New oligoethylene ester derivatives of 5-iodo-2′-deoxyuridine as dermal prodrugs: Synthesis, physicochemical properties, and skin permeation studies

Journal of Pharmaceutical Sciences

Volumn 91, Issue 1, 2002, Pages 171-179

  Bonina, Francesco Paolo ^a   Rimoli, Maria Grazia ^b   Avallone, Lucia ^b   Barbato, Francesco ^b   Amato, Marzia ^b   Puglia, Carmelo ^a   Ricci, Maurizio ^c   De Caprariis, Paolo ^d  

^a UNIVERSITY OF CATANIA   (Italy)

^b UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^c UNIVERSITY OF PERUGIA   (Italy)

^d UNIVERSITY OF SASSARI   (Italy)

Author keywords

Dermal prodrugs; IDU; In vitro; SCE membranes

Indexed keywords

DIETHYLENE GLYCOL 3' O SUCCINYL 5 IODO 2' DEOXYURIDINE ESTER DERIVATIVE; ESTER DERIVATIVE; HEXAETHYLENE GLYCOL 3' O SUCCINYL 5 IODO 2' DEOXYURIDINE ESTER DERIVATIVE; IDOXURIDINE; PENTAETHYLENE GLYCOL 3' O SUCCINYL 5 IODO 2' DEOXYURIDINE ESTER DERIVATIVE; PRODRUG; TETRAETHYLENE GLYCOL 3' O SUCCINYL 5 IODO 2' DEOXYURIDINE ESTER DERIVATIVE; TRIETHYLENE GLYCOL 3' O SUCCINYL 5 IODO 2' DEOXYURIDINE ESTER DERIVATIVE; UNCLASSIFIED DRUG;

ADULT; ARTICLE; DRUG ABSORPTION; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN TISSUE; IN VITRO STUDY; LIPOPHILICITY; PARTITION COEFFICIENT; SKIN PERMEABILITY;

EID: 0036143282     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/jps.1174     Document Type: Article

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