-
1
-
-
6044256350
-
4-Thiazolidones: Centenarian history, current status and perspectives for modern organic and medicinal chemistry
-
Lesyk R. B., Zimenkovsky B. S. 4-Thiazolidones: centenarian history, current status and perspectives for modern organic and medicinal chemistry. Curr. Org. Chem. 2004. 8, N 16. P. 1547-1577.
-
(2004)
Curr. Org. Chem
, vol.8
, Issue.16
, pp. 1547-1577
-
-
Lesyk, R.B.1
Zimenkovsky, B.S.2
-
3
-
-
67650261319
-
Rhodanine as a privileged scaffold in drug discovery
-
Tomasic T., Masic L. P. Rhodanine as a privileged scaffold in drug discovery. Curr. Med. Chem. 2009.16, N 13. P. 1596-1629.
-
(2009)
Curr. Med. Chem
, vol.16
, Issue.13
, pp. 1596-1629
-
-
Tomasic, T.1
Masic, L.P.2
-
4
-
-
0032484224
-
Potent antidiabetic thiazolidinedione with unique peroxisome proliferator-activated receptor gammaactivating properties
-
Reginato M. J., Bailey S. T., Krakow S. L., Minami C., Ishii S., Tanaka H., Lazar M. A. A potent antidiabetic thiazolidinedione with unique peroxisome proliferator-activated receptor gammaactivating properties. J. Biol. Chem. 1998. 273, N 49. P. 32679-32684.
-
(1998)
J. Biol. Chem
, vol.273
, Issue.49
, pp. 32679-32684
-
-
Reginato, M.J.1
Bailey, S.T.2
Krakow, S.L.3
Minami, C.4
Ishii, S.5
Tanaka, H.6
Lazar, M.7
-
5
-
-
0021828899
-
Aldose reductase inhibitors: A potential new class of agents for the pharmacological control of certain diabetic complications
-
Kador P. F., Kinoshita J. H., Sharpless N. E. Aldose reductase inhibitors: a potential new class of agents for the pharmacological control of certain diabetic complications. J. Med. Chem. 1985. 28, N 7. P. 841-849.
-
(1985)
J. Med. Chem
, vol.28
, Issue.7
, pp. 841-849
-
-
Kador, P.F.1
Kinoshita, J.H.2
Sharpless, N.E.3
-
6
-
-
0042574211
-
Mishaux C. Dual inhibition of cyclooxygenase-2 (COX-2) and 5-lipoxygenase (5-LOX) as a new strategy to provide safer non-steroidal anti-inflammatory drugs
-
Charlier C., Mishaux C. Dual inhibition of cyclooxygenase-2 (COX-2) and 5-lipoxygenase (5-LOX) as a new strategy to provide safer non-steroidal anti-inflammatory drugs. Eur. J. Med. Chem. 2003. 38, N 7 8. P. 645-659.
-
(2003)
Eur. J. Med. Chem
, vol.38
, Issue.7-8
, pp. 645-659
-
-
Charlier, C.1
-
7
-
-
85038483264
-
-
th ed.-New Jersey
-
The Merck Index.Eds M. J. O'Neil et al.:13th ed.-New Jersey, 2001. 1818 p.
-
The Merck Index
, vol.2001
, pp. 1818
-
-
-
8
-
-
0037169976
-
Benzylidene rhodanines as novel inhibitors of UDP-N-ace-tylmuramate/L-alanine ligase
-
Sim M. M., Ng S. B., Buss A. D., Crasta S. C., Goh K. L., Lee S. K. Benzylidene rhodanines as novel inhibitors of UDP-N-ace-tylmuramate/L-alanine ligase. Bioorg. Med. Chem. Lett. 2002. 12, N 4.P. 697-699.
