Exploration of inhibitors for diaminopimelate aminotransferase

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 6, 2010, Pages 2141-2151

  Fan, Chenguang ^a   Clay, Matthew D ^b   Deyholos, Michael K ^a   Vederas, John C ^a  

^a UNIVERSITY OF ALBERTA   (Canada)

^b St Mary's University College   (Canada)

Author keywords

Aminotransferase; Arabidopsis thaliana; Chlamydia; Diaminopimelate (DAP); Enzyme inhibition; Lysine biosynthesis; Pyridoxal 5 phosphate (PLP)

Indexed keywords

AMINOTRANSFERASE; AMINOTRANSFERASE INHIBITOR; ANTIBIOTIC AGENT; DIAMINOPIMELATE AMINOTRANSFERASE; DIAMINOPIMELATE AMINOTRANSFERASE INHIBITOR; HERBICIDE; PYRIDOXAL 5 PHOSPHATE; UNCLASSIFIED DRUG;

ARABIDOPSIS; ARTICLE; CATALYSIS; CHLAMYDIA; DRUG DESIGN; DRUG SYNTHESIS; ENZYME INHIBITOR INTERACTION; IC 50; NONHUMAN; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

DIAMINOPIMELIC ACID; DRUG DESIGN; ENZYME INHIBITORS; HYDRAZINES; MOLECULAR STRUCTURE; RHODANINE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSAMINASES;

ARABIDOPSIS THALIANA; CHLAMYDIA; EMBRYOPHYTA; MAMMALIA;

EID: 77649233456     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.02.001     Document Type: Article

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