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Volumn 2, Issue SUPPL. 1, 2010, Pages 79-85

Transdermal delivery of ibuprofen and its prodrugs by passive diffusion and iontophoresis

Author keywords

Ibuprofen; Iontophoresis; Prodrug; Transdermal

Indexed keywords

2,4, ISOBUTYL PHENYL ETHYL PROPIONATE; IBUPROFEN; PRODRUG; UNCLASSIFIED DRUG;

EID: 77953427178     PISSN: None     EISSN: 09751491     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (11)

References (40)
  • 1
    • 23944473192 scopus 로고    scopus 로고
    • Synthesis and transdermal penetration of NSAID glycoside esters
    • Henk S, Jaco CB, Jonathan H, Jeanetta du P. Synthesis and transdermal penetration of NSAID glycoside esters. Int J Pharm 2005; 301: 71-79.
    • (2005) Int J Pharm , vol.301 , pp. 71-79
    • Henk, S.1    Jaco, C.B.2    Jonathan, H.3    Jeanetta du, P.4
  • 2
    • 20644441011 scopus 로고    scopus 로고
    • Determination of ibuprofen in dog plasma by liquid chromatography and application in pharmacokinetic studies of an ibuprofen prodrug in dogs
    • Peng W, Meiling Q, Lihe L, Lin F. Determination of ibuprofen in dog plasma by liquid chromatography and application in pharmacokinetic studies of an ibuprofen prodrug in dogs. J Pharm Biomed Anal 2005; 38: 714-719.
    • (2005) J Pharm Biomed Anal , vol.38 , pp. 714-719
    • Peng, W.1    Meiling, Q.2    Lihe, L.3    Lin, F.4
  • 3
    • 77953386471 scopus 로고    scopus 로고
    • Synthesis, pharmacological activity and hydrolytic behavior of ethylenediamine and benzathine conjugates of ibuprofen
    • Nithar RC, Amol AK, Santosh PG. Synthesis, pharmacological activity and hydrolytic behavior of ethylenediamine and benzathine conjugates of ibuprofen. Eur J Med Chem 2007; 20: 1-5
    • (2007) Eur J Med Chem , vol.20 , pp. 1-5
    • Nithar, R.C.1    Amol, A.K.2    Santosh, P.G.3
  • 4
    • 0034898142 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of ketoprofen, naproxen and diclofenac
    • Francesco P B, Carmelo P, Tony B, Paolo de C, Francesco P, Maria G R, Antonella S. In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of ketoprofen, naproxen and diclofenac. Eur J Pharm Sci 2001; 14: 123-134.
    • (2001) Eur J Pharm Sci , vol.14 , pp. 123-134
    • Francesco, P.B.1    Carmelo, P.2    Tony, B.3    Paolo de, C.4    Francesco, P.5    Maria, G.R.6    Antonella, S.7
  • 5
    • 33750522775 scopus 로고    scopus 로고
    • Pharmacological activity and hydrolysis behavior of novel ibuprofen glucopyranoside conjugates
    • Xiangguo Z, Xinyi T, Dongzhi W, Qingxun. Pharmacological activity and hydrolysis behavior of novel ibuprofen glucopyranoside conjugates. Eur J Med Chem 2006; 41: 1352- 1358
    • (2006) Eur J Med Chem , vol.41 , pp. 1352-1358
    • Xiangguo, Z.1    Xinyi, T.2    Dongzhi, W.3    Qingxun4
  • 6
    • 33646797058 scopus 로고    scopus 로고
    • Synthesis and study of controlled release of ibuprofen from the new acrylic type polymers
    • Mirzaagha B. Synthesis and study of controlled release of ibuprofen from the new acrylic type polymers. Int J Pharm 2006; 316: 68-73.
    • (2006) Int J Pharm , vol.316 , pp. 68-73
    • Mirzaagha, B.1
  • 7
    • 26444539505 scopus 로고    scopus 로고
    • Synthesis of ibuprofen eugenol ester and its Microemulsion Formulation for Parenteral Delivery