-
(2002)
Bioorg. Med. Chem. Lett
, vol.12
, Issue.4
, pp. 697-699
-
-
Sim, M.M.1
Ng, S.B.2
Buss, A.D.3
Crasta, S.C.4
Goh, K.L.5
Lee, S.K.6
-
9
-
-
0037279491
-
Peroxisome proliferator activated receptor-gamma ligands as potent antineoplastic agents
-
Theocharisa S., Margeli A., Kouraklis G. Peroxisome proliferator activated receptor-gamma ligands as potent antineoplastic agents. Curr. Med. Chem. Anticancer Agents. 2003. 3, N 3. P. 239-251.
-
(2003)
Curr. Med. Chem. Anticancer Agents
, vol.3
, Issue.3
, pp. 239-251
-
-
Theocharisa, S.1
Margeli, A.2
Kouraklis, G.3
-
10
-
-
0034406481
-
PPAR-gamma agonists: Therapeutic role in diabetes, inflammation and cancer
-
Murphy G. J., Holder J. C. PPAR-gamma agonists: therapeutic role in diabetes, inflammation and cancer. Trends Pharmacol. Sci. 2000. 21, N 12. P. 469-474.
-
(2000)
Trends Pharmacol. Sci
, vol.21
, Issue.12
, pp. 469-474
-
-
Murphy, G.J.1
Holder, J.C.2
-
11
-
-
0035150803
-
Identification of small-molecule inhibitors of interaction between the BH3 domain and Bcl-xL
-
Degterev A., Lugovskoy A., Cardone M., Mulley B., Wagner G., Mitchison T., Yuan J. Identification of small-molecule inhibitors of interaction between the BH3 domain and Bcl-xL. Nat. Cell Biol. 2001. 3, N 2. P. 173-182.
-
(2001)
Nat. Cell Biol
, vol.3
, Issue.2
, pp. 173-182
-
-
Degterev, A.1
Lugovskoy, A.2
Cardone, M.3
Mulley, B.4
Wagner, G.5
Mitchison, T.6
Yuan, J.7
-
12
-
-
0035834057
-
Photochemically enhanced binding of small molecules to the tumor necrosis factor receptor-1 inhibits the binding of TNF-alpha
-
Carter P. H., Scherle P. A., Muckelbauer J. K., Voss M. E., Liu R.-Q., Thompson L. A., Tebben A. J., Solomon K. A., Lo Y. C., Li Z., Strzemienski P., Yang G., Falahatpisheh N., Xu M., Wu Z., Farrow N. A., Ramnarayan K., Wang J., Rideout D., Yalamoori V., Domaille P., Underwood D. J., Trzaskos J. M., Friedman S. M., Newton R. C., Decicco C. P. Photochemically enhanced binding of small molecules to the tumor necrosis factor receptor-1 inhibits the binding of TNF-alpha. Proc. Natl Acad. Sci. USA. 2001. 98, N 21. P. 11879-11884.
-
(2001)
Proc. Natl Acad. Sci. USA
, vol.98
, Issue.21
, pp. 11879-11884
-
-
Carter, P.H.1
Scherle, P.A.2
Muckelbauer, J.K.3
Voss, M.E.4
Liu, R.-Q.5
Thompson, L.A.6
Tebben, A.J.7
Solomon, K.A.8
Lo, Y.C.9
Li, Z.10
Strzemienski, P.11
Yang, G.12
Falahatpisheh, N.13
Xu, M.14
Wu, Z.15
Farrow, N.A.16
Ramnarayan, K.17
Wang, J.18
Rideout, D.19
Yalamoori, V.20
Domaille, P.21
Underwood, D.J.22
Trzaskos, J.M.23
Friedman, S.M.24
Newton, R.C.25
Decicco, C.P.26
more..
-
13
-
-
51349107262
-
Structure-activity relationship study of a novel necroptosis inhibitor, necro-statin-7
-
Zheng W., Degterev A., Hsu E., Yuan J., Yuan C. Structure-activity relationship study of a novel necroptosis inhibitor, necro-statin-7. Bioorg. Med. Chem. Lett. 2008. 18, N 18. P. 4932-4935.
