Corrigendum to "Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C" [Bioorg. Med. Chem. Lett. 19 (2009) 5392] (DOI:10.1016/j.bmcl.2009.07.114);Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 18, 2009, Pages 5392-5396

  Guay, Daniel ^a   Beaulieu, Christian ^a   Jagadeeswar Reddy, T ^a   Zamboni, Robert ^a   Methot, Nathalie ^a   Rubin, Joel ^a   Ethier, Diane ^a   David Percival, M ^a  

^a MERCK FROSST CENTRE FOR THERAPEUTIC RESEARCH   (Canada)

Author keywords

Cathepsin C; Dipeptide nitrile; Dipeptidyl peptidase I

Indexed keywords

ALANINE DERIVATIVE; ANTIINFLAMMATORY AGENT; CYCLOPROPANE DERIVATIVE; DIPEPTIDYL NITRILE DERIVATIVE; DIPEPTIDYL PEPTIDASE I; ENZYME INHIBITOR; HYDROLASE; N [N (3 CARBOXYOXIRANE 2 CARBONYL)LEUCYL]AGMATINE; NITRILE; SULFUR; THIENYL ALANINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; DRUG CLEARANCE; DRUG CYTOTOXICITY; DRUG DESIGN; DRUG HALF LIFE; DRUG MECHANISM; DRUG METABOLISM; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PROTEIN FUNCTION; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALS; CATHEPSIN C; CELL LINE; DIPEPTIDES; HUMANS; NITRILES; RATS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 68949132704     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.09.043     Document Type: Erratum

References (29)

1. Ishidoh K., Muno D., Sato N., and Kominami E. J. Biol. Chem. 266 (1991) 16312
2. McGuire M.J., Lipsky P.E., and Thiele D.L. Arch. Biochem. Biophys. 295 (1992) 280
3. Mallen-St Clair J., Pham C.T., Villalta S.A., Caughey G.H., and Wolters P.J. J. Clin. Invest. 113 (2004) 628
4. Adkinson A.M., Raptis S.Z., Kelley D.G., and Pham C.T. J. Clin. Invest. 109 (2002) 363
5. Pham C.T., and Ley T.J. Proc. Natl. Acad. Sci. U.S.A. 96 (1999) 8627
6. Wolters P.J., Pham C.T., Muilenburg D.J., Ley T.J., and Caughey G.H. J. Biol. Chem. 276 (2001) 18551
7. Sheth P.D., Pedersen J., Walls A.F., and McEuen A.R. Biochem. Pharmacol. 66 (2003) 2251
8. Ohbayashi H. IDrugs 5 (2002) 910
9. Conese M., Copreni E., DiGioia S., DeRinaldis P., and Fumarulo R. J. Cyst. Fibros. 2 (2003) 129
10. Turk D., Janjic V., Stern D., Podobnik M., Lamba D., Dahl S., Lauritzen C., Pedersen J., Turk V., and Tuck B. EMBO 20 (2001) 6570
11. Molgaard A., Arnau J., Lauritzen C., Larsen S., Petersen G., and Pedersen J. Biochem. J. 401 (2007) 645
12. Tran T.V., Ellis K.A., Kam C.-M., Hudig D., and Powers J.C. Arch. Biochem. Biophys. 403 (2002) 160
13. Thiele, D. L.; Lipsky, P. E.; McGuire, M. J. U.S. Patent 5602,102, 1997.
14. Green G.D.J., and Shaw E. J. Biol. Chem. 256 (1981) 1923
15. Kam C.-M., Götz M.G., Koot G., McGuire M., Thiele D., Hudig D., and Powers J.C. Arch. Biochem. Biophys. 427 (2004) 123
16. Yuan F., Verhelst S.H.L., Blum G., Coussens L.M., and Bogyo M. J. Am. Chem. Soc. 128 (2006) 5616
17. Demuth, H.-U.; Heiser, U.; Niestroj, A. WO 03/022871 A2, 2003.
18. Barrett A.J., Kembhavi A.A., Brown M.A., Kirschke H., Knight C.G., Tamai M., and Hanada K. Biochem. J. 201 (1982) 189
19. Thompson S.A., Andrews P.R., and Hanzlik R.P. J. Med. Chem. 29 (1986) 104
20. Bondebjerg J., Fuglsang H., Valeur K.R., Pedersen J., and Naerum L. Bioorg. Med. Chem. Lett. 16 (2006) 3614
21. Bondebjerg J., Fuglsang H., Valeur K.R., Kaznelson D.W., Hansen J.A., Pedersen R.O., Krogh B.O., Jensen B.S., Lauritzen C., Petersen G., Pedersen J., and Naerum L. Bioorg. Med. Chem. 13 (2005) 4408
22. Horn M., Pavlik M., Doleckova L., Baudys M., and Mares M. Eur. J. Biochem. 267 (2000) 3330
23. Mucha A., Pawelczak M., Hurek J., and Kafarski P. Bioorg. Med. Chem. Lett. 14 (2004) 3113
24. Gauthier J.Y., Black W.C., Courchesne I., Cromlish W., Desmarais S., Houle R., Lamontagne S., Li C.S., Massé F., McKay D.J., Ouellet M., Robichaud J., Truchon J.-F., Truong V.-L., Wang Q., and Percival M.D. Bioorg. Med. Chem. Lett. 17 (2007) 4929
25. Gauthier J.Y., Chauret N., Cromlish W., Desmarais S., Duong L.T., Falgueyret J.-P., Kimmel D.B., Lamontagne S., Léger S., LeRiche T., Li C.S., Massé F., McKay D.J., Nicoll-Griffith D.A., Oballa R.M., Palmer J.T., Percival M.D., Riendeau D., Robichaud J., Rodan G.A., Rodan S.B., Seto C., Thérien M., Truong V.-L., Venuti M.C., Wesolowski G., Young R.N., Zamboni R., and Black W.C. Bioorg. Med. Chem. Lett. 18 (2008) 923
26. Robichaud J., Black W.C., Thérien M., Paquet J., Oballa R.M., Bayly C.I., McKay D.J., Wang Q., Isabel E., Léger S., Mellon C., Kimmel D.B., Wesolowski G., Percival M.D., Massé F., Desmarais S., Falgueyret J.P., and Crane S.N. J. Med. Chem. 51 (2008) 6410
27. Davies H.M.L., Bruzinski P.R., Lake D.H., Kong N., and Fall M.J. J. Am. Chem. Soc. 118 (1996) 6897
28. Methot N., Rubin J., Guay D., Beaulieu C., Ethier D., Reddy T.J., Riendeau D., and Percival M.D. J. Biol. Chem. 282 (2007) 20836
29. Methot N., Guay D., Rubin J., Ethier D., Ortega K., Wong S., Normandin D., Beaulieu C., Reddy T.J., Riendeau D., and Percival M.D. Mol. Pharmacol. 73 (2008) 1857