaporation method to prepare pH-responsive microparticles. Int J Pharm 2009; 377: 135-141.
    • (2009) Int J Pharm , vol.377 , pp. 135-141
    • Nilkumhang, S.1    Basit, A.W.2
  • 42
    • 77953469221 scopus 로고    scopus 로고
    • Preparation and evaluation of polymeric carbamazepine spherical crystals by emulsion solvent diffusion technique
    • Yadav A, Yadav V,. Preparation and evaluation of polymeric carbamazepine spherical crystals by emulsion solvent diffusion technique. Asia J Pharm 2009; 3: 18-25.
    • (2009) Asia J Pharm , vol.3 , pp. 18-25
    • Yadav, A.1    Yadav, V.2
  • 43
    • 0000187747 scopus 로고
    • Thermoanalysis of microspheres
    • Dubernet C,. Thermoanalysis of microspheres. Thermochim Acta 1995; 248: 259-269.
    • (1995) Thermochim Acta , vol.248 , pp. 259-269
    • Dubernet, C.1
  • 44
    • 58149321881 scopus 로고
    • Study of a theophylline-Eudragit L mixture using a combined system of microscopic Fourier-transform infrared spectroscopy and differential scanning calorimetry
    • Lin S-Y, et al,. Study of a theophylline-Eudragit L mixture using a combined system of microscopic Fourier-transform infrared spectroscopy and differential scanning calorimetry. Thermochim Acta 1995; 245: 153-166.
    • (1995) Thermochim Acta , vol.245 , pp. 153-166
    • Lin, S.-Y.1
  • 45
    • 0037074120 scopus 로고    scopus 로고
    • Preparation and characterisation of hydrocortisone particles using a supercritical fluids extraction process
    • DOI 10.1016/S0378-5173(01)00870-5, PII S0378517301008705
    • Velaga SP, et al,. Preparation and characterisation of hydrocortisone particles using a supercritical fluids extraction process. Int J Pharm 2002; 231: 155-166. (Pubitemid 34033675)
    • (2002) International Journal of Pharmaceutics , vol.231 , Issue.2 , pp. 155-166
    • Velaga, S.P.1    Ghaderi, R.2    Carlfors, J.3
  • 46
    • 2342494846 scopus 로고    scopus 로고
    • FT-IR imaging and Raman microscopic study of poly(ethylene terephthalate) film processed with supercritical CO2
    • Fleming OS, et al,. FT-IR imaging and Raman microscopic study of poly(ethylene terephthalate) film processed with supercritical CO2. Vibrational Spectrosc 2004; 35: 3-7.
    • (2004) Vibrational Spectrosc , vol.35 , pp. 3-7
    • Fleming, O.S.1
  • 47
    • 0346731827 scopus 로고
    • Analytical potential of near-infrared fourier transform Raman spectra in the detection of solid transition metal carbonyl steroid hormones
    • Salmain M, et al,. Analytical potential of near-infrared fourier transform Raman spectra in the detection of solid transition metal carbonyl steroid hormones. J Raman Spectrosc 1995; 26: 31-38.
    • (1995) J Raman Spectrosc , vol.26 , pp. 31-38
    • Salmain, M.1


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