-
(2008)
Bioorg. Med. Chem. Lett
, vol.18
, Issue.18
, pp. 4932-4935
-
-
Zheng, W.1
Degterev, A.2
Hsu, E.3
Yuan, J.4
Yuan, C.5
-
14
-
-
33746763743
-
Discovery of small molecule integrin avb3 antagonists as novel anticancer agents
-
Dayam R., Aiello F., Deng J., Wu Y., Garofalo A., Chen X., Nea- mati N. Discovery of small molecule integrin avb3 antagonists as novel anticancer agents. J. Med. Chem. 2006. 49, N 15. P. 4526-4534.
-
(2006)
J. Med. Chem
, vol.49
, Issue.15
, pp. 4526-4534
-
-
Dayam, R.1
Aiello, F.2
Deng, J.3
Wu, Y.4
Garofalo, A.5
Chen, X.6
Nea- Mati, N.7
-
15
-
-
20644458125
-
Rhodanine derivatives as inhibitors of JSP-1
-
Cutshall N. S., O’Day C., Prezhdo M. Rhodanine derivatives as inhibitors of JSP-1. Bioorg. Med. Chem. Lett. 2005. 15, N 14. P. 3374-3379.
-
(2005)
Bioorg. Med. Chem. Lett
, vol.15
, Issue.14
, pp. 3374-3379
-
-
Cutshall, N.S.1
O’Day, C.2
Prezhdo, M.3
-
16
-
-
59449108140
-
Synthesis and evaluation of novel inhibitors of Pim-1 and Pim-2 protein kinases
-
Xia Z., Knaak C., Ma J., Beharry Z. M., McInnes C., Wang W., Kraft A. S., Smith C. D. Synthesis and evaluation of novel inhibitors of Pim-1 and Pim-2 protein kinases. J. Med. Chem. 2009. 52, N 1. P. 74-86.
-
(2009)
J. Med. Chem
, vol.52
, Issue.1
, pp. 74-86
-
-
Xia, Z.1
Knaak, C.2
Ma, J.3
Beharry, Z.M.4
McInnes, C.5
Wang, W.6
Kraft, A.S.7
Smith, C.D.8
-
17
-
-
20344368812
-
G. 5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel anti-inflammatory agents
-
Ottana R., Maccari R., Barreca M. L., Bruno G., Rotondo A., Rossi A., Chiricosta G., Di Paola R., Sautebin L., Cuzzocrea S., Vigorita M. G. 5-Arylidene-2-imino-4-thiazolidinones: design and synthesis of novel anti-inflammatory agents. Bioorg. Med. Chem. 2005. 13, N 13. P. 4243-4252.
-
(2005)
Bioorg. Med. Chem
, vol.13
, Issue.13
, pp. 4243-4252
-
-
Ottana, R.1
Maccari, R.2
Barreca, M.L.3
Bruno, G.4
Rotondo, A.5
Rossi, A.6
Chiricosta, G.7
Di Paola, R.8
Sautebin, L.9
Cuzzocrea, S.10
Vigorita, M.11
-
18
-
-
79957675488
-
Khyluk D. Anticancer potential of 4-azolidones and related heterocycles
-
Lesyk R., Zimenkovsky B., Kaminskyy D., Holota S., Atamanyuk D., Havryluk D., Nektegayev I., Kazmirchuk G., Subtel’na I., Roman O., Kryshchyshyn A., Khyluk D. Anticancer potential of 4-azolidones and related heterocycles. Annal. UMCS. Sectio DDD. 2006. 19, N 1. P. 107-110.
-
(2006)
Annal. UMCS. Sectio DDD
, vol.19
, Issue.1
, pp. 107-110
-
-
Lesyk, R.1
Zimenkovsky, B.2
Kaminskyy, D.3
Holota, S.4
Atamanyuk, D.5
Havryluk, D.6
Nektegayev, I.7
Kazmirchuk, G.8
Subtel’Na, I.9
Roman, O.10
Kryshchyshyn, A.11
-
19
-
-
0031855661
-
New thiazolidones-4 with pyrazolone-5 substituent as the potential NSAIDs
-
Lesyk R., Vladzimirska O., Zimenkovsky B., Horishny V., Nektegayev I., Solyanyk V., Vovk O. New thiazolidones-4 with pyrazolone-5 substituent as the potential NSAIDs. Bol. Chim. Farm. 1998. 137, N 6. P. 210-217.
