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Volumn 5, Issue 10, 2010, Pages 1701-1705

20S proteasome inhibition: Designing noncovalent linear peptide mimics of the natural product TMC-95A

(11) Groll, Michael a Gallastegui, Nerea a Maréchal, Xavier b Le Ravalec, Virginie c Basse, Nicolas b Richy, Nicolas c Genin, Emilie c Huber, Robert d Moroder, Luis d Vidal, Jölle c Reboud Ravaux, Michèle b

a TECHNICAL UNIVERSITY OF MUNICH (Germany)

b SORBONNE UNIVERSITÉ (France)

c UNIVERSITÉ DE RENNES 1 (France)

d MAX PLANCK INSTITUTE OF BIOCHEMISTRY (Germany)

Author keywords

Crystallographic analysis; Enzymes; Inhibitors; Natural products; Proteasomes

Indexed keywords

3 HYDROXY 2 OXYINDOLE; LACTACYSTIN BETA LACTONE; OXINDOLE; PROTEASOME; PROTEASOME INHIBITOR; SALINOSPORAMIDE A; TMC 95A; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ARTICLE; COMPLEX FORMATION; COVALENT BOND; CRYSTAL STRUCTURE; DRUG STRUCTURE; ENZYME INHIBITION; ENZYME SPECIFICITY; HYDROGEN BOND; IC 50; PRIORITY JOURNAL;

BINDING SITES; CATALYTIC DOMAIN; CRYSTALLOGRAPHY, X-RAY; PEPTIDES, CYCLIC; PROTEASE INHIBITORS; PROTEASOME ENDOPEPTIDASE COMPLEX;

EID: 77957656769 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000293 Document Type: Article

Times cited : (47)

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