    • Xiuli Z, Dawei C, Ping G, Pingtian D, and Kexin. Synthesis of ibuprofen eugenol ester and its Microemulsion Formulation for Parenteral Delivery. Chem Pharm Bull53(10) 1246-1250 (2005).
    • (2005) Chem Pharm Bull53 , pp. 1246-1250
    • Xiuli, Z.1    Dawei, C.2    Ping, G.3    Pingtian, D.4    Kexin5
  • 8
    • 77953457451 scopus 로고    scopus 로고
    • J Aukunuru1, C Bonepally and V Guduri. Preparation, characterization and optimization of ibuprofen ointment intended for topical and systemic delivery. Trop J Pharmaceut Res 2007; 6 (4): 855-860.
    • J Aukunuru1, C Bonepally and V Guduri. Preparation, characterization and optimization of ibuprofen ointment intended for topical and systemic delivery. Trop J Pharmaceut Res 2007; 6 (4): 855-860.
  • 9
    • 0032472340 scopus 로고    scopus 로고
    • Paul WS, Adrian CW and Brian WB. Transdermal delivery from eutectic systems: enhanced permeation of a model drug, ibuprofen. J Contr Release 1998; 50: 297-308
    • Paul WS, Adrian CW and Brian WB. Transdermal delivery from eutectic systems: enhanced permeation of a model drug, ibuprofen. J Contr Release 1998; 50: 297-308.
  • 10
    • 17844389701 scopus 로고    scopus 로고
    • SE Cross and MS Roberts. Physical enhancement of transdermal drug application: is delivery technology keeping up with pharmaceutical development? Curr Drug Deliv 2004; 1: 81-92.
    • SE Cross and MS Roberts. Physical enhancement of transdermal drug application: is delivery technology keeping up with pharmaceutical development? Curr Drug Deliv 2004; 1: 81-92.
  • 12
    • 17844373273 scopus 로고    scopus 로고
    • Transdermal drug delivery: Penetration enhancement techniques
    • Heather AE, Benson. Transdermal drug delivery: penetration enhancement techniques. Curr Drug Deliv 2005; 2:23-33.
    • (2005) Curr Drug Deliv , vol.2 , pp. 23-33
    • Heather, A.E.1    Benson2
  • 13
    • 0023235207 scopus 로고
    • Effect of penetration enhancers on the permeaton of mannitol hydrocortisone and progesterone through human skin
    • Barry BW, Bennett SL. Effect of penetration enhancers on the permeaton of mannitol hydrocortisone and progesterone through human skin. J Pharm Pharmacol 1987; 39:535-546.
    • (1987) J Pharm Pharmacol , vol.39 , pp. 535-546
    • Barry, B.W.1    Bennett, S.L.2
  • 14
    • 28244485413 scopus 로고    scopus 로고
    • Guang Yan, S Kevin Li, William IH. Evaluation of constant current alternating current iontophoresis for transdermal drug delivery. J Contr Release 2005; 110:141-150
    • Guang Yan, S Kevin Li, William IH. Evaluation of constant current alternating current iontophoresis for transdermal drug delivery. J Contr Release 2005; 110:141-150.
  • 15
  • 17
    • 34547707208 scopus 로고    scopus 로고
    • Iontophoretic drug delivery
    • N.K. Jain, ed, C.B.S. Publishers and Distributors, New Delhi
    • RK Khar and A Nanda, Iontophoretic drug delivery, in: Controlled and novel drug delivery system, N.K. Jain, ed., C.B.S. Publishers and Distributors, New Delhi, 2005; 191-207.
    • (2005) Controlled and novel drug delivery system , pp. 191-207
    • Khar, R.K.1    Nanda, A.2
  • 18
    • 33846090269 scopus 로고    scopus 로고
    • Iontophoresis - An approach for controlled drug delivery: A Review
    • Nitin D, Vikas B, Sanjula B, Alka A and Javed A. Iontophoresis - An approach for controlled drug delivery: A Review. Curr Drug Deliv 2007; 4: 1-10.