-
(1998)
Bol. Chim. Farm
, vol.137
, Issue.6
, pp. 210-217
-
-
Lesyk, R.1
Vladzimirska, O.2
Zimenkovsky, B.3
Horishny, V.4
Nektegayev, I.5
Solyanyk, V.6
Vovk, O.7
-
20
-
-
85038520025
-
Pharmaco logical screening and 2D-QSAR analysis of anti-inflammatory activity of 4-thiazolidone derivatives
-
Lesyk R. B., Artemenko A. G., Zimenkovsky B. S., Kuz’min V. E., Nektegayev I. O., Roman O. M., Atamanyuk D. V. Pharmaco logical screening and 2D-QSAR analysis of anti-inflammatory activity of 4-thiazolidone derivatives. Farmacevtychnyj Zhur. 2003. N 3. P. 58-61.
-
(2003)
Farmacevtychnyj Zhur
, vol.3
, pp. 58-61
-
-
Lesyk, R.B.1
Artemenko, A.G.2
Zimenkovsky, B.S.3
Kuz’Min, V.E.4
Nektegayev, I.O.5
Roman, O.M.6
Atamanyuk, D.V.7
-
21
-
-
1342312167
-
Synthesis and antinflammatory activity of some 2-aryl-amino-2-thiazoline-4-ones
-
Lesyk R., Zimenkovsky B., Subtelna I., Nektegayev I., Kazmirchuk G. Synthesis and antinflammatory activity of some 2-aryl-amino-2-thiazoline-4-ones. Acta Pol. Pharm. 2003. 60, N 6. P. 457-466.
-
(2003)
Acta Pol. Pharm
, vol.60
, Issue.6
, pp. 457-466
-
-
Lesyk, R.1
Zimenkovsky, B.2
Subtelna, I.3
Nektegayev, I.4
Kazmirchuk, G.5
-
22
-
-
6044243058
-
Synthesis and studing of antimicrobial activity of azolidine derivatives with 2-(2-chlorobenzyloxy)-5-nitrophenyl fragment in molecules
-
Lesyk R., Zimenkovsky B., Kutsyk R. V., Atamanyuk D. V., Semenciv G. M. Synthesis and studing of antimicrobial activity of azolidine derivatives with 2-(2-chlorobenzyloxy)-5-nitrophenyl fragment in molecules. Farmacevtychnyj Zhur. 2003. N 2. P. 52-56.
-
(2003)
Farmacevtychnyj Zhur
, vol.2
, pp. 52-56
-
-
Lesyk, R.1
Zimenkovsky, B.2
Kutsyk, R.V.3
Atamanyuk, D.V.4
Semenciv, G.M.5
-
23
-
-
33750880872
-
Synthesis and antimicrobial activity of 2,4-dioxothiazolidine-5-acetic acid amides
-
Zimenkovskii B. S., Kutsyk R. V., Lesyk R. B., Matyichuk V. S., Obushak N. D., Klyufinska T. I. Synthesis and antimicrobial activity of 2,4-dioxothiazolidine-5-acetic acid amides. Pharm. Chem. J. 2006. 40, N 6. P. 303-306.
-
(2006)
Pharm. Chem. J
, vol.40
, Issue.6
, pp. 303-306
-
-
Zimenkovskii, B.S.1
Kutsyk, R.V.2
Lesyk, R.B.3
Matyichuk, V.S.4
Obushak, N.D.5
Klyufinska, T.I.6
-
24
-
-
0033619971
-
3-Oxyarylthiazolidones-4 and their choleretic activity
-
Nektegayev I., Lesyk R. 3-Oxyarylthiazolidones-4 and their choleretic activity. Sci. Pharm. 1999. 67. P. 227-230.
