Phenoxy herbicides and fibrates potently inhibit the human chemosensory receptor subunit T1R3

Journal of Medicinal Chemistry

Volumn 52, Issue 21, 2009, Pages 6931-6935

  Maillet, Emeline L ^a   Margolskee, Robert F ^b   Mosinger, Bedrich ^b  

^a MOUNT SINAI SCHOOL OF MEDICINE   (United States)

^b MONELL CHEMICAL SENSES CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID DERIVATIVE; CALCIUM; DNA; FIBRIC ACID DERIVATIVE; G PROTEIN COUPLED RECEPTOR; HERBICIDE; LACTISOLE; PHENOXY HERBICIDE; PHENOXYAURIN; PROTEIN SUBUNIT; PROTEIN T1R3; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CHEMICAL STRUCTURE; CONTROLLED STUDY; HUMAN; HUMAN CELL; HYPERLIPIDEMIA; NON INSULIN DEPENDENT DIABETES MELLITUS; NONHUMAN; PROTEIN DOMAIN; PROTEIN EXPRESSION;

2,4-DICHLOROPHENOXYACETIC ACID; ANIMALS; ANTILIPEMIC AGENTS; BENZENE DERIVATIVES; BEZAFIBRATE; CELL LINE; CERCOPITHECIDAE; CLOFIBRIC ACID; GEMFIBROZIL; HERBICIDES; HUMANS; INDOLEACETIC ACIDS; MICE; PROTEIN SUBUNITS; RECEPTORS, G-PROTEIN-COUPLED; RECOMBINANT FUSION PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 71049152983     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm900823s     Document Type: Article

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