    • (2007) Curr Drug Deliv , vol.4 , pp. 1-10
    • Nitin, D.1    Vikas, B.2    Sanjula, B.3    Alka, A.4    Javed, A.5
  • 19
    • 77953416025 scopus 로고    scopus 로고
    • rd ed. Newyork: A Wiley interscience publications; 2004. p.240,348-351.
    • rd ed. Newyork: A Wiley interscience publications; 2004. p.240,348-351.
  • 21
    • 0033987103 scopus 로고    scopus 로고
    • The influence of the physicochemical characteristics and pharmacokinetic properties of selected NSAID's on their transdermal absorption
    • Estelle B, Jeanetta P, Douw GM, Colleen G, Francois JR. The influence of the physicochemical characteristics and pharmacokinetic properties of selected NSAID's on their transdermal absorption. Int J Pharm 2000; 193:261-264.
    • (2000) Int J Pharm , vol.193 , pp. 261-264
    • Estelle, B.1    Jeanetta, P.2    Douw, G.M.3    Colleen, G.4    Francois, J.R.5
  • 23
    • 4043124619 scopus 로고    scopus 로고
    • Efficacy of topical non-steroidal anti-inflammatory drugs in the treatment of osteoarthritis: Meta-analysis of randomized controlled trials
    • Jinying L, Weiya Z, Adrian J, Michael D. Efficacy of topical non-steroidal anti-inflammatory drugs in the treatment of osteoarthritis: meta-analysis of randomized controlled trials. BMJ, 2004; 329:324.
    • (2004) BMJ , vol.329 , pp. 324
    • Jinying, L.1    Weiya, Z.2    Adrian, J.3    Michael, D.4
  • 24
    • 0026557715 scopus 로고
    • Ester and amide prodrugs of ibuprofen and naproxen; synthesis, ant-inflammatory activity and gastrointestinal toxicity
    • Vrinda R. Shanbhag, A. Michael C, Rajeev G, Anju H, Ronald MD. Ester and amide prodrugs of ibuprofen and naproxen; synthesis, ant-inflammatory activity and gastrointestinal toxicity. J Pharm Sci 1992; 81:249-154.
    • (1992) J Pharm Sci , vol.81 , pp. 249-154
    • Vrinda, R.1    Shanbhag, A.2    Michael, C.3    Rajeev, G.4    Anju, H.5    Ronald, M.D.6
  • 25
    • 77953472520 scopus 로고    scopus 로고
    • Therapeutic outcome confirmed for transdermal ibuprofen, pharmalicencing.com; TransDermal Technologies, Inc. PressRelease issued 5th February 2002.
    • Therapeutic outcome confirmed for transdermal ibuprofen, pharmalicencing.com; TransDermal Technologies, Inc. PressRelease issued 5th February 2002.
  • 26
    • 40749130499 scopus 로고    scopus 로고
    • In vivo pharmacokinetic studies of prodrugs of ibuprofen
    • Abha D, Deshpande SG. In vivo pharmacokinetic studies of prodrugs of ibuprofen. Indian J Pharmaceut Sci 2007; 69:824- 827.
    • (2007) Indian J Pharmaceut Sci , vol.69 , pp. 824-827
    • Abha, D.1    Deshpande, S.G.2
  • 28
    • 0034687579 scopus 로고    scopus 로고
    • Sang-Cheol Chi. Enhancing effect of polyoxyethylene alkyl ethers on the skin permeation of ibuprofen
    • Eun-Seok P, Si-Young C Mikyoung H, Sang-Cheol Chi. Enhancing effect of polyoxyethylene alkyl ethers on the skin permeation of ibuprofen. Int J Pharm 2000; 209:109-119.
    • (2000) Int J Pharm , vol.209 , pp. 109-119
    • Eun-Seok, P.1    Si-Young, C.2    Mikyoung, H.3
  • 29
    • 0023567428 scopus 로고
    • Effects of vehicles and prodrug properties and their interactions on the delivery of 6-mercaptopurine through skin: Bisacyloxymethyl-6-mercaptopurine prodrugs