-
(1999)
Sci. Pharm
, vol.67
, pp. 227-230
-
-
Nektegayev, I.1
Lesyk, R.2
-
25
-
-
85038482867
-
Antioxidant activity of 5-arylidene-2,4-thazolidinedione-3-alkanoic acid derivatives
-
Lukyanchuk V. D., Zimenkovsky B. S., Lesyk R. B., Nemyatykh O. D., Nektegayev I. O. Antioxidant activity of 5-arylidene-2,4-thazolidinedione-3-alkanoic acid derivatives. J. Pharm. Pharmacol. 2002. 54, Suppl. S. 1.
-
(2002)
J. Pharm. Pharmacol
, vol.54
, pp. 1
-
-
Lukyanchuk, V.D.1
Zimenkovsky, B.S.2
Lesyk, R.B.3
Nemyatykh, O.D.4
Nektegayev, I.O.5
-
26
-
-
0028906786
-
Some practical considerations and applications of the national cancer institute in vitro anticancer drug discovery screen
-
Boyd M. R., Paull K. D. Some practical considerations and applications of the national cancer institute in vitro anticancer drug discovery screen. Drug Dev. Res. 1995. 34, N 2. P. 91-109.
-
(1995)
Drug Dev. Res
, vol.34
, Issue.2
, pp. 91-109
-
-
Boyd, M.R.1
Paull, K.D.2
-
27
-
-
84965822602
-
Feasibility of drug screening with panels of human tumor cell lines using a microculture tetrazolium assay
-
Alley M. C., Scudiero D. A., Monks A., Hursey M. L., Czerwinski M. J., Fine D. L., Abbott B. J., Mayo J. G., Shoemaker R. H., Boyd M. R. Feasibility of drug screening with panels of human tumor cell lines using a microculture tetrazolium assay. Cancer Res. 1988. 48, N 3. P. 589-601.
-
(1988)
Cancer Res
, vol.48
, Issue.3
, pp. 589-601
-
-
Alley, M.C.1
Scudiero, D.A.2
Monks, A.3
Hursey, M.L.4
Czerwinski, M.J.5
Fine, D.L.6
Abbott, B.J.7
Mayo, J.G.8
Shoemaker, R.H.9
Boyd, M.R.10
-
28
-
-
0025775062
-
Feasibility of a high-flux anticancer drug screen using a diverse panel of cultured human tumor cell lines
-
Monks A., Scudiero D., Skehan P., Shoemaker R., Paull K., Vistica D., Hose C., Langley J., Cronise P., Vaigro-Wolff A., Gray-Goodrich M., Campbell H., Mayo J., Boyd M. Feasibility of a high-flux anticancer drug screen using a diverse panel of cultured human tumor cell lines. J. Natl Cancer. Inst. 1991. 83, N 11. P. 757-766.
-
(1991)
J. Natl Cancer. Inst
, vol.83
, Issue.11
, pp. 757-766
-
-
Monks, A.1
Scudiero, D.2
Skehan, P.3
Shoemaker, R.4
Paull, K.5
Vistica, D.6
Hose, C.7
Langley, J.8
Cronise, P.9
Vaigro-Wolff, A.10
Gray-Goodrich, M.11
Campbell, H.12
Mayo, J.13
Boyd, M.14
-
30
-
-
33749011163
-
The NCI60 human tumour cell line anticancer drug screen
-
Shoemaker R. H. The NCI60 human tumour cell line anticancer drug screen. Nat. Rev. Cancer. 2006. 6, N 10. P. 813-823.
-
(2006)
Nat. Rev. Cancer
, vol.6
, Issue.10
, pp. 813-823
-
-
Shoemaker, R.H.1
-
31
-
-
33745167386
-
Anticancer thiopyrano[2,3-d][1,3]thiazol-2-ones with norbornane moiety. Synthesis, cytotoxicity, physico-chemical properties, and computational studies
-
Lesyk R., Zimenkovsky B., Atamanyuk D., Jensen F., Kiec-Kononowicz K., Gzella A. Anticancer thiopyrano[2,3-d][1,3]thiazol-2-ones with norbornane moiety. Synthesis, cytotoxicity, physico-chemical properties, and computational studies. Bioorg. Med. Chem. 2006. 14, N 15. P. 5230-5240.
