The third intracellular loop stabilizes the inactive state of the neuropeptide Y1 receptor

Journal of Biological Chemistry

Volumn 283, Issue 48, 2008, Pages 33337-33346

  Chee, Melissa J S ^a   Mörl, Karin ^b   Lindner, Diana ^b   Merten, Nicole ^b   Zamponi, Gerald W ^c   Light, Peter E ^a   Beck Sickinger, Annette G ^b   Colmers, William F ^a  

^a UNIVERSITY OF ALBERTA   (Canada)

^b UNIVERSITY OF LEIPZIG   (Germany)

^c UNIVERSITY OF CALGARY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

ACTIVATION ANALYSIS; BIOCHEMISTRY; ELECTROPHYSIOLOGY; FLOW INTERACTIONS;

BIOCHEMICAL ASSAYS; CHIMERIC PROTEINS; CLASS I; CONSTITUTIVELY ACTIVES; COUPLED RECEPTORS; ELECTROPHYSIOLOGICAL ASSAYS; INTRAMOLECULAR INTERACTIONS; LIGAND BINDINGS; METABOLITE LEVELS; NEUROPEPTIDE; OPIOID RECEPTORS; POINT MUTATIONS; PURINOCEPTORS; RECEPTOR ACTIVATIONS; RECEPTOR ACTIVITIES; STABILIZING INTERACTIONS; THIRD INTRACELLULAR LOOPS; TRANSMEMBRANE DOMAINS;

SIGNAL TRANSDUCTION;

CHIMERIC PROTEIN; GUANINE NUCLEOTIDE BINDING PROTEIN; MU OPIATE RECEPTOR; NEUROPEPTIDE Y1 RECEPTOR; PURINERGIC P2Y12 RECEPTOR;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; ELECTROPHYSIOLOGY; GENE LOCUS; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN EXPRESSION; PROTEIN METABOLISM; RECEPTOR AFFINITY; SIGNAL TRANSDUCTION;

ANIMALS; CERCOPITHECUS AETHIOPS; COS CELLS; GTP-BINDING PROTEIN ALPHA SUBUNITS, GI-GO; GTP-BINDING PROTEIN ALPHA SUBUNITS, GQ-G11; HUMANS; POINT MUTATION; PROTEIN STRUCTURE, SECONDARY; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, NEUROPEPTIDE Y; RECEPTORS, OPIOID, MU; RECEPTORS, PURINERGIC P2; RECOMBINANT FUSION PROTEINS; SIGNAL TRANSDUCTION;

EID: 57749114748     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M804671200     Document Type: Article

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