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Archives of Biochemistry and Biophysics

Volumn 507, Issue 2, 2011, Pages 212-218

Harmine is an ATP-competitive inhibitor for dual-specificity tyrosine phosphorylation-regulated kinase 1A (Dyrk1A)

(3) Adayev, Tatyana a Wegiel, Jerzy a Hwang, Yu Wen a

a NEW YORK STATE INSTITUTE FOR BASIC RESEARCH IN DEVELOPMENTAL DISABILITIES (United States)

Author keywords

ATP binding pocket; Beta carbolines; Kinase inhibitors; Resistant mutants

Indexed keywords

ADENOSINE TRIPHOSPHATE; DUAL SPECIFICITY PHOSPHORYLATION REGULATED KINASE 1A; HARMINE; MAGNESIUM ION; PHOSPHOTRANSFERASE; UNCLASSIFIED DRUG;

ARTICLE; ENZYME ACTIVITY; ENZYME BINDING; ENZYME INHIBITION; ENZYME KINETICS; ENZYME PHOSPHORYLATION; ENZYME STRUCTURE; PRIORITY JOURNAL;

ADENOSINE TRIPHOSPHATE; ANIMALS; BINDING, COMPETITIVE; HARMINE; KINETICS; MICE; MUTAGENESIS, SITE-DIRECTED; MUTATION; NIH 3T3 CELLS; PROTEIN KINASE INHIBITORS; PROTEIN-SERINE-THREONINE KINASES; PROTEIN-TYROSINE KINASES; SUBSTRATE SPECIFICITY;

EID: 79951946396 PISSN: 00039861 EISSN: 10960384 Source Type: Journal
DOI: 10.1016/j.abb.2010.12.024 Document Type: Article

Times cited : (95)

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