-
(2006)
Bioorg. Med. Chem
, vol.14
, Issue.15
, pp. 5230-5240
-
-
Lesyk, R.1
Zimenkovsky, B.2
Atamanyuk, D.3
Jensen, F.4
Kiec-Kononowicz, K.5
Gzella, A.6
-
32
-
-
34248173947
-
New 5-substituted thiazolo[3,2-b][1,2,4]triazol-6-ones: Synthesis and anticancer evaluation
-
Lesyk R., Vladzimirska O., Holota S., Zaprutko L., Gzella A. New 5-substituted thiazolo[3,2-b][1,2,4]triazol-6-ones: synthesis and anticancer evaluation. Eur. J. Med. Chem. 2007. 42, N 5. P. 641-648.
-
(2007)
Eur. J. Med. Chem
, vol.5
, Issue.42
, pp. 641-648
-
-
Lesyk, R.1
Vladzimirska, O.2
Holota, S.3
Zaprutko, L.4
Gzella, A.5
-
33
-
-
42449130916
-
Synthesis and anti-cancer activity of novel thiopyrano[2,3-d]thiazole-based compounds containing norbornane moiety
-
Atamanyuk D., Zimenkovsky B., Lesyk R. Synthesis and anti-cancer activity of novel thiopyrano[2,3-d]thiazole-based compounds containing norbornane moiety. J. Sulf. Chem. 2008. 29, N 2. P. 151-162.
-
(2008)
J. Sulf. Chem
, vol.29
, Issue.2
, pp. 151-162
-
-
Atamanyuk, D.1
Zimenkovsky, B.2
Lesyk, R.3
-
34
-
-
45549086278
-
A new domino-Knoevenagel-hetero-Diels-Alder reaction
-
Matiychuk V. S., Lesyk R. B., Obushak M. D., Gzella A., Atamanyuk D. V., Ostapiuk Y. V., Kryshchyshyn A. P. A new domino-Knoevenagel-hetero-Diels-Alder reaction. Tetrahedron Lett. 2008. 49, N 31. P. 4648-4651.
-
(2008)
Tetrahedron Lett
, vol.49
, Issue.31
, pp. 4648-4651
-
-
Matiychuk, V.S.1
Lesyk, R.B.2
Obushak, M.D.3
Gzella, A.4
Atamanyuk, D.V.5
Ostapiuk, Y.V.6
Kryshchyshyn, A.P.7
-
35
-
-
61349169067
-
Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity
-
Havrylyuk D., Zimenkovsky B., Vasylenko O., Zaprutko L., Gzella A., Lesyk R. Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity. Eur. J. Med. Chem. 2009. 44, N 4. Р. 1396-1404.
-
(2009)
Eur. J. Med. Chem
, vol.44
, Issue.4
, pp. 1396-1404
-
-
Havrylyuk, D.1
Zimenkovsky, B.2
Vasylenko, O.3
Zaprutko, L.4
Gzella, A.5
Lesyk, R.6
-
36
-
-
67650456265
-
Synthesis and in vitro anticancer activity of 2,4-azolidinedione-acetic acids derivatives
-
Kaminskyy D., Zimenkovsky B., Lesyk R. Synthesis and in vitro anticancer activity of 2,4-azolidinedione-acetic acids derivatives. Eur. J. Med. Chem. 2009. 44, N 9. Р. 3627-3636.
-
(2009)
Eur. J. Med. Chem
, vol.44
, Issue.9
, pp. 3627-3636
-
-
Kaminskyy, D.1
Zimenkovsky, B.2
Lesyk, R.3
-
37
-
-
69249231104
-
Synthesis and antitumor activity of novel 2-thioxo-4-thiazolidinones with benzothiazole moieties
-
Mosula L., Zimenkovsky B., Havrylyuk D., Missir A.-V., Chirita I. C., Lesyk R. Synthesis and antitumor activity of novel 2-thioxo-4-thiazolidinones with benzothiazole moieties. Farmacia. 2009. 57, N 3. P. 321-330.
