Activity-dependent targeting of TRPV1 with a pore-permeating capsaicin analog

Proceedings of the National Academy of Sciences of the United States of America

Volumn 108, Issue 20, 2011, Pages 8497-8502

  Li, Hui ^a   Wang, Shu ^a   Chuang, Alexander Y ^b   Cohen, Bruce E ^c   Chuang, Huai Hu ^b  

^a Department of Molecular Biology and Genetics   (United States)

^b Lowell High School   (United States)

^c LAWRENCE BERKELEY NATIONAL LABORATORY   (United States)

Author keywords

Activity dependent capsaicinoids; Hyperalgesia; Ion permeation; Selective analgesia

Indexed keywords

CALCIUM; CAPSAICIN DERIVATIVE; DYE; PHOSPHOTRANSFERASE; SODIUM CHANNEL BLOCKING AGENT; VANILLOID RECEPTOR 1; VANILLOID RECEPTOR AGONIST;

ARTICLE; CALCIUM TRANSPORT; COVALENT BOND; DRUG TARGETING; ELECTRIC CURRENT; ENZYME ACTIVATION; HUMAN; HUMAN CELL; ION TRANSPORT; NOCICEPTION; OXIDATION; PRIORITY JOURNAL; RECEPTOR UPREGULATION; SENSORY NERVE CELL; SODIUM CURRENT;

ANIMALS; BIOLOGICAL TRANSPORT; CAPSAICIN; CELL MEMBRANE PERMEABILITY; HUMANS; RATS; TRPV CATION CHANNELS;

EID: 79957733084     PISSN: 00278424     EISSN: 10916490     Source Type: Journal    
DOI: 10.1073/pnas.1018550108     Document Type: Article

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