    • Waranis RP, Sloan KB. Effects of vehicles and prodrug properties and their interactions on the delivery of 6-mercaptopurine through skin: bisacyloxymethyl-6-mercaptopurine prodrugs. J Pharm Sci 1987; 76: 587-95.
    • (1987) J Pharm Sci , vol.76 , pp. 587-595
    • Waranis, R.P.1    Sloan, K.B.2
  • 31
    • 0032767766 scopus 로고
    • Synthesis and evaluation of anti-inflamamtory activity of 2-(4 isobutyl phenyl) propionyl derivatives of amino acids and peptides
    • Belagali SL, Himaja M. Synthesis and evaluation of anti-inflamamtory activity of 2-(4 isobutyl phenyl) propionyl derivatives of amino acids and peptides. Ind J Chem 1991; 38: 505-507.
    • (1991) Ind J Chem , vol.38 , pp. 505-507
    • Belagali, S.L.1    Himaja, M.2
  • 32
    • 0036143282 scopus 로고    scopus 로고
    • New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: Synthesis, physicochemical properties, and skin permeation studies
    • Bonina FP, Rimoli MG, Avallone L, Barbato F, Amato M, Puglia C. et al. New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical properties, and skin permeation studies. J Pharm Sci 2002; 91: 171.
    • (2002) J Pharm Sci , vol.91 , pp. 171
    • Bonina, F.P.1    Rimoli, M.G.2    Avallone, L.3    Barbato, F.4    Amato, M.5    Puglia, C.6
  • 36
    • 0031754210 scopus 로고    scopus 로고
    • Prodrugs of gestodene for matrix-type transdermal drug delivery systems
    • Lipp R, Laurent H, Gunther C, Riedl J, Esperling P, Tauber U. Prodrugs of gestodene for matrix-type transdermal drug delivery systems. Pharm Res 1998; 15: 1419-24.
    • (1998) Pharm Res , vol.15 , pp. 1419-1424
    • Lipp, R.1    Laurent, H.2    Gunther, C.3    Riedl, J.4    Esperling, P.5    Tauber, U.6
  • 37
    • 19344374256 scopus 로고    scopus 로고
    • The effects of electrically assisted methods on transdermal delivery of nalbuphine benzoate and sebacoyl dinalbuphine ester from solutions and hydrogels
    • Jeng-Fen H, Sunga KC, Oliver YH, Jhi-Joung W, Yi-Hsin L, Jia-You F. The effects of electrically assisted methods on transdermal delivery of nalbuphine benzoate and sebacoyl dinalbuphine ester from solutions and hydrogels. Int J Pharm 2005; 297:162-171.
    • (2005) Int J Pharm , vol.297 , pp. 162-171
    • Jeng-Fen, H.1    Sunga, K.C.2    Oliver, Y.H.3    Jhi-Joung, W.4    Yi-Hsin, L.5    Jia-You, F.6
  • 38
    • 67650096770 scopus 로고    scopus 로고
    • Transdermal delivery of atenolol: Effect of prodrugs and iontophoresis
    • Anroop B, Ghosh B, Parcha V, Khanam J. Transdermal delivery of atenolol: Effect of prodrugs and iontophoresis. Curr Drug Deliv 2009; 6: 280-290.
    • (2009) Curr Drug Deliv , vol.6 , pp. 280-290
    • Anroop, B.1    Ghosh, B.2    Parcha, V.3    Khanam, J.4
  • 39
    • 0033976976 scopus 로고    scopus 로고
    • Guy RH, Kalia YN, Delgado-Charro MB, Merino V, Lopez A, Marro D. Iontophoresis: electrorepulsion and electroosmosis. J Control Release 2000; 64: 129-32
    • Guy RH, Kalia YN, Delgado-Charro MB, Merino V, Lopez A, Marro D. Iontophoresis: electrorepulsion and electroosmosis. J Control Release 2000; 64: 129-32.
  • 40
    • 0035289973 scopus 로고    scopus 로고
    • The role of electroosmotic flow in transdermal iontophoresis
    • Michael JP. The role of electroosmotic flow in transdermal iontophoresis. Adv Drug Deliv Rev 2001; 46: 281-305.
    • (2001) Adv Drug Deliv Rev , vol.46 , pp. 281-305
    • Michael, J.P.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.