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Volumn 50, Issue 5, 1996, Pages 1364-1375

Pharmacology of the human γ-aminobutyric acid(A) receptor α4 subunit expressed in Xenopus laevis oocytes

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; 8 AZIDO 5,6 DIHYDRO 5 METHYL 6 OXO 4H IMIDAZO[1,5 A][1,4]BENZODIAZEPINE 3 CARBOXYLIC ACID ETHYL ESTER; BRETAZENIL; DIAZEPAM; FLUMAZENIL;

EID: 0029807606     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (82)

References (49)
  • 4
    • 0002437069 scopus 로고
    • A receptor channel: A mechanism for interaction with a multitude of central nervous system functions
    • (H. Möhler and M. Da Prada, eds.). Roche, Basel
    • A receptor channel: a mechanism for interaction with a multitude of central nervous system functions, in The Challenge of Neuropharmacology (H. Möhler and M. Da Prada, eds.). Roche, Basel, 15-39 (1994).
    • (1994) The Challenge of Neuropharmacology , pp. 15-39
    • Haefely, W.E.1
  • 10
    • 0025193448 scopus 로고
    • γ-Aminobutyric acid A receptor α5-subunit creates novel type II benzodiazepine receptor pharmacology
    • Pritchett, D. B., and P. H. Seeburg. γ-Aminobutyric acid A receptor α5-subunit creates novel type II benzodiazepine receptor pharmacology. J. Neurochem. 54:1802-1804 (1990).
    • (1990) J. Neurochem. , vol.54 , pp. 1802-1804
    • Pritchett, D.B.1    Seeburg, P.H.2
  • 14
    • 0026612363 scopus 로고
    • A receptor subunit mRNAs in the rat brain. I. Telencephalon, diencephalon, mesencephalon
    • A receptor subunit mRNAs in the rat brain. I. Telencephalon, diencephalon, mesencephalon. J. Neurosci. 12:1040-1062 (1992).
    • (1992) J. Neurosci. , vol.12 , pp. 1040-1062
    • Wisden, W.1    Laurie, D.J.2    Monyer, H.3    Seeburg, P.H.4
  • 15
    • 0026615116 scopus 로고
    • - ion channels modulated by multiple drug Binding sites
    • - ion channels modulated by multiple drug Binding sites. Trends Pharmacol. Sci. 18:446-450 (1992).
    • (1992) Trends Pharmacol. Sci. , vol.18 , pp. 446-450
    • Sieghart, W.1
  • 16
    • 0026052215 scopus 로고
    • The clinical use of barbiturates in neurological disorders
    • Smith, M. C., and B. J. Riskin. The clinical use of barbiturates in neurological disorders. Drugs 42:365-378 (1991).
    • (1991) Drugs , vol.42 , pp. 365-378
    • Smith, M.C.1    Riskin, B.J.2
  • 19
    • 0028801074 scopus 로고
    • A receptor complex: The pharmacological properties and therapeutic potential of epalons
    • A receptor complex: the pharmacological properties and therapeutic potential of epalons. Crit. Rev. Neurobiol. 9:207-227 (1995).
    • (1995) Crit. Rev. Neurobiol. , vol.9 , pp. 207-227
    • Gee, K.W.1    McCauley, L.D.2    Lan, N.C.3
  • 21
    • 0028987216 scopus 로고
    • Different subunit requirements for volatile and nonvolatile anesthetics at γ-aminobutyric acid type A receptors
    • Harris, B. D., G. Wong, E. J. Moody, and P. Skolnick. Different subunit requirements for volatile and nonvolatile anesthetics at γ-aminobutyric acid type A receptors. Mol. Pharmacol. 47:363-367 (1995).
    • (1995) Mol. Pharmacol. , vol.47 , pp. 363-367
    • Harris, B.D.1    Wong, G.2    Moody, E.J.3    Skolnick, P.4
  • 22
    • 0025917512 scopus 로고
    • GABA receptor mechanisms in the central nervous system
    • Sivilotti, L., and A. Nistri. GABA receptor mechanisms in the central nervous system. Prog. Neurobiol. 36:35-92 (1991).
    • (1991) Prog. Neurobiol. , vol.36 , pp. 35-92
    • Sivilotti, L.1    Nistri, A.2
  • 23
    • 0028981088 scopus 로고
    • A receptor subtypes
    • A receptor subtypes. Pharmacol. Rev. 47:181-234 (1995).
    • (1995) Pharmacol. Rev. , vol.47 , pp. 181-234
    • Sieghart, W.1
  • 24
    • 0024471585 scopus 로고
    • 3H]Ro15-4513 binding in intact cultured cerebellar granule cells
    • 3H]Ro15-4513 binding in intact cultured cerebellar granule cells. Eur. J. Pharmacol. 169:53-60 (1989).
    • (1989) Eur. J. Pharmacol. , vol.169 , pp. 53-60
    • Malminiemi, O.1    Korpi, E.R.2
  • 27
    • 0025193448 scopus 로고
    • γ-Aminobutyric acid A receptor α5-subunit creates novel type II benzodiazepine receptor pharmacology
    • Pritchett, D. B., and P. H. Seeburg. γ-Aminobutyric acid A receptor α5-subunit creates novel type II benzodiazepine receptor pharmacology. J. Neurochem. 54:1802-1804 (1990).
    • (1990) J. Neurochem. , vol.54 , pp. 1802-1804
    • Pritchett, D.B.1    Seeburg, P.H.2
  • 31
    • 0028972886 scopus 로고
    • A receptor α4 subunit: Identification of a unique diazepam-insensitive binding site
    • A receptor α4 subunit: identification of a unique diazepam-insensitive binding site. Eur. J. Pharmacol. 291:319-325 (1995).