-
(2009)
Farmacia
, vol.57
, Issue.3
, pp. 321-330
-
-
Mosula, L.1
Zimenkovsky, B.2
Havrylyuk, D.3
Missir, A.-V.4
Chirita, I.C.5
Lesyk, R.6
-
38
-
-
61449246586
-
-
Phosphorus, Sulfur, and Silicon and the Related Elements
-
Havrylyuk D., Zimenkovsky B., Lesyk R. Synthesis and anticancer activity of novel nonfused bicyclic thiazolidinone derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements. 2009. 184, N 3. Р. 638-650.
-
(2009)
Synthesis and Anticancer Activity of Novel Nonfused Bicyclic Thiazolidinone Derivatives
, vol.184
, Issue.3
, pp. 638-650
-
-
Havrylyuk, D.1
Zimenkovsky, B.2
Lesyk, R.3
-
39
-
-
77955311711
-
Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activity
-
Subtel'na I., Atamanyuk D., Szymanska E., Kiec-Kononowicz K., Zimenkovsky B., Vasylenko O., Gzella A., Lesyk R. Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activity. Bioorg. Med. Chem. 2010. 18, N 14. P. 5090-5102.
-
(2010)
Bioorg. Med. Chem
, vol.18
, Issue.14
, pp. 5090-5102
-
-
Subtel'na, I.1
Atamanyuk, D.2
Szymanska, E.3
Kiec-Kononowicz, K.4
Zimenkovsky, B.5
Vasylenko, O.6
Gzella, A.7
Lesyk, R.8
-
40
-
-
77957844111
-
Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety
-
Havrylyuk D., Mosula L., Zimenkovsky B., Vasylenko O., Gzella A., Lesyk R. Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety. Eur. J. Med. Chem. 2010. 45, N 11. P. 5012-5021.
-
(2010)
Eur. J. Med. Chem
, vol.45
, Issue.11
, pp. 5012-5021
-
-
Havrylyuk, D.1
Mosula, L.2
Zimenkovsky, B.3
Vasylenko, O.4
Gzella, A.5
Lesyk, R.6
-
41
-
-
73949084441
-
Hybrid pharmacophore design and synthesis of isatin-benzothiazole analogs for their anti-breast cancer activity
-
Solomon V. R., Hu C., Lee H. Hybrid pharmacophore design and synthesis of isatin-benzothiazole analogs for their anti-breast cancer activity. Bioorg. Med. Chem. 2009. 17, N 21. P. 7585-7592.
-
(2009)
Bioorg. Med. Chem
, vol.17
, Issue.21
, pp. 7585-7592
-
-
Solomon, V.R.1
Hu, C.2
Lee, H.3
-
42
-
-
77952221554
-
Structure-anticancer activity relationships among 4-azolidinone-3-carboxylic acids derivatives
-
Kaminskyy D. V., Lesyk R. B. Structure-anticancer activity relationships among 4-azolidinone-3-carboxylic acids derivatives. Biopolym. Cell. 2010. 26, N 2. P. 136-145.
-
(2010)
Biopolym. Cell
, vol.26
, Issue.2
, pp. 136-145
-
-
Kaminskyy, D.V.1
Lesyk, R.B.2
-
43
-
-
67650346935
-
Synthesis and biological activity of 4-thiazolidinone-3-acetic acids derivatives
-
Каminskyy D. V., Lesyk R. B. Synthesis and biological activity of 4-thiazolidinone-3-acetic acids derivatives. Farmacevtychnyj Zhur. 2008. N 3. P. 70-78.
-
(2008)
Farmacevtychnyj Zhur
, vol.3
, pp. 70-78
-
-
Каminskyy, D.V.1
Lesyk, R.B.2
-
44
-
-
42449118666
-
5-Ylidene-2-thioxo-4-thiazolidinone-3-succinic acids and their derivatives: Synthesis, anticancer activity, QSAR-analysis
-
Каminskyy D. V., Roman O. M., Atamanyuk D. V., Lesyk R. B. 5-Ylidene-2-thioxo-4-thiazolidinone-3-succinic acids and their derivatives: synthesis, anticancer activity, QSAR-analysis. J. Org. Pharm. Chem. 2006. 4, N 1 (13). P. 41-48.