    • (1995) Eur. J. Pharmacol. , vol.291 , pp. 319-325
    • Yang, W.1    Drewe, J.A.2    Lan, N.C.3
  • 32
    • 0028177173 scopus 로고
    • 3H]Ro15-4513 binding in rodent brain and cultured cerebellar neuronal cells
    • 3H]Ro15-4513 binding in rodent brain and cultured cerebellar neuronal cells. Neurochem. Res. 19:289-295 (1994).
    • (1994) Neurochem. Res. , vol.19 , pp. 289-295
    • Ito, Y.1    Abiko, E.2    Mitaani, K.3    Fukuda, H.4
  • 38
    • 0026438362 scopus 로고
    • Partial agonists of benzodiazepine receptors for the treatment of epilepsy, sleep, and anxiety disorders
    • (G. Biggio, A. Concas, and E. Costa, eds.). Raven Press, New York
    • Haefely, W., M. Fackham, P. Schoch, J. R. Martin, E. P. Bonetti, J.-L. Moreau, F. Jenck, and J. G. Richards. Partial agonists of benzodiazepine receptors for the treatment of epilepsy, sleep, and anxiety disorders, in GABAergic Synoptic Transmission (G. Biggio, A. Concas, and E. Costa, eds.). Raven Press, New York, 379-394 (1992).
    • (1992) GABAergic Synoptic Transmission , pp. 379-394
    • Haefely, W.1    Fackham, M.2    Schoch, P.3    Martin, J.R.4    Bonetti, E.P.5    Moreau, J.-L.6    Jenck, F.7    Richards, J.G.8
  • 39
    • 0023612491 scopus 로고
    • Pharmacology of the pyrazolo-type compounds: Agonist, antagonist and inverse agonist actions
    • Bennett, D. A. Pharmacology of the pyrazolo-type compounds: agonist, antagonist and inverse agonist actions. Physiol. Behav. 41:241-245 (1987).
    • (1987) Physiol. Behav. , vol.41 , pp. 241-245
    • Bennett, D.A.1
  • 42
    • 0026495803 scopus 로고
    • Effects of the triazole derivative loreclezole (R72063) on stimulus induced ionic and field potential responses and on different patterns of epileptiform activity induced by low magnesium in rat entorhinal cortex-hippocampal slices
    • Zhang, C. L., and U. Heinemann. Effects of the triazole derivative loreclezole (R72063) on stimulus induced ionic and field potential responses and on different patterns of epileptiform activity induced by low magnesium in rat entorhinal cortex-hippocampal slices. Naunyn-Schmiedeberg's Arch. Pharmacol. 346:581-587 (1992).
    • (1992) Naunyn-Schmiedeberg's Arch. Pharmacol. , vol.346 , pp. 581-587
    • Zhang, C.L.1    Heinemann, U.2
  • 44
    • 0029417325 scopus 로고
    • A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site
    • A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site. Mol. Pharmacol. 48:965-969 (1995).
    • (1995) Mol. Pharmacol. , vol.48 , pp. 965-969
    • Stevenson, A.1    Wingrove, P.B.2    Whiting, P.J.3    Wafford, K.A.4
  • 45
    • 0028011989 scopus 로고
    • A receptors identify a 67-kDa protein in rat brain membranes
    • A receptors identify a 67-kDa protein in rat brain membranes. J. Neurochem. 62:764-769 (1994).
    • (1994) J. Neurochem. , vol.62 , pp. 764-769
    • Kern, W.1    Sieghart, W.2
  • 47
    • 0030024882 scopus 로고    scopus 로고
    • Cloning of cDNAs encoding the human γ-aminobutyric acid type A receptor α6 subunit and characterization of the pharmacology of α6-containing receptors
    • Hadingham, K. L., E. M. Garrett, K. A. Wafford, C. Bain, R. P. Heavens, J. S. Sirinathsinghji, and P. J. Whiting. Cloning of cDNAs encoding the human γ-aminobutyric acid type A receptor α6 subunit and characterization of the pharmacology of α6-containing receptors. Mol. Pharmacol. 49:253-259 (1996).
    • (1996) Mol. Pharmacol. , vol.49 , pp. 253-259
    • Hadingham, K.L.1    Garrett, E.M.2    Wafford, K.A.3    Bain, C.4    Heavens, R.P.5    Sirinathsinghji, J.S.6    Whiting, P.J.7
  • 48
    • 0028225120 scopus 로고
    • Pharmacologic effects and abuse liability of bretazenil, diazepam, and alprazolam in humans
    • Busto, U., H. L. Kaplan, L. Zawertailo, and E. M. Sellers. Pharmacologic effects and abuse liability of bretazenil, diazepam, and alprazolam in humans. Clin. Pharmacol. Ther. 55:451-463 (1994).
    • (1994) Clin. Pharmacol. Ther. , vol.55 , pp. 451-463
    • Busto, U.1    Kaplan, H.L.2    Zawertailo, L.3    Sellers, E.M.4
  • 49
    • 0027233914 scopus 로고
    • Synthetic and computerassisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors
    • Wong, G., K. F. Koehler, P. Skolnick, Z. Q. Gu, D. Ananthan, P. Schonholzer, W. Hunkeler, W. Zhang, and J. M. Cook. Synthetic and computerassisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors. J. Med. Chem. 36:1820-1830 (1993).
    • (1993) J. Med. Chem. , vol.36 , pp. 1820-1830
    • Wong, G.1    Koehler, K.F.2    Skolnick, P.3    Gu, Z.Q.4    Ananthan, D.5    Schonholzer, P.6    Hunkeler, W.7    Zhang, W.8    Cook, J.M.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.