-
(2006)
J. Org. Pharm. Chem
, vol.4
, Issue.1-13
, pp. 41-48
-
-
Каminskyy, D.V.1
Roman, O.M.2
Atamanyuk, D.V.3
Lesyk, R.B.4
-
45
-
-
85038524792
-
Synthesis and antitumor activity evaluation of 3,5a,6,11b-tetrahydro-2H,5H-chromeno[4',3':4,5]thiopyrano[2,3-d]thiazole derivatives
-
Kryshchyshyn A. P., Zimenkovsky B. S., Zaprutko L., Lesyk R. B. Synthesis and antitumor activity evaluation of 3,5a,6,11b-tetrahydro-2H,5H-chromeno[4',3':4,5]thiopyrano[2,3-d]thiazole derivatives. J. Org. Pharm. Chem. 2010. 8, N 1 (29). P. 37-43.
-
(2010)
J. Org. Pharm. Chem
, vol.8
, Issue.1-29
, pp. 37-43
-
-
-
46
-
-
84860471866
-
Synthesis and anticancer activity in vitro of isothiochromеno[3,4-d]thiazole derivatives
-
Kryshchyshyn A., Zimenkovsky B., Lesyk R. Synthesis and anticancer activity in vitro of isothiochromеno[3,4-d]thiazole derivatives. Annal. UMCS. Sectio DDD. 2008. 21, N 1. P. 247-251.
-
(2008)
Annal. UMCS. Sectio DDD
, vol.21
, Issue.1
, pp. 247-251
-
-
Kryshchyshyn, A.1
Zimenkovsky, B.2
Lesyk, R.3
-
47
-
-
0036136167
-
COMPARE: A web accessible tool for investigating mechanisms of cell growth inhibition
-
Zaharevitz D. W., Holbeck S. L., Bowerman C., Svetlik P. A. COMPARE: a web accessible tool for investigating mechanisms of cell growth inhibition. J. Mol. Graph. Model. 2002. 20, N 4. P. 297-303.
-
(2002)
J. Mol. Graph. Model
, vol.20
, Issue.4
, pp. 297-303
-
-
Zaharevitz, D.W.1
Holbeck, S.L.2
Bowerman, C.3
Svetlik, P.A.4
-
48
-
-
0024312538
-
Display and analysis of patterns of differential activity of drugs against human tumor cell lines: Development of mean graph and COMPARE algorithm
-
Paull K. D., Shoemaker R. H., Hodes L., Monks A., Scudiero D. A., Rubinstein L., Plowman J., Boyd M. R. Display and analysis of patterns of differential activity of drugs against human tumor cell lines: development of mean graph and COMPARE algorithm. J. Natl Cancer Inst. 1989. 81, N 14. P. 1088-1092.
-
(1989)
J. Natl Cancer Inst
, vol.81
, Issue.14
, pp. 1088-1092
-
-
Paull, K.D.1
Shoemaker, R.H.2
Hodes, L.3
Monks, A.4
Scudiero, D.A.5
Rubinstein, L.6
Plowman, J.7
Boyd, M.R.8
-
49
-
-
5444274954
-
Identification of the protein binding region of S-trityl-L-cysteine, a new potent inhibitor of the mitotic kinesin Eg5
-
Brier S., Lemaire D., Debonis S., Forest E., Kozielski F. Identification of the protein binding region of S-trityl-L-cysteine, a new potent inhibitor of the mitotic kinesin Eg5. Biochemistry. 2004. 43, N 41. P. 13072-13082.
-
(2004)
Biochemistry
, vol.43
, Issue.41
, pp. 13072-13082
-
-
Brier, S.1
Lemaire, D.2
Debonis, S.3
Forest, E.4
Kozielski